Compile Data Set for Download or QSAR
maximum 50k data
Found 6 Enz. Inhib. hit(s) with all data for entry = 6345
TargetEukaryotic elongation factor 2 kinase(Homo sapiens (Human))
The University of Texas At Austin

LigandPNGBDBM123834(4-(3-methoxyphenyl)-2,6-dioxo-3,5-piperidinedicarb...)
Affinity DataIC50:  2.50E+4nMAssay Description:WT eEF-2K (2 nM) was preincubated with various concentrations of inhibitors (0-1000 uM) in assay buffer containing CaCl2 (150 uM), calmodulin (1 uM),...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEukaryotic elongation factor 2 kinase(Homo sapiens (Human))
The University of Texas At Austin

LigandPNGBDBM123836(4-(3,4-dichlorophenyl)-2,6-dioxopiperidine-3,5-dic...)
Affinity DataIC50:  3.00E+4nMAssay Description:WT eEF-2K (2 nM) was preincubated with various concentrations of inhibitors (0-1000 uM) in assay buffer containing CaCl2 (150 uM), calmodulin (1 uM),...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEukaryotic elongation factor 2 kinase(Homo sapiens (Human))
The University of Texas At Austin

LigandPNGBDBM123835(4‐(2‐methylphenyl)‐2,6‐dio...)
Affinity DataIC50:  3.30E+4nMAssay Description:WT eEF-2K (2 nM) was preincubated with various concentrations of inhibitors (0-1000 uM) in assay buffer containing CaCl2 (150 uM), calmodulin (1 uM),...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEukaryotic elongation factor 2 kinase(Homo sapiens (Human))
The University of Texas At Austin

LigandPNGBDBM123837(4‐(4‐methylphenyl)‐2,6‐dio...)
Affinity DataIC50:  4.60E+4nMAssay Description:WT eEF-2K (2 nM) was preincubated with various concentrations of inhibitors (0-1000 uM) in assay buffer containing CaCl2 (150 uM), calmodulin (1 uM),...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEukaryotic elongation factor 2 kinase(Homo sapiens (Human))
The University of Texas At Austin

LigandPNGBDBM123839(4‐(2,6‐dichlorophenyl)‐2,6‐...)
Affinity DataIC50:  5.70E+4nMAssay Description:WT eEF-2K (2 nM) was preincubated with various concentrations of inhibitors (0-1000 uM) in assay buffer containing CaCl2 (150 uM), calmodulin (1 uM),...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEukaryotic elongation factor 2 kinase(Homo sapiens (Human))
The University of Texas At Austin

LigandPNGBDBM123838(4‐(3‐hydroxyphenyl)‐2,6‐di...)
Affinity DataIC50:  6.60E+4nMAssay Description:WT eEF-2K (2 nM) was preincubated with various concentrations of inhibitors (0-1000 uM) in assay buffer containing CaCl2 (150 uM), calmodulin (1 uM),...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed