Compile Data Set for Download or QSAR
maximum 50k data
Found 41 Enz. Inhib. hit(s) with all data for entry = 50044762
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50028990(CHEMBL3339169)
Affinity DataIC50:  3nMAssay Description:Inhibition of human 11-betaHSD1 by biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50028997(CHEMBL3339176)
Affinity DataIC50:  5nMAssay Description:Inhibition of human 11-betaHSD1 by biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50028991(CHEMBL3339170)
Affinity DataIC50:  9nMAssay Description:Inhibition of human 11-betaHSD1 by biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50028989(CHEMBL3339168)
Affinity DataIC50:  9nMAssay Description:Inhibition of human 11-betaHSD1 by biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM32518(pyridine amide, 9)
Affinity DataIC50:  17nMAssay Description:Inhibition of human 11-betaHSD1 by biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50028992(CHEMBL3339171)
Affinity DataIC50:  20nMAssay Description:Inhibition of human 11-betaHSD1 by biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50028996(CHEMBL3339175)
Affinity DataIC50:  30nMAssay Description:Inhibition of human 11-betaHSD1 by biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM32499(pyridine amide, 8)
Affinity DataIC50:  46nMAssay Description:Inhibition of human 11-betaHSD1 by biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50028998(CHEMBL3339177)
Affinity DataIC50:  47nMAssay Description:Inhibition of human 11-betaHSD1 by biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50028983(CHEMBL3339161)
Affinity DataIC50:  49nMAssay Description:Inhibition of human 11-betaHSD1 by biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50028982(CHEMBL3339160)
Affinity DataIC50:  52nMAssay Description:Inhibition of human 11-betaHSD1 by biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50028977(CHEMBL3339159)
Affinity DataIC50:  55nMAssay Description:Inhibition of human 11-betaHSD1 by biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50028985(CHEMBL3339163)
Affinity DataIC50:  79nMAssay Description:Inhibition of human 11-betaHSD1 by biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50028986(CHEMBL3339164)
Affinity DataIC50:  92nMAssay Description:Inhibition of human 11-betaHSD1 by biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50028999(CHEMBL3339178)
Affinity DataIC50:  110nMAssay Description:Inhibition of human 11-betaHSD1 by biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50028987(CHEMBL3339165)
Affinity DataIC50:  120nMAssay Description:Inhibition of human 11-betaHSD1 by biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50028984(CHEMBL3339162)
Affinity DataIC50:  120nMAssay Description:Inhibition of human 11-betaHSD1 by biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50029013(CHEMBL3337473)
Affinity DataIC50:  160nMAssay Description:Inhibition of human 11-betaHSD1 by biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50028973(CHEMBL260370)
Affinity DataIC50:  160nMAssay Description:Inhibition of human 11-betaHSD1 by biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50028988(CHEMBL3339167)
Affinity DataIC50:  180nMAssay Description:Inhibition of human 11-betaHSD1 by biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50029008(CHEMBL3339188)
Affinity DataIC50:  180nMAssay Description:Inhibition of human 11-betaHSD1 by biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50029008(CHEMBL3339188)
Affinity DataIC50:  180nMAssay Description:Inhibition of human 11-betaHSD1 by biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50029002(CHEMBL3339182)
Affinity DataIC50:  220nMAssay Description:Inhibition of human 11-betaHSD1 by biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50029009(CHEMBL3339189)
Affinity DataIC50:  220nMAssay Description:Inhibition of human 11-betaHSD1 by biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50028975(CHEMBL3339158)
Affinity DataIC50:  310nMAssay Description:Inhibition of human 11-betaHSD1 by biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50029003(CHEMBL3339183)
Affinity DataIC50:  320nMAssay Description:Inhibition of human 11-betaHSD1 by biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50029011(CHEMBL3339191)
Affinity DataIC50:  320nMAssay Description:Inhibition of human 11-betaHSD1 by biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50029012(CHEMBL3339192)
Affinity DataIC50:  430nMAssay Description:Inhibition of human 11-betaHSD1 by biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50028974(CHEMBL3339157)
Affinity DataIC50:  720nMAssay Description:Inhibition of human 11-betaHSD1 by biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50028994(CHEMBL3339173)
Affinity DataIC50:  980nMAssay Description:Inhibition of human 11-betaHSD1 by biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50029010(CHEMBL3339190)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of human 11-betaHSD1 by biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50029005(CHEMBL3339185)
Affinity DataIC50:  2.60E+3nMAssay Description:Inhibition of human 11-betaHSD1 by biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50029004(CHEMBL3339184)
Affinity DataIC50:  5.80E+3nMAssay Description:Inhibition of human 11-betaHSD1 by biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50028995(CHEMBL3339174)
Affinity DataIC50:  1.10E+4nMAssay Description:Inhibition of human 11-betaHSD1 by biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50029007(CHEMBL3339187)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibition of human 11-betaHSD1 by biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50029001(CHEMBL3339180)
Affinity DataIC50:  1.60E+4nMAssay Description:Inhibition of human 11-betaHSD1 by biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50028993(CHEMBL3339172)
Affinity DataIC50:  1.80E+4nMAssay Description:Inhibition of human 11-betaHSD1 by biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50029015(CHEMBL3339194)
Affinity DataIC50:  2.10E+4nMAssay Description:Inhibition of human 11-betaHSD1 by biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50029014(CHEMBL3339193)
Affinity DataIC50:  2.10E+4nMAssay Description:Inhibition of human 11-betaHSD1 by biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50029006(CHEMBL3339186)
Affinity DataIC50:  2.50E+4nMAssay Description:Inhibition of human 11-betaHSD1 by biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50029000(CHEMBL3339179)
Affinity DataIC50:  2.60E+4nMAssay Description:Inhibition of human 11-betaHSD1 by biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed