Compile Data Set for Download or QSAR
maximum 50k data
Found 4 Enz. Inhib. hit(s) with all data for entry = 50044735
TargetBile acid receptor(Homo sapiens (Human))
University Of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50028026(CHEMBL3342065)
Affinity DataEC50:  9.00E+3nMAssay Description:Agonist activity at FXR (unknown origin) expressed in human HepG2 cells assessed as receptor transactivation at 100 nM to 50 uM incubated for 16 hrs ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
University Of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50028027(CHEMBL3342086)
Affinity DataEC50:  400nMAssay Description:Agonist activity at GP-BAR1 (unknown origin) in human HEK293 cells assessed as receptor transactivation at 100 nM to 50 uM incubated for 16 hrs by CR...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
University Of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50028028(CHEMBL3342082)
Affinity DataEC50:  1.03E+3nMAssay Description:Agonist activity at GP-BAR1 (unknown origin) in human HEK293 cells assessed as receptor transactivation at 100 nM to 50 uM incubated for 16 hrs by CR...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBile acid receptor(Homo sapiens (Human))
University Of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50028027(CHEMBL3342086)
Affinity DataEC50:  2.00E+3nMAssay Description:Agonist activity at FXR (unknown origin) expressed in human HepG2 cells assessed as receptor transactivation at 100 nM to 50 uM incubated for 16 hrs ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed