Compile Data Set for Download or QSAR
maximum 50k data
Report error Found 65 Enz. Inhib. hit(s) with all data for entry = 50035803
TargetMu-type opioid receptor(Guinea pig)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50017233(CHEMBL592 | LEVO-DROMORAN | LEVORPHANOL)
Affinity DataIC50:  0.600nMAssay Description:Inhibitory activity against opioid receptor mu of guinea pig brain using [3H]DAGO radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Guinea pig)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50017059(3,4-Dibromo-N-methyl-N-(1-methyl-1-aza-spiro[4.5]d...)
Affinity DataIC50:  2nMAssay Description:Inhibitory activity against opioid receptor mu of guinea pig brain using [3H]DAGO radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50017233(CHEMBL592 | LEVO-DROMORAN | LEVORPHANOL)
Affinity DataIC50:  2.90nMAssay Description:Inhibitory activity against opioid receptor delta of guinea pig was determined by using [3H]DADLE radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank


TargetMu-type opioid receptor(Guinea pig)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50017065(3,4-Dichloro-N-methyl-N-(1-methyl-1-aza-spiro[4.5]...)
Affinity DataIC50:  6.30nMAssay Description:Inhibitory activity against opioid receptor mu of guinea pig brain using [3H]DAGO radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Guinea pig)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50017060(CHEMBL553991 | N-Methyl-N-(1-methyl-1-aza-spiro[4....)
Affinity DataIC50:  12nMAssay Description:Inhibitory activity against opioid receptor mu of guinea pig brain using [3H]DAGO radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Guinea pig)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50017061(4-Bromo-2-chloro-N-methyl-N-(1-methyl-1-aza-spiro[...)
Affinity DataIC50:  16nMAssay Description:Inhibitory activity against opioid receptor mu of guinea pig brain using [3H]DAGO radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Guinea pig)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50017071(4-Bromo-N-methyl-N-(1-methyl-1-aza-spiro[4.5]dec-6...)
Affinity DataIC50:  17nMAssay Description:Inhibitory activity against opioid receptor mu of guinea pig brain using [3H]DAGO radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Guinea pig)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50017078(4-Bromo-2,N-dimethyl-N-(1-methyl-1-aza-spiro[4.5]d...)
Affinity DataIC50:  21nMAssay Description:Inhibitory activity against opioid receptor mu of guinea pig brain using [3H]DAGO radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Guinea pig)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50017068(2-(3,4-Dichloro-phenyl)-N-methyl-N-(1-methyl-1-aza...)
Affinity DataIC50:  87nMAssay Description:Inhibitory activity against Opioid receptor mu 1 of guinea pig brain using [3H]DAG0 radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Guinea pig)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50017059(3,4-Dibromo-N-methyl-N-(1-methyl-1-aza-spiro[4.5]d...)
Affinity DataIC50:  105nMAssay Description:Binding inhibition against opioid receptor kappa of guinea pig was determined using [3H]ethylketocyclazocineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Guinea pig)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50017064(4,N-Dimethyl-N-(1-methyl-1-aza-spiro[4.5]dec-6-yl)...)
Affinity DataIC50:  150nMAssay Description:Inhibitory activity against opioid receptor mu of guinea pig brain using [3H]DAGO radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Guinea pig)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50017077(3,4-Dichloro-N-(1-methyl-1-aza-spiro[4.5]dec-6-yl)...)
Affinity DataIC50:  210nMAssay Description:Inhibitory activity against opioid receptor mu of guinea pig brain using [3H]DAGO radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Guinea pig)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50017072(4-Bromo-N-cyclopropylmethyl-N-(1-methyl-1-aza-spir...)
Affinity DataIC50:  220nMAssay Description:Inhibitory activity against opioid receptor mu of guinea pig brain using [3H]DAGO radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Guinea pig)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50017074(2-(3,4-Dichloro-phenyl)-N-(1-methyl-1-aza-spiro[4....)
Affinity DataIC50:  250nMAssay Description:Inhibitory activity against Opioid receptor mu 1 of guinea pig brain using [3H]DAG0 radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Guinea pig)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50017065(3,4-Dichloro-N-methyl-N-(1-methyl-1-aza-spiro[4.5]...)
Affinity DataIC50:  309nMAssay Description:Binding inhibition against opioid receptor kappa of guinea pig was determined using [3H]ethylketocyclazocineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Guinea pig)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50017079(4-Chloro-N-(1-methyl-1-aza-spiro[4.5]dec-6-yl)-ben...)
