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Found 14 Enz. Inhib. hit(s) with all data for entry = 50044661
TargetProteinase-activated receptor 4(Homo sapiens (Human))
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM50024253(CHEMBL3334887)
Affinity DataIC50:  66nMAssay Description:Antagonist activity at PAR4 in PAR-4-AP-stimulated human platelets compound pretreated for 5 mins by fluorescent PAC1 integrin alpha2bb3 activation a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM50024254(CHEMBL125021)
Affinity DataIC50:  130nMAssay Description:Antagonist activity at PAR4 in PAR-4-AP-stimulated human platelets compound pretreated for 5 mins by fluorescent PAC1 integrin alpha2bb3 activation a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM50024252(CHEMBL1609104)
Affinity DataIC50:  140nMAssay Description:Antagonist activity at PAR4 in PAR-4-AP-stimulated human platelets compound pretreated for 5 mins by fluorescent PAC1 integrin alpha2bb3 activation a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM50024255(CHEMBL3334944)
Affinity DataIC50:  279nMAssay Description:Antagonist activity at PAR4 in PAR-4-AP-stimulated human platelets compound pretreated for 5 mins by fluorescent PAC1 integrin alpha2bb3 activation a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM50024258(CHEMBL3334941)
Affinity DataIC50:  336nMAssay Description:Antagonist activity at PAR4 in PAR-4-AP-stimulated human platelets compound pretreated for 5 mins by fluorescent PAC1 integrin alpha2bb3 activation a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM50024259(CHEMBL3334940)
Affinity DataIC50:  646nMAssay Description:Antagonist activity at PAR4 in PAR-4-AP-stimulated human platelets compound pretreated for 5 mins by fluorescent PAC1 integrin alpha2bb3 activation a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM50024260(CHEMBL3334939)
Affinity DataIC50:  785nMAssay Description:Antagonist activity at PAR4 in PAR-4-AP-stimulated human platelets compound pretreated for 5 mins by fluorescent PAC1 integrin alpha2bb3 activation a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM50024257(CHEMBL3334942)
Affinity DataIC50:  793nMAssay Description:Antagonist activity at PAR4 in PAR-4-AP-stimulated human platelets compound pretreated for 5 mins by fluorescent PAC1 integrin alpha2bb3 activation a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM50024256(CHEMBL3334943)
Affinity DataIC50:  5.13E+3nMAssay Description:Antagonist activity at PAR4 in PAR-4-AP-stimulated human platelets compound pretreated for 5 mins by fluorescent PAC1 integrin alpha2bb3 activation a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM50024261(CHEMBL3334901)
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at PAR4 in PAR-4-AP-stimulated human platelets compound pretreated for 5 mins by fluorescent PAC1 integrin alpha2bb3 activation a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM50024252(CHEMBL1609104)
Affinity DataIC50:  1.00E+4nMAssay Description:Antagonist activity at PAR1 in PAR-1-AP-stimulated human platelets compound pretreated for 5 mins by fluorescent PAC1 integrin alpha2bb3 activation a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM50024253(CHEMBL3334887)
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at PAR1 in PAR-1-AP-stimulated human platelets compound pretreated for 5 mins by fluorescent PAC1 integrin alpha2bb3 activation a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM50024262(CHEMBL3334933)
Affinity DataIC50:  1.00E+4nMAssay Description:Antagonist activity at PAR4 in PAR-4-AP-stimulated human platelets compound pretreated for 5 mins by fluorescent PAC1 integrin alpha2bb3 activation a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM50024254(CHEMBL125021)
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at PAR1 in PAR-1-AP-stimulated human platelets compound pretreated for 5 mins by fluorescent PAC1 integrin alpha2bb3 activation a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed