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Report error Found 21 Enz. Inhib. hit(s) with all data for entry = 6323
TargetGenome polyprotein(Hepacivirus C)
University of Wisconsin-Milwaukee

LigandPNGBDBM61947(6-bromanyl-2-phenyl-1,2-benzothiazol-3-one | 6-bro...)
Affinity DataIC50:  700nMpH: 7.5 T: 23°CAssay Description:Binding assays containing 25 mM MOPS pH 7.5, 1.25 mM MgCl2, 20 nM Cy5-dT15, and 200 nM NS3h_1b were incubated 5 min at RT. Following addition of indi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGenome polyprotein(Hepacivirus C)
University of Wisconsin-Milwaukee

LigandPNGBDBM34233(2-Phenyl-benzo[d]isoselenazol-3-one | 2-Phenyl-ben...)
Affinity DataIC50:  1.40E+3nMpH: 7.5 T: 23°CAssay Description:Binding assays containing 25 mM MOPS pH 7.5, 1.25 mM MgCl2, 20 nM Cy5-dT15, and 200 nM NS3h_1b were incubated 5 min at RT. Following addition of indi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGenome polyprotein(Hepacivirus C)
University of Wisconsin-Milwaukee

LigandPNGBDBM61939(5,6-bis(fluoranyl)-2-phenyl-1,2-benzothiazol-3-one...)
Affinity DataIC50:  1.50E+3nMpH: 7.5 T: 23°CAssay Description:Binding assays containing 25 mM MOPS pH 7.5, 1.25 mM MgCl2, 20 nM Cy5-dT15, and 200 nM NS3h_1b were incubated 5 min at RT. Following addition of indi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGenome polyprotein(Hepacivirus C)
University of Wisconsin-Milwaukee

LigandPNGBDBM46667(2-phenyl-1,2-benzothiazol-3-one | 2-phenyl-1,2-ben...)
Affinity DataIC50:  1.90E+3nMpH: 7.5 T: 23°CAssay Description:Binding assays containing 25 mM MOPS pH 7.5, 1.25 mM MgCl2, 20 nM Cy5-dT15, and 200 nM NS3h_1b were incubated 5 min at RT. Following addition of indi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGenome polyprotein(Hepacivirus C)
University of Wisconsin-Milwaukee

LigandPNGBDBM61966(KSC-09-149B | KUC105615N | N-(2-chlorophenyl)-2-(3...)
Affinity DataIC50:  1.90E+3nMpH: 7.5 T: 23°CAssay Description:Binding assays containing 25 mM MOPS pH 7.5, 1.25 mM MgCl2, 20 nM Cy5-dT15, and 200 nM NS3h_1b were incubated 5 min at RT. Following addition of indi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGenome polyprotein(Hepacivirus C)
University of Wisconsin-Milwaukee

LigandPNGBDBM61969(KSC-09-140B | KUC105618N | N-(2-bromophenyl)-2-(3-...)
Affinity DataIC50:  2.00E+3nMpH: 7.5 T: 23°CAssay Description:Binding assays containing 25 mM MOPS pH 7.5, 1.25 mM MgCl2, 20 nM Cy5-dT15, and 200 nM NS3h_1b were incubated 5 min at RT. Following addition of indi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGenome polyprotein(Hepacivirus C)
University of Wisconsin-Milwaukee

LigandPNGBDBM61942(2-(3-keto-1,2-benzothiazol-2-yl)-N-(o-tolyl)acetam...)
Affinity DataIC50:  3.90E+3nMpH: 7.5 T: 23°CAssay Description:Binding assays containing 25 mM MOPS pH 7.5, 1.25 mM MgCl2, 20 nM Cy5-dT15, and 200 nM NS3h_1b were incubated 5 min at RT. Following addition of indi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGenome polyprotein(Hepacivirus C)
University of Wisconsin-Milwaukee

LigandPNGBDBM61965(KSC-09-149A | KUC105614N | N-(2-fluorophenyl)-2-(3...)
Affinity DataIC50:  5.60E+3nMpH: 7.5 T: 23°CAssay Description:Binding assays containing 25 mM MOPS pH 7.5, 1.25 mM MgCl2, 20 nM Cy5-dT15, and 200 nM NS3h_1b were incubated 5 min at RT. Following addition of indi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGenome polyprotein(Hepacivirus C)
University of Wisconsin-Milwaukee

LigandPNGBDBM61942(2-(3-keto-1,2-benzothiazol-2-yl)-N-(o-tolyl)acetam...)
Affinity DataIC50:  5.60E+3nMpH: 7.5 T: 23°CAssay Description:Binding assays containing 25 mM MOPS pH 7.5, 1.25 mM MgCl2, 20 nM Cy5-dT15, and 200 nM NS3h_1b were incubated 5 min at RT. Following addition of indi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGenome polyprotein(Hepacivirus C)
University of Wisconsin-Milwaukee

LigandPNGBDBM61964(2-(3-keto-1,2-benzothiazol-2-yl)-N-phenyl-propiona...)
Affinity DataIC50:  6.30E+3nMpH: 7.5 T: 23°CAssay Description:Binding assays containing 25 mM MOPS pH 7.5, 1.25 mM MgCl2, 20 nM Cy5-dT15, and 200 nM NS3h_1b were incubated 5 min at RT. Following addition of indi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGenome polyprotein(Hepacivirus C)
University of Wisconsin-Milwaukee

LigandPNGBDBM61970(KSC-09-140C | KUC105619N | N-(2-iodanylphenyl)-2-(...)
Affinity DataIC50:  7.80E+3nMpH: 7.5 T: 23°CAssay Description:Binding assays containing 25 mM MOPS pH 7.5, 1.25 mM MgCl2, 20 nM Cy5-dT15, and 200 nM NS3h_1b were incubated 5 min at RT. Following addition of indi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGenome polyprotein(Hepacivirus C)
University of Wisconsin-Milwaukee

LigandPNGBDBM61949(KSC-4-295 | KUC105342N | N-(3-bromophenyl)-2-(3-ke...)
Affinity DataIC50:  1.20E+4nMpH: 7.5 T: 23°CAssay Description:Binding assays containing 25 mM MOPS pH 7.5, 1.25 mM MgCl2, 20 nM Cy5-dT15, and 200 nM NS3h_1b were incubated 5 min at RT. Following addition of indi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGenome polyprotein(Hepacivirus C)
University of Wisconsin-Milwaukee

LigandPNGBDBM61957(3-(3-keto-1,2-benzothiazol-2-yl)-N-phenyl-propiona...)
Affinity DataIC50:  1.50E+4nMpH: 7.5 T: 23°CAssay Description:Binding assays containing 25 mM MOPS pH 7.5, 1.25 mM MgCl2, 20 nM Cy5-dT15, and 200 nM NS3h_1b were incubated 5 min at RT. Following addition of indi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetGenome polyprotein(Hepacivirus C)
University of Wisconsin-Milwaukee

LigandPNGBDBM123128(1‐(4‐bromo‐2‐nitrophenyl)p...)
Affinity DataIC50:  2.20E+4nMpH: 7.5 T: 23°CAssay Description:Binding assays containing 25 mM MOPS pH 7.5, 1.25 mM MgCl2, 20 nM Cy5-dT15, and 200 nM NS3h_1b were incubated 5 min at RT. Following addition of indi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGenome polyprotein(Hepacivirus C)
University of Wisconsin-Milwaukee

LigandPNGBDBM123129(1-(3-nitro-phenyl)-pyrrole-2,5-dione (17) | CID236...)
Affinity DataIC50:  2.30E+4nMpH: 7.5 T: 23°CAssay Description:Binding assays containing 25 mM MOPS pH 7.5, 1.25 mM MgCl2, 20 nM Cy5-dT15, and 200 nM NS3h_1b were incubated 5 min at RT. Following addition of indi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGenome polyprotein(Hepacivirus C)
University of Wisconsin-Milwaukee

LigandPNGBDBM61961(2-(3-keto-1,2-benzothiazol-2-yl)-N-[2-(trifluorome...)
Affinity DataIC50:  2.80E+4nMpH: 7.5 T: 23°CAssay Description:Binding assays containing 25 mM MOPS pH 7.5, 1.25 mM MgCl2, 20 nM Cy5-dT15, and 200 nM NS3h_1b were incubated 5 min at RT. Following addition of indi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGenome polyprotein(Hepacivirus C)
University of Wisconsin-Milwaukee

LigandPNGBDBM123130(1-(2-bromo-4-methylphenyl)-1H-pyrrole-2,5-dione (1...)
Affinity DataIC50:  3.30E+4nMpH: 7.5 T: 23°CAssay Description:Binding assays containing 25 mM MOPS pH 7.5, 1.25 mM MgCl2, 20 nM Cy5-dT15, and 200 nM NS3h_1b were incubated 5 min at RT. Following addition of indi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGenome polyprotein(Hepacivirus C)
University of Wisconsin-Milwaukee

LigandPNGBDBM50247587(2,5-diphenylisothiazol-3(2H)-one | CHEMBL500224 | ...)
Affinity DataIC50: >1.00E+5nMpH: 7.5 T: 23°CAssay Description:Binding assays containing 25 mM MOPS pH 7.5, 1.25 mM MgCl2, 20 nM Cy5-dT15, and 200 nM NS3h_1b were incubated 5 min at RT. Following addition of indi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGenome polyprotein(Hepacivirus C)
University of Wisconsin-Milwaukee

LigandPNGBDBM61938(1-methyl-2-phenyl-3-indazolone | 1-methyl-2-phenyl...)
Affinity DataIC50: >1.00E+5nMpH: 7.5 T: 23°CAssay Description:Binding assays containing 25 mM MOPS pH 7.5, 1.25 mM MgCl2, 20 nM Cy5-dT15, and 200 nM NS3h_1b were incubated 5 min at RT. Following addition of indi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGenome polyprotein(Hepacivirus C)
University of Wisconsin-Milwaukee

LigandPNGBDBM50220832(CHEMBL8211 | N-ethylmaleimide)
Affinity DataIC50:  5.30E+5nMpH: 7.5 T: 23°CAssay Description:Binding assays containing 25 mM MOPS pH 7.5, 1.25 mM MgCl2, 20 nM Cy5-dT15, and 200 nM NS3h_1b were incubated 5 min at RT. Following addition of indi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGenome polyprotein(Hepacivirus C)
University of Wisconsin-Milwaukee

LigandPNGBDBM50376514(IODOACETAMIDE)
Affinity DataIC50:  2.00E+6nMpH: 7.5 T: 23°CAssay Description:Binding assays containing 25 mM MOPS pH 7.5, 1.25 mM MgCl2, 20 nM Cy5-dT15, and 200 nM NS3h_1b were incubated 5 min at RT. Following addition of indi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed