Compile Data Set for Download or QSAR
maximum 50k data
Found 2 Enz. Inhib. hit(s) with all data for entry = 50044870
TargetCaspase-1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50033886(CHEMBL2047937 | Ethyl 2-((2-Chlorophenyl)(Hydroxy)...)
Affinity DataKi:  9.60E+3nMAssay Description:Inhibition of caspase 1 (unknown origin) using N-acetyl-Tyr-Val-Ala-Asp-para-nitroanilide substrate assessed as rate of para-nitroanilide release by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50433441(PARTHENOLIDE)
Affinity DataKi:  1.06E+4nMAssay Description:Inhibition of caspase 1 (unknown origin) using N-acetyl-Tyr-Val-Ala-Asp-para-nitroanilide substrate assessed as rate of para-nitroanilide release by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed