Compile Data Set for Download or QSAR
Report error Found 30 Enz. Inhib. hit(s) with all data for entry = 50044734
TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50052524((S)-N-((S)-1-{[(S)-1-({[(S)-1-((S)-1-Carbamoyl-3-m...)
Affinity DataEC50:  11nMAssay Description:Agonist activity at human NK3R expressed in CHO cells assessed as potentiation of senktide-induced effectMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2016
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50299467((5S,8S,14S,17S,20S,23S,26S,29S,32S)-26-((1H-imidaz...)
Affinity DataIC50: 12nMAssay Description:Displacement of [125I]His3, MePhe7 from human NK3R expressed in CHO cell membranes by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2016
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Rat)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50052524((S)-N-((S)-1-{[(S)-1-({[(S)-1-((S)-1-Carbamoyl-3-m...)
Affinity DataEC50:  13nMAssay Description:Agonist activity at rat NK3RMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2016
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50028021(CHEMBL3361404)
Affinity DataEC50:  16nMAssay Description:Agonist activity at human NK3R expressed in CHO cells assessed as potentiation of senktide-induced effectMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2016
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Rat)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50028021(CHEMBL3361404)
Affinity DataEC50:  19nMAssay Description:Agonist activity at rat NK3RMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2016
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50028014(CHEMBL3361397)
Affinity DataIC50: 22nMAssay Description:Displacement of [125I]His3, MePhe7 from human NK3R expressed in CHO cell membranes by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2016
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50028015(CHEMBL3361398)
Affinity DataIC50: 43nMAssay Description:Displacement of [125I]His3, MePhe7 from human NK3R expressed in CHO cell membranes by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2016
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50052524((S)-N-((S)-1-{[(S)-1-({[(S)-1-((S)-1-Carbamoyl-3-m...)
Affinity DataIC50: 56nMAssay Description:Displacement of [125I]His3, MePhe7 from human NK3R expressed in CHO cell membranes by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2016
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50028021(CHEMBL3361404)
Affinity DataIC50: 56nMAssay Description:Displacement of [125I]His3, MePhe7 from human NK3R expressed in CHO cell membranes by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2016
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50028016(CHEMBL3361399)
Affinity DataIC50: 59nMAssay Description:Displacement of [125I]His3, MePhe7 from human NK3R expressed in CHO cell membranes by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2016
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50299467((5S,8S,14S,17S,20S,23S,26S,29S,32S)-26-((1H-imidaz...)
Affinity DataEC50:  64nMAssay Description:Agonist activity at human NK3R expressed in CHO cells assessed as induction of Ca2+ influx by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2016
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50028016(CHEMBL3361399)
Affinity DataEC50:  91nMAssay Description:Agonist activity at human NK3R expressed in CHO cells assessed as induction of Ca2+ influx by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2016
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50028025(CHEMBL3361408)
Affinity DataEC50:  100nMAssay Description:Agonist activity at human NK3R expressed in CHO cells assessed as potentiation of senktide-induced effectMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2016
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50028017(CHEMBL3361400)
Affinity DataEC50:  240nMAssay Description:Agonist activity at human NK3R expressed in CHO cells assessed as induction of Ca2+ influx by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2016
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50028015(CHEMBL3361398)
Affinity DataEC50:  280nMAssay Description:Agonist activity at human NK3R expressed in CHO cells assessed as induction of Ca2+ influx by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2016
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50028014(CHEMBL3361397)
Affinity DataEC50:  330nMAssay Description:Agonist activity at human NK3R expressed in CHO cells assessed as induction of Ca2+ influx by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2016
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50028018(CHEMBL3361401)
Affinity DataEC50:  350nMAssay Description:Agonist activity at human NK3R expressed in CHO cells assessed as induction of Ca2+ influx by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2016
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50028025(CHEMBL3361408)
Affinity DataIC50: 360nMAssay Description:Displacement of [125I]His3, MePhe7 from human NK3R expressed in CHO cell membranes by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2016
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50028024(CHEMBL3361407)
Affinity DataEC50:  370nMAssay Description:Agonist activity at human NK3R expressed in CHO cells assessed as potentiation of senktide-induced effectMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2016
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50028022(CHEMBL3361405)
Affinity DataEC50:  920nMAssay Description:Agonist activity at human NK3R expressed in CHO cells assessed as potentiation of senktide-induced effectMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2016
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50028024(CHEMBL3361407)
Affinity DataIC50: 1.10E+3nMAssay Description:Displacement of [125I]His3, MePhe7 from human NK3R expressed in CHO cell membranes by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2016
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50028023(CHEMBL3361406)
Affinity DataEC50:  1.90E+3nMAssay Description:Agonist activity at human NK3R expressed in CHO cells assessed as potentiation of senktide-induced effectMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2016
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50028018(CHEMBL3361401)
Affinity DataIC50: 2.30E+3nMAssay Description:Displacement of [125I]His3, MePhe7 from human NK3R expressed in CHO cell membranes by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2016
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50028017(CHEMBL3361400)
Affinity DataIC50: 2.90E+3nMAssay Description:Displacement of [125I]His3, MePhe7 from human NK3R expressed in CHO cell membranes by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2016
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50028023(CHEMBL3361406)
Affinity DataIC50: 1.30E+4nMAssay Description:Displacement of [125I]His3, MePhe7 from human NK3R expressed in CHO cell membranes by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2016
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50028022(CHEMBL3361405)
Affinity DataIC50: 1.90E+4nMAssay Description:Displacement of [125I]His3, MePhe7 from human NK3R expressed in CHO cell membranes by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2016
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50028019(CHEMBL3361402)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human NK3R expressed in CHO cells assessed as induction of Ca2+ influx by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2016
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50028020(CHEMBL3361403)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human NK3R expressed in CHO cells assessed as induction of Ca2+ influx by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2016
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50028019(CHEMBL3361402)
Affinity DataIC50: 1.00E+7nMAssay Description:Displacement of [125I]His3, MePhe7 from human NK3R expressed in CHO cell membranes by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2016
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50028020(CHEMBL3361403)
Affinity DataIC50: 1.00E+7nMAssay Description:Displacement of [125I]His3, MePhe7 from human NK3R expressed in CHO cell membranes by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2016
Entry Details Article
PubMed