Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50044689
TargetAcetylcholinesterase(Rat)
Hunan University

Curated by ChEMBL
LigandPNGBDBM50026058(CHEMBL3335259)
Affinity DataKi:  2.75E+3nMAssay Description:Inhibition of Sprague-Dawley rat brain AChE by Michaelis-Menten equationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetAcetylcholinesterase(Rat)
Hunan University

Curated by ChEMBL
LigandPNGBDBM50026058(CHEMBL3335259)
Affinity DataIC50: 4.15E+3nMAssay Description:Inhibition of Sprague-Dawley rat brain AChE using acetylthiocholin iodide as substrate preincubated for 25 mins by Ellman's/UV-vis spectroscopy analy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetAcetylcholinesterase(Rat)
Hunan University

Curated by ChEMBL
LigandPNGBDBM50026058(CHEMBL3335259)
Affinity DataKi:  4.58E+3nMAssay Description:Inhibition of Sprague-Dawley rat brain AChE using acetylthiocholin iodide as substrate by Michaelis-Menten equationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetAcetylcholinesterase(Rat)
Hunan University

Curated by ChEMBL
LigandPNGBDBM10620(3-[(1S)-1-(dimethylamino)ethyl]phenyl N-ethyl-N-me...)
Affinity DataIC50: 1.05E+4nMAssay Description:Inhibition of Sprague-Dawley rat brain AChE using acetylthiocholin iodide as substrate preincubated for 25 mins by Ellman's/UV-vis spectroscopy analy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetAcetylcholinesterase(Rat)
Hunan University

Curated by ChEMBL
LigandPNGBDBM50026061(CHEMBL3335261)
Affinity DataIC50: 1.24E+4nMAssay Description:Inhibition of Sprague-Dawley rat brain AChE using acetylthiocholin iodide as substrate preincubated for 25 mins by Ellman's/UV-vis spectroscopy analy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetAcetylcholinesterase(Rat)
Hunan University

Curated by ChEMBL
LigandPNGBDBM50026062(CHEMBL3335256)
Affinity DataIC50: 1.51E+4nMAssay Description:Inhibition of Sprague-Dawley rat brain AChE using acetylthiocholin iodide as substrate preincubated for 25 mins by Ellman's/UV-vis spectroscopy analy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetAcetylcholinesterase(Rat)
Hunan University

Curated by ChEMBL
LigandPNGBDBM50026064(CHEMBL3335258)
Affinity DataIC50: 1.61E+4nMAssay Description:Inhibition of Sprague-Dawley rat brain AChE using acetylthiocholin iodide as substrate preincubated for 25 mins by Ellman's/UV-vis spectroscopy analy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetAcetylcholinesterase(Rat)
Hunan University

Curated by ChEMBL
LigandPNGBDBM50026065(CHEMBL3335255)
Affinity DataIC50: 1.88E+4nMAssay Description:Inhibition of Sprague-Dawley rat brain AChE using acetylthiocholin iodide as substrate preincubated for 25 mins by Ellman's/UV-vis spectroscopy analy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetAcetylcholinesterase(Rat)
Hunan University

Curated by ChEMBL
LigandPNGBDBM50026063(CHEMBL3335257)
Affinity DataIC50: 5.48E+4nMAssay Description:Inhibition of Sprague-Dawley rat brain AChE using acetylthiocholin iodide as substrate preincubated for 25 mins by Ellman's/UV-vis spectroscopy analy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetAcetylcholinesterase(Rat)
Hunan University

Curated by ChEMBL
LigandPNGBDBM50026060(CHEMBL3335260)
Affinity DataIC50: 2.65E+5nMAssay Description:Inhibition of Sprague-Dawley rat brain AChE using acetylthiocholin iodide as substrate preincubated for 25 mins by Ellman's/UV-vis spectroscopy analy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed