Compile Data Set for Download or QSAR
maximum 50k data
Found 57 Enz. Inhib. hit(s) with all data for entry = 6829
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Universiti Kebangsaan Malaysia, Jalan Raja Muda Abdul Aziz

LigandPNGBDBM17638(2-{1-[(4-chlorophenyl)carbonyl]-5-methoxy-2-methyl...)
Affinity DataIC50:  220nMpH: 8.0 T: 2°CAssay Description:100 mM Tris澦Cl buffer, pH 8.0 containing 1 然 heme and COX-1 (ovine) or COX-2(human recombinant), which was preincubated for 10 min in a water bath ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Universiti Kebangsaan Malaysia, Jalan Raja Muda Abdul Aziz

LigandPNGBDBM153295(3-(2,3-Dihydro-benzo[1,4]dioxin-6-yl)-5-(4-dimethy...)
Affinity DataIC50:  440nMpH: 8.0 T: 2°CAssay Description:100 mM Tris澦Cl buffer, pH 8.0 containing 1 然 heme and COX-1 (ovine) or COX-2(human recombinant), which was preincubated for 10 min in a water bath ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2 group V(Homo sapiens (Human))
Universiti Kebangsaan Malaysia, Jalan Raja Muda Abdul Aziz

LigandPNGBDBM18207((1R,2S,10S,11S,13R,14R,15S,17S)-1-fluoro-14,17-dih...)
Affinity DataIC50:  620nMpH: 7.5 T: 2°CAssay Description:Briefly, sn-2ester bond of the substrate 1,2-bis(heptanoylthio)-glycerophosphocholine was hydrolyzed by PLA2-V followed by the exposure of free thiol...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Universiti Kebangsaan Malaysia, Jalan Raja Muda Abdul Aziz

LigandPNGBDBM153297(3-(2,3-Dihydro-benzo[1,4]dioxin-6-yl)-5-(4,7- dime...)
Affinity DataIC50:  940nMpH: 8.0 T: 2°CAssay Description:100 mM Tris澦Cl buffer, pH 8.0 containing 1 然 heme and COX-1 (ovine) or COX-2(human recombinant), which was preincubated for 10 min in a water bath ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Universiti Kebangsaan Malaysia, Jalan Raja Muda Abdul Aziz

LigandPNGBDBM153294(3-Benzofuran-2-yl-5-(2,3-dimethoxy-naphthalen-1-yl...)
Affinity DataIC50:  990nMpH: 8.0 T: 2°CAssay Description:100 mM Tris澦Cl buffer, pH 8.0 containing 1 然 heme and COX-1 (ovine) or COX-2(human recombinant), which was preincubated for 10 min in a water bath ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Universiti Kebangsaan Malaysia, Jalan Raja Muda Abdul Aziz

LigandPNGBDBM153289(3-(2,3-Dihydro-benzo[1,4]dioxin-6-yl)-5-(4-dimethy...)
Affinity DataIC50:  1.12E+3nMpH: 8.0 T: 2°CAssay Description:100 mM Tris澦Cl buffer, pH 8.0 containing 1 然 heme and COX-1 (ovine) or COX-2(human recombinant), which was preincubated for 10 min in a water bath ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Universiti Kebangsaan Malaysia, Jalan Raja Muda Abdul Aziz

LigandPNGBDBM153296(3-(2,3-Dihydro-benzo[1,4]dioxin-6-yl)-5-(2,3-dimet...)
Affinity DataIC50:  1.17E+3nMpH: 8.0 T: 2°CAssay Description:100 mM Tris澦Cl buffer, pH 8.0 containing 1 然 heme and COX-1 (ovine) or COX-2(human recombinant), which was preincubated for 10 min in a water bath ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Universiti Kebangsaan Malaysia, Jalan Raja Muda Abdul Aziz

LigandPNGBDBM153292(3-Benzofuran-2-yl-5-(4-dimethylamino-naphthalen-1-...)
Affinity DataIC50:  1.87E+3nMpH: 8.0 T: 2°CAssay Description:100 mM Tris澦Cl buffer, pH 8.0 containing 1 然 heme and COX-1 (ovine) or COX-2(human recombinant), which was preincubated for 10 min in a water bath ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Universiti Kebangsaan Malaysia, Jalan Raja Muda Abdul Aziz

LigandPNGBDBM153293(3-Benzofuran-2-yl-5-(4,7-dimethoxy-naphthalen-1-yl...)
Affinity DataIC50:  2.14E+3nMpH: 8.0 T: 2°CAssay Description:100 mM Tris澦Cl buffer, pH 8.0 containing 1 然 heme and COX-1 (ovine) or COX-2(human recombinant), which was preincubated for 10 min in a water bath ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Universiti Kebangsaan Malaysia, Jalan Raja Muda Abdul Aziz

LigandPNGBDBM153291(3-(2,3-Dihydro-benzo[1,4]dioxin-6-yl)-5-(4,7- dime...)
Affinity DataIC50:  2.82E+3nMpH: 8.0 T: 2°CAssay Description:100 mM Tris澦Cl buffer, pH 8.0 containing 1 然 heme and COX-1 (ovine) or COX-2(human recombinant), which was preincubated for 10 min in a water bath ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Universiti Kebangsaan Malaysia, Jalan Raja Muda Abdul Aziz

LigandPNGBDBM153290(3-(2,3-Dihydro-benzo[1,4]dioxin-6-yl)-5-(2,3-dimet...)
Affinity DataIC50:  3.42E+3nMpH: 8.0 T: 2°CAssay Description:100 mM Tris澦Cl buffer, pH 8.0 containing 1 然 heme and COX-1 (ovine) or COX-2(human recombinant), which was preincubated for 10 min in a water bath ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Universiti Kebangsaan Malaysia, Jalan Raja Muda Abdul Aziz

LigandPNGBDBM17638(2-{1-[(4-chlorophenyl)carbonyl]-5-methoxy-2-methyl...)
Affinity DataIC50:  3.44E+3nMpH: 8.0 T: 2°CAssay Description:100 mM Tris澦Cl buffer, pH 8.0 containing 1 然 heme and COX-1 (ovine) or COX-2(human recombinant), which was preincubated for 10 min in a water bath ...More data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Universiti Kebangsaan Malaysia, Jalan Raja Muda Abdul Aziz

LigandPNGBDBM153286(3-Benzofuran-2-yl-5-(4-dimethylamino-naphthalen-1-...)
Affinity DataIC50:  4.53E+3nMpH: 8.0 T: 2°CAssay Description:100 mM Tris澦Cl buffer, pH 8.0 containing 1 然 heme and COX-1 (ovine) or COX-2(human recombinant), which was preincubated for 10 min in a water bath ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Universiti Kebangsaan Malaysia, Jalan Raja Muda Abdul Aziz

LigandPNGBDBM153294(3-Benzofuran-2-yl-5-(2,3-dimethoxy-naphthalen-1-yl...)
Affinity DataIC50:  5.02E+3nMpH: 8.0 T: 2°CAssay Description:100 mM Tris澦Cl buffer, pH 8.0 containing 1 然 heme and COX-1 (ovine) or COX-2(human recombinant), which was preincubated for 10 min in a water bath ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2 group V(Homo sapiens (Human))
Universiti Kebangsaan Malaysia, Jalan Raja Muda Abdul Aziz

LigandPNGBDBM153297(3-(2,3-Dihydro-benzo[1,4]dioxin-6-yl)-5-(4,7- dime...)
Affinity DataIC50:  5.12E+3nMpH: 7.5 T: 2°CAssay Description:Briefly, sn-2ester bond of the substrate 1,2-bis(heptanoylthio)-glycerophosphocholine was hydrolyzed by PLA2-V followed by the exposure of free thiol...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Universiti Kebangsaan Malaysia, Jalan Raja Muda Abdul Aziz

LigandPNGBDBM153283(1-(2,3-Dihydro-benzo[1,4]dioxin-6-yl)-3-(4-dimethy...)
Affinity DataIC50:  7.06E+3nMpH: 8.0 T: 2°CAssay Description:100 mM Tris澦Cl buffer, pH 8.0 containing 1 然 heme and COX-1 (ovine) or COX-2(human recombinant), which was preincubated for 10 min in a water bath ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPhospholipase A2 group V(Homo sapiens (Human))
Universiti Kebangsaan Malaysia, Jalan Raja Muda Abdul Aziz

LigandPNGBDBM153291(3-(2,3-Dihydro-benzo[1,4]dioxin-6-yl)-5-(4,7- dime...)
Affinity DataIC50:  7.12E+3nMpH: 7.5 T: 2°CAssay Description:Briefly, sn-2ester bond of the substrate 1,2-bis(heptanoylthio)-glycerophosphocholine was hydrolyzed by PLA2-V followed by the exposure of free thiol...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Universiti Kebangsaan Malaysia, Jalan Raja Muda Abdul Aziz

LigandPNGBDBM153287(3-Benzofuran-2-yl-5-(4,7-dimethoxy-naphthalen-1-yl...)
Affinity DataIC50:  7.22E+3nMpH: 8.0 T: 2°CAssay Description:100 mM Tris澦Cl buffer, pH 8.0 containing 1 然 heme and COX-1 (ovine) or COX-2(human recombinant), which was preincubated for 10 min in a water bath ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Universiti Kebangsaan Malaysia, Jalan Raja Muda Abdul Aziz

LigandPNGBDBM153288(3-Benzofuran-2-yl-5-(2,3-dimethoxy-naphthalen-1-yl...)
Affinity DataIC50:  8.06E+3nMpH: 8.0 T: 2°CAssay Description:100 mM Tris澦Cl buffer, pH 8.0 containing 1 然 heme and COX-1 (ovine) or COX-2(human recombinant), which was preincubated for 10 min in a water bath ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Universiti Kebangsaan Malaysia, Jalan Raja Muda Abdul Aziz

LigandPNGBDBM153285(1-(2,3-Dihydro-benzo[1,4]dioxin-6-yl)-3-(4,7-dimet...)
Affinity DataIC50:  8.22E+3nMpH: 8.0 T: 2°CAssay Description:100 mM Tris澦Cl buffer, pH 8.0 containing 1 然 heme and COX-1 (ovine) or COX-2(human recombinant), which was preincubated for 10 min in a water bath ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2 group V(Homo sapiens (Human))
Universiti Kebangsaan Malaysia, Jalan Raja Muda Abdul Aziz

LigandPNGBDBM153294(3-Benzofuran-2-yl-5-(2,3-dimethoxy-naphthalen-1-yl...)
Affinity DataIC50:  8.46E+3nMpH: 7.5 T: 2°CAssay Description:Briefly, sn-2ester bond of the substrate 1,2-bis(heptanoylthio)-glycerophosphocholine was hydrolyzed by PLA2-V followed by the exposure of free thiol...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Universiti Kebangsaan Malaysia, Jalan Raja Muda Abdul Aziz

LigandPNGBDBM153292(3-Benzofuran-2-yl-5-(4-dimethylamino-naphthalen-1-...)
Affinity DataIC50:  9.10E+3nMpH: 8.0 T: 2°CAssay Description:100 mM Tris澦Cl buffer, pH 8.0 containing 1 然 heme and COX-1 (ovine) or COX-2(human recombinant), which was preincubated for 10 min in a water bath ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2 group V(Homo sapiens (Human))
Universiti Kebangsaan Malaysia, Jalan Raja Muda Abdul Aziz

LigandPNGBDBM153288(3-Benzofuran-2-yl-5-(2,3-dimethoxy-naphthalen-1-yl...)
Affinity DataIC50:  9.17E+3nMpH: 7.5 T: 2°CAssay Description:Briefly, sn-2ester bond of the substrate 1,2-bis(heptanoylthio)-glycerophosphocholine was hydrolyzed by PLA2-V followed by the exposure of free thiol...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Universiti Kebangsaan Malaysia, Jalan Raja Muda Abdul Aziz

LigandPNGBDBM153280(1-Benzofuran-2-yl-3-(4-dimethylamino-naphthalen-1-...)
Affinity DataIC50:  9.27E+3nMpH: 8.0 T: 2°CAssay Description:100 mM Tris澦Cl buffer, pH 8.0 containing 1 然 heme and COX-1 (ovine) or COX-2(human recombinant), which was preincubated for 10 min in a water bath ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Universiti Kebangsaan Malaysia, Jalan Raja Muda Abdul Aziz

LigandPNGBDBM153295(3-(2,3-Dihydro-benzo[1,4]dioxin-6-yl)-5-(4-dimethy...)
Affinity DataIC50:  9.72E+3nMpH: 8.0 T: 2°CAssay Description:100 mM Tris澦Cl buffer, pH 8.0 containing 1 然 heme and COX-1 (ovine) or COX-2(human recombinant), which was preincubated for 10 min in a water bath ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Universiti Kebangsaan Malaysia, Jalan Raja Muda Abdul Aziz

LigandPNGBDBM153288(3-Benzofuran-2-yl-5-(2,3-dimethoxy-naphthalen-1-yl...)
Affinity DataIC50:  1.03E+4nMpH: 8.0 T: 2°CAssay Description:100 mM Tris澦Cl buffer, pH 8.0 containing 1 然 heme and COX-1 (ovine) or COX-2(human recombinant), which was preincubated for 10 min in a water bath ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Universiti Kebangsaan Malaysia, Jalan Raja Muda Abdul Aziz

LigandPNGBDBM153293(3-Benzofuran-2-yl-5-(4,7-dimethoxy-naphthalen-1-yl...)
Affinity DataIC50:  1.11E+4nMpH: 8.0 T: 2°CAssay Description:100 mM Tris澦Cl buffer, pH 8.0 containing 1 然 heme and COX-1 (ovine) or COX-2(human recombinant), which was preincubated for 10 min in a water bath ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Universiti Kebangsaan Malaysia, Jalan Raja Muda Abdul Aziz

LigandPNGBDBM153284(1-(2,3-Dihydro-benzo[1,4]dioxin-6-yl)-3-(2,3-dimet...)
Affinity DataIC50:  1.11E+4nMpH: 8.0 T: 2°CAssay Description:100 mM Tris澦Cl buffer, pH 8.0 containing 1 然 heme and COX-1 (ovine) or COX-2(human recombinant), which was preincubated for 10 min in a water bath ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Universiti Kebangsaan Malaysia, Jalan Raja Muda Abdul Aziz

LigandPNGBDBM153297(3-(2,3-Dihydro-benzo[1,4]dioxin-6-yl)-5-(4,7- dime...)
Affinity DataIC50:  1.20E+4nMpH: 8.0 T: 2°CAssay Description:100 mM Tris澦Cl buffer, pH 8.0 containing 1 然 heme and COX-1 (ovine) or COX-2(human recombinant), which was preincubated for 10 min in a water bath ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Universiti Kebangsaan Malaysia, Jalan Raja Muda Abdul Aziz

LigandPNGBDBM153282(1-Benzofuran-2-yl-3-(2,3-dimethoxy-naphthalen-1-yl...)
Affinity DataIC50:  1.22E+4nMpH: 8.0 T: 2°CAssay Description:100 mM Tris澦Cl buffer, pH 8.0 containing 1 然 heme and COX-1 (ovine) or COX-2(human recombinant), which was preincubated for 10 min in a water bath ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Universiti Kebangsaan Malaysia, Jalan Raja Muda Abdul Aziz

LigandPNGBDBM153296(3-(2,3-Dihydro-benzo[1,4]dioxin-6-yl)-5-(2,3-dimet...)
Affinity DataIC50:  1.23E+4nMpH: 8.0 T: 2°CAssay Description:100 mM Tris澦Cl buffer, pH 8.0 containing 1 然 heme and COX-1 (ovine) or COX-2(human recombinant), which was preincubated for 10 min in a water bath ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Universiti Kebangsaan Malaysia, Jalan Raja Muda Abdul Aziz

LigandPNGBDBM153287(3-Benzofuran-2-yl-5-(4,7-dimethoxy-naphthalen-1-yl...)
Affinity DataIC50:  1.23E+4nMpH: 8.0 T: 2°CAssay Description:100 mM Tris澦Cl buffer, pH 8.0 containing 1 然 heme and COX-1 (ovine) or COX-2(human recombinant), which was preincubated for 10 min in a water bath ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Universiti Kebangsaan Malaysia, Jalan Raja Muda Abdul Aziz

LigandPNGBDBM153285(1-(2,3-Dihydro-benzo[1,4]dioxin-6-yl)-3-(4,7-dimet...)
Affinity DataIC50:  1.25E+4nMpH: 8.0 T: 2°CAssay Description:100 mM Tris澦Cl buffer, pH 8.0 containing 1 然 heme and COX-1 (ovine) or COX-2(human recombinant), which was preincubated for 10 min in a water bath ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Universiti Kebangsaan Malaysia, Jalan Raja Muda Abdul Aziz

LigandPNGBDBM153282(1-Benzofuran-2-yl-3-(2,3-dimethoxy-naphthalen-1-yl...)
Affinity DataIC50:  1.25E+4nMpH: 8.0 T: 2°CAssay Description:100 mM Tris澦Cl buffer, pH 8.0 containing 1 然 heme and COX-1 (ovine) or COX-2(human recombinant), which was preincubated for 10 min in a water bath ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Universiti Kebangsaan Malaysia, Jalan Raja Muda Abdul Aziz

LigandPNGBDBM153291(3-(2,3-Dihydro-benzo[1,4]dioxin-6-yl)-5-(4,7- dime...)
Affinity DataIC50:  1.26E+4nMpH: 8.0 T: 2°CAssay Description:100 mM Tris澦Cl buffer, pH 8.0 containing 1 然 heme and COX-1 (ovine) or COX-2(human recombinant), which was preincubated for 10 min in a water bath ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2 group V(Homo sapiens (Human))
Universiti Kebangsaan Malaysia, Jalan Raja Muda Abdul Aziz

LigandPNGBDBM153282(1-Benzofuran-2-yl-3-(2,3-dimethoxy-naphthalen-1-yl...)
Affinity DataIC50:  1.27E+4nMpH: 7.5 T: 2°CAssay Description:Briefly, sn-2ester bond of the substrate 1,2-bis(heptanoylthio)-glycerophosphocholine was hydrolyzed by PLA2-V followed by the exposure of free thiol...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Universiti Kebangsaan Malaysia, Jalan Raja Muda Abdul Aziz

LigandPNGBDBM153289(3-(2,3-Dihydro-benzo[1,4]dioxin-6-yl)-5-(4-dimethy...)
Affinity DataIC50:  1.32E+4nMpH: 8.0 T: 2°CAssay Description:100 mM Tris澦Cl buffer, pH 8.0 containing 1 然 heme and COX-1 (ovine) or COX-2(human recombinant), which was preincubated for 10 min in a water bath ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2 group V(Homo sapiens (Human))
Universiti Kebangsaan Malaysia, Jalan Raja Muda Abdul Aziz

LigandPNGBDBM153293(3-Benzofuran-2-yl-5-(4,7-dimethoxy-naphthalen-1-yl...)
Affinity DataIC50:  1.46E+4nMpH: 7.5 T: 2°CAssay Description:Briefly, sn-2ester bond of the substrate 1,2-bis(heptanoylthio)-glycerophosphocholine was hydrolyzed by PLA2-V followed by the exposure of free thiol...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Universiti Kebangsaan Malaysia, Jalan Raja Muda Abdul Aziz

LigandPNGBDBM153286(3-Benzofuran-2-yl-5-(4-dimethylamino-naphthalen-1-...)
Affinity DataIC50:  1.46E+4nMpH: 8.0 T: 2°CAssay Description:100 mM Tris澦Cl buffer, pH 8.0 containing 1 然 heme and COX-1 (ovine) or COX-2(human recombinant), which was preincubated for 10 min in a water bath ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Universiti Kebangsaan Malaysia, Jalan Raja Muda Abdul Aziz

LigandPNGBDBM153281(1-Benzofuran-2-yl-3-(4,7-dimethoxy-naphthalen-1-yl...)
Affinity DataIC50:  1.50E+4nMpH: 8.0 T: 2°CAssay Description:100 mM Tris澦Cl buffer, pH 8.0 containing 1 然 heme and COX-1 (ovine) or COX-2(human recombinant), which was preincubated for 10 min in a water bath ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2 group V(Homo sapiens (Human))
Universiti Kebangsaan Malaysia, Jalan Raja Muda Abdul Aziz

LigandPNGBDBM153295(3-(2,3-Dihydro-benzo[1,4]dioxin-6-yl)-5-(4-dimethy...)
Affinity DataIC50:  1.72E+4nMpH: 7.5 T: 2°CAssay Description:Briefly, sn-2ester bond of the substrate 1,2-bis(heptanoylthio)-glycerophosphocholine was hydrolyzed by PLA2-V followed by the exposure of free thiol...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2 group V(Homo sapiens (Human))
Universiti Kebangsaan Malaysia, Jalan Raja Muda Abdul Aziz

LigandPNGBDBM153296(3-(2,3-Dihydro-benzo[1,4]dioxin-6-yl)-5-(2,3-dimet...)
Affinity DataIC50:  1.73E+4nMpH: 7.5 T: 2°CAssay Description:Briefly, sn-2ester bond of the substrate 1,2-bis(heptanoylthio)-glycerophosphocholine was hydrolyzed by PLA2-V followed by the exposure of free thiol...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Universiti Kebangsaan Malaysia, Jalan Raja Muda Abdul Aziz

LigandPNGBDBM153290(3-(2,3-Dihydro-benzo[1,4]dioxin-6-yl)-5-(2,3-dimet...)
Affinity DataIC50:  1.78E+4nMpH: 8.0 T: 2°CAssay Description:100 mM Tris澦Cl buffer, pH 8.0 containing 1 然 heme and COX-1 (ovine) or COX-2(human recombinant), which was preincubated for 10 min in a water bath ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Universiti Kebangsaan Malaysia, Jalan Raja Muda Abdul Aziz

LigandPNGBDBM153284(1-(2,3-Dihydro-benzo[1,4]dioxin-6-yl)-3-(2,3-dimet...)
Affinity DataIC50:  1.85E+4nMpH: 8.0 T: 2°CAssay Description:100 mM Tris澦Cl buffer, pH 8.0 containing 1 然 heme and COX-1 (ovine) or COX-2(human recombinant), which was preincubated for 10 min in a water bath ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2 group V(Homo sapiens (Human))
Universiti Kebangsaan Malaysia, Jalan Raja Muda Abdul Aziz

LigandPNGBDBM153285(1-(2,3-Dihydro-benzo[1,4]dioxin-6-yl)-3-(4,7-dimet...)
Affinity DataIC50:  1.91E+4nMpH: 7.5 T: 2°CAssay Description:Briefly, sn-2ester bond of the substrate 1,2-bis(heptanoylthio)-glycerophosphocholine was hydrolyzed by PLA2-V followed by the exposure of free thiol...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Universiti Kebangsaan Malaysia, Jalan Raja Muda Abdul Aziz

LigandPNGBDBM153281(1-Benzofuran-2-yl-3-(4,7-dimethoxy-naphthalen-1-yl...)
Affinity DataIC50:  1.91E+4nMpH: 8.0 T: 2°CAssay Description:100 mM Tris澦Cl buffer, pH 8.0 containing 1 然 heme and COX-1 (ovine) or COX-2(human recombinant), which was preincubated for 10 min in a water bath ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2 group V(Homo sapiens (Human))
Universiti Kebangsaan Malaysia, Jalan Raja Muda Abdul Aziz

LigandPNGBDBM153290(3-(2,3-Dihydro-benzo[1,4]dioxin-6-yl)-5-(2,3-dimet...)
Affinity DataIC50:  1.92E+4nMpH: 7.5 T: 2°CAssay Description:Briefly, sn-2ester bond of the substrate 1,2-bis(heptanoylthio)-glycerophosphocholine was hydrolyzed by PLA2-V followed by the exposure of free thiol...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2 group V(Homo sapiens (Human))
Universiti Kebangsaan Malaysia, Jalan Raja Muda Abdul Aziz

LigandPNGBDBM153287(3-Benzofuran-2-yl-5-(4,7-dimethoxy-naphthalen-1-yl...)
Affinity DataIC50:  2.11E+4nMpH: 7.5 T: 2°CAssay Description:Briefly, sn-2ester bond of the substrate 1,2-bis(heptanoylthio)-glycerophosphocholine was hydrolyzed by PLA2-V followed by the exposure of free thiol...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2 group V(Homo sapiens (Human))
Universiti Kebangsaan Malaysia, Jalan Raja Muda Abdul Aziz

LigandPNGBDBM153292(3-Benzofuran-2-yl-5-(4-dimethylamino-naphthalen-1-...)
Affinity DataIC50:  2.22E+4nMpH: 7.5 T: 2°CAssay Description:Briefly, sn-2ester bond of the substrate 1,2-bis(heptanoylthio)-glycerophosphocholine was hydrolyzed by PLA2-V followed by the exposure of free thiol...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2 group V(Homo sapiens (Human))
Universiti Kebangsaan Malaysia, Jalan Raja Muda Abdul Aziz

LigandPNGBDBM153289(3-(2,3-Dihydro-benzo[1,4]dioxin-6-yl)-5-(4-dimethy...)
Affinity DataIC50:  2.22E+4nMpH: 7.5 T: 2°CAssay Description:Briefly, sn-2ester bond of the substrate 1,2-bis(heptanoylthio)-glycerophosphocholine was hydrolyzed by PLA2-V followed by the exposure of free thiol...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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