Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 50044735
TargetG-protein coupled bile acid receptor 1(Human)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50028027(CHEMBL3342086)
Affinity DataEC50:  400nMAssay Description:Agonist activity at GP-BAR1 (unknown origin) in human HEK293 cells assessed as receptor transactivation at 100 nM to 50 uM incubated for 16 hrs by CR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2016
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50028028(CHEMBL3342082)
Affinity DataEC50:  1.03E+3nMAssay Description:Agonist activity at GP-BAR1 (unknown origin) in human HEK293 cells assessed as receptor transactivation at 100 nM to 50 uM incubated for 16 hrs by CR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2016
Entry Details Article
PubMed
TargetBile acid receptor(Human)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50028027(CHEMBL3342086)
Affinity DataEC50:  2.00E+3nMAssay Description:Agonist activity at FXR (unknown origin) expressed in human HepG2 cells assessed as receptor transactivation at 100 nM to 50 uM incubated for 16 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2016
Entry Details Article
PubMed
TargetBile acid receptor(Human)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50028026(CHEMBL3342065)
Affinity DataEC50:  9.00E+3nMAssay Description:Agonist activity at FXR (unknown origin) expressed in human HepG2 cells assessed as receptor transactivation at 100 nM to 50 uM incubated for 16 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2016
Entry Details Article
PubMed