Affinity DataIC50:  550nMAssay Description:Inhibitory activity against opioid receptor mu of guinea pig brain using [3H]DAGO radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Guinea pig)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50017070(4-Bromo-N-isobutyl-N-(1-methyl-1-aza-spiro[4.5]dec...)
Affinity DataIC50:  580nMAssay Description:Inhibitory activity against opioid receptor mu of guinea pig brain using [3H]DAGO radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Guinea pig)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50017063(4-Bromo-N-(1-methyl-1-aza-spiro[4.5]dec-6-yl)-benz...)
Affinity DataIC50:  600nMAssay Description:Inhibitory activity against opioid receptor mu of guinea pig brain using [3H]DAGO radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Guinea pig)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50017060(CHEMBL553991 | N-Methyl-N-(1-methyl-1-aza-spiro[4....)
Affinity DataIC50:  670nMAssay Description:Binding inhibition against opioid receptor kappa of guinea pig was determined using [3H]ethylketocyclazocineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Guinea pig)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50017071(4-Bromo-N-methyl-N-(1-methyl-1-aza-spiro[4.5]dec-6...)
Affinity DataIC50:  670nMAssay Description:Binding inhibition against opioid receptor kappa of guinea pig was determined using [3H]ethylketocyclazocineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Guinea pig)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50017076(2-(4-Bromo-phenyl)-N-(1-methyl-1-aza-spiro[4.5]dec...)
Affinity DataIC50:  720nMAssay Description:Inhibitory activity against Opioid receptor mu 1 of guinea pig brain using [3H]DAGO radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Guinea pig)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50017078(4-Bromo-2,N-dimethyl-N-(1-methyl-1-aza-spiro[4.5]d...)
Affinity DataIC50:  880nMAssay Description:Binding inhibition against opioid receptor kappa of guinea pig was determined using [3H]ethylketocyclazocineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Guinea pig)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50017066(4-Methoxy-N-(1-methyl-1-aza-spiro[4.5]dec-6-yl)-be...)
Affinity DataIC50:  2.20E+3nMAssay Description:Inhibitory activity against opioid receptor mu of guinea pig brain using [3H]DAGO radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50017059(3,4-Dibromo-N-methyl-N-(1-methyl-1-aza-spiro[4.5]d...)
Affinity DataIC50:  2.30E+3nMAssay Description:Inhibitory activity against opioid receptor delta of guinea pig was determined by using [3H]DADLE radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Guinea pig)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50017067(CHEMBL25386 | N-(1-Methyl-1-aza-spiro[4.5]dec-6-yl...)
Affinity DataIC50:  2.80E+3nMAssay Description:Binding inhibition against opioid receptor kappa of guinea pig was determined using [3H]ethylketocyclazocineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Guinea pig)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50017072(4-Bromo-N-cyclopropylmethyl-N-(1-methyl-1-aza-spir...)
Affinity DataIC50:  2.80E+3nMAssay Description:Binding inhibition against opioid receptor kappa of guinea pig was determined using [3H]ethylketocyclazocineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50017074(2-(3,4-Dichloro-phenyl)-N-(1-methyl-1-aza-spiro[4....)
Affinity DataIC50:  5.80E+3nMAssay Description:Inhibitory activity against Opioid receptor delta 1 of guinea pig was determined by using [3H]DADLE radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50017072(4-Bromo-N-cyclopropylmethyl-N-(1-methyl-1-aza-spir...)
Affinity DataIC50:  6.30E+3nMAssay Description:Inhibitory activity against opioid receptor delta of guinea pig was determined by using [3H]DADLE radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50017061(4-Bromo-2-chloro-N-methyl-N-(1-methyl-1-aza-spiro[...)
Affinity DataIC50:  9.00E+3nMAssay Description:Inhibitory activity against opioid receptor delta of guinea pig was determined by using [3H]DADLE radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50017060(CHEMBL553991 | N-Methyl-N-(1-methyl-1-aza-spiro[4....)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibitory activity against opioid receptor delta of guinea pig was determined by using [3H]DADLE radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50017071(4-Bromo-N-methyl-N-(1-methyl-1-aza-spiro[4.5]dec-6...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibitory activity against opioid receptor delta of guinea pig was determined by using [3H]DADLE radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Guinea pig)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50017077(3,4-Dichloro-N-(1-methyl-1-aza-spiro[4.5]dec-6-yl)...)
Affinity DataIC50: >1.00E+4nMAssay Description:Binding inhibition against opioid receptor kappa of guinea pig was determined using [3H]ethylketocyclazocineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Guinea pig)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50017064(4,N-Dimethyl-N-(1-methyl-1-aza-spiro[4.5]dec-6-yl)...)
Affinity DataIC50: >1.00E+4nMAssay Description:Binding inhibition against opioid receptor kappa of guinea pig was determined using [3H]ethylketocyclazocineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Guinea pig)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50017068(2-(3,4-Dichloro-phenyl)-N-methyl-N-(1-methyl-1-aza...)
Affinity DataIC50: >1.00E+4nMAssay Description:Binding inhibition against Opioid receptor kappa 1 of guinea pig was determined using [3H]ethylketocyclazocineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50017063(4-Bromo-N-(1-methyl-1-aza-spiro[4.5]dec-6-yl)-benz...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibitory activity against opioid receptor delta of guinea pig was determined by using [3H]DADLE radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50017078(4-Bromo-2,N-dimethyl-N-(1-methyl-1-aza-spiro[4.5]d...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibitory activity against opioid receptor delta of guinea pig was determined by using [3H]DADLE radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50017062(3-Bromo-N-(1-methyl-1-aza-spiro[4.5]dec-6-yl)-benz...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibitory activity against opioid receptor delta of guinea pig was determined by using [3H]DADLE radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Guinea pig)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50017074(2-(3,4-Dichloro-phenyl)-N-(1-methyl-1-aza-spiro[4....)
Affinity DataIC50: >1.00E+4nMAssay Description:Binding inhibition against Opioid receptor kappa 1 of guinea pig was determined using [3H]ethylketocyclazocineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Guinea pig)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50017076(2-(4-Bromo-phenyl)-N-(1-methyl-1-aza-spiro[4.5]dec...)
Affinity DataIC50: >1.00E+4nMAssay Description:Binding inhibition against Opioid receptor kappa 1 of guinea pig was determined using [3H]ethylketocyclazocineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Guinea pig)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50017073(4-Fluoro-N-(1-methyl-1-aza-spiro[4.5]dec-6-yl)-ben...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibitory activity against opioid receptor mu of guinea pig brain using [3H]DAGO radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Guinea pig)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50017066(4-Methoxy-N-(1-methyl-1-aza-spiro[4.5]dec-6-yl)-be...)
Affinity DataIC50: >1.00E+4nMAssay Description:Binding inhibition against opioid receptor kappa of guinea pig was determined using [3H]ethylketocyclazocineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Guinea pig)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50017067(CHEMBL25386 | N-(1-Methyl-1-aza-spiro[4.5]dec-6-yl...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibitory activity against opioid receptor mu of guinea pig brain using [3H]DAGO radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Guinea pig)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50017073(4-Fluoro-N-(1-methyl-1-aza-spiro[4.5]dec-6-yl)-ben...)
Affinity DataIC50: >1.00E+4nMAssay Description:Binding inhibition against opioid receptor kappa of guinea pig was determined using [3H]ethylketocyclazocineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Guinea pig)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50017079(4-Chloro-N-(1-methyl-1-aza-spiro[4.5]dec-6-yl)-ben...)
Affinity DataIC50: >1.00E+4nMAssay Description:Binding inhibition against opioid receptor kappa of guinea pig was determined using [3H]ethylketocyclazocineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50017058(2-Bromo-N-(1-methyl-1-aza-spiro[4.5]dec-6-yl)-benz...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibitory activity against opioid receptor delta of guinea pig was determined by using [3H]DADLE radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50017064(4,N-Dimethyl-N-(1-methyl-1-aza-spiro[4.5]dec-6-yl)...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibitory activity against opioid receptor delta of guinea pig was determined by using [3H]DADLE radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Guinea pig)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50017063(4-Bromo-N-(1-methyl-1-aza-spiro[4.5]dec-6-yl)-benz...)
Affinity DataIC50: >1.00E+4nMAssay Description:Binding inhibition against opioid receptor kappa of guinea pig was determined using [3H]ethylketocyclazocineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Guinea pig)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50017069(4-Bromo-N-(1-methyl-1-aza-spiro[4.5]dec-6-yl)-benz...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibitory activity against Opioid receptor mu 1 of guinea pig brain using [3H]DAGO radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Guinea pig)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50017061(4-Bromo-2-chloro-N-methyl-N-(1-methyl-1-aza-spiro[...)
Affinity DataIC50: >1.00E+4nMAssay Description:Binding inhibition against opioid receptor kappa of guinea pig was determined using [3H]ethylketocyclazocineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Guinea pig)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50017058(2-Bromo-N-(1-methyl-1-aza-spiro[4.5]dec-6-yl)-benz...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibitory activity against opioid receptor mu of guinea pig brain using [3H]DAGO radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

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