Report error Found 93 Enz. Inhib. hit(s) with all data for entry = 50044994
Affinity DataKi: 11nMAssay Description:Displacement of [3H]WIN-55212-2 from human CB2R expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 19nMAssay Description:Agonist activity at human CB2R expressed in CHO cells assessed as reduction in forskolin-induced cAMP accumulation by beta-galactosidase based comple...More data for this Ligand-Target Pair
Affinity DataKi: 23nMAssay Description:Displacement of [3H]WIN-55212-2 from human CB2R expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 27nMAssay Description:Agonist activity at human CB2R expressed in CHO cells assessed as reduction in forskolin-induced cAMP accumulation by beta-galactosidase based comple...More data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:Displacement of [3H]WIN-55212-2 from human CB2R expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 32nMAssay Description:Agonist activity at human CB2R expressed in CHO cells assessed as reduction in forskolin-induced cAMP accumulation by beta-galactosidase based comple...More data for this Ligand-Target Pair
Affinity DataEC50: 33nMAssay Description:Agonist activity at human CB2R expressed in CHO cells assessed as reduction in forskolin-induced cAMP accumulation by beta-galactosidase based comple...More data for this Ligand-Target Pair
Affinity DataEC50: 37nMAssay Description:Agonist activity at human CB2R expressed in CHO cells assessed as reduction in forskolin-induced cAMP accumulation by beta-galactosidase based comple...More data for this Ligand-Target Pair
Affinity DataEC50: 39nMAssay Description:Agonist activity at human CB2R expressed in CHO cells assessed as reduction in forskolin-induced cAMP accumulation by beta-galactosidase based comple...More data for this Ligand-Target Pair
Affinity DataEC50: 42nMAssay Description:Agonist activity at human CB2R expressed in CHO cells assessed as reduction in forskolin-induced cAMP accumulation by beta-galactosidase based comple...More data for this Ligand-Target Pair
Affinity DataEC50: 46nMAssay Description:Agonist activity at human CB2R expressed in CHO cells assessed as reduction in forskolin-induced cAMP accumulation by beta-galactosidase based comple...More data for this Ligand-Target Pair
Affinity DataEC50: 48nMAssay Description:Agonist activity at human CB2R expressed in CHO cells assessed as reduction in forskolin-induced cAMP accumulation by beta-galactosidase based comple...More data for this Ligand-Target Pair
Affinity DataEC50: 49nMAssay Description:Agonist activity at human CB2R expressed in CHO cells assessed as reduction in forskolin-induced cAMP accumulation by beta-galactosidase based comple...More data for this Ligand-Target Pair
Affinity DataEC50: 53nMAssay Description:Agonist activity at human CB2R expressed in CHO cells assessed as reduction in forskolin-induced cAMP accumulation by beta-galactosidase based comple...More data for this Ligand-Target Pair
Affinity DataEC50: 57nMAssay Description:Agonist activity at human CB2R expressed in CHO cells assessed as reduction in forskolin-induced cAMP accumulation by beta-galactosidase based comple...More data for this Ligand-Target Pair
Affinity DataKi: 61nMAssay Description:Displacement of [3H]CP55940 from human CB1R expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 73nMAssay Description:Agonist activity at human CB2R expressed in CHO cells assessed as reduction in forskolin-induced cAMP accumulation by beta-galactosidase based comple...More data for this Ligand-Target Pair
Affinity DataEC50: 75nMAssay Description:Agonist activity at human CB2R expressed in CHO cells assessed as reduction in forskolin-induced cAMP accumulation by beta-galactosidase based comple...More data for this Ligand-Target Pair
Affinity DataEC50: 76nMAssay Description:Agonist activity at human CB2R expressed in CHO cells assessed as reduction in forskolin-induced cAMP accumulation by beta-galactosidase based comple...More data for this Ligand-Target Pair
Affinity DataEC50: 92nMAssay Description:Agonist activity at human CB2R expressed in CHO cells assessed as reduction in forskolin-induced cAMP accumulation by beta-galactosidase based comple...More data for this Ligand-Target Pair
Affinity DataEC50: 106nMAssay Description:Agonist activity at human CB2R expressed in CHO cells assessed as reduction in forskolin-induced cAMP accumulation by beta-galactosidase based comple...More data for this Ligand-Target Pair
Affinity DataEC50: 112nMAssay Description:Agonist activity at human CB2R expressed in CHO cells assessed as reduction in forskolin-induced cAMP accumulation by beta-galactosidase based comple...More data for this Ligand-Target Pair
Affinity DataEC50: 113nMAssay Description:Agonist activity at human CB2R expressed in CHO cells assessed as reduction in forskolin-induced cAMP accumulation by beta-galactosidase based comple...More data for this Ligand-Target Pair
Affinity DataEC50: 144nMAssay Description:Agonist activity at human CB2R expressed in CHO cells assessed as reduction in forskolin-induced cAMP accumulation by beta-galactosidase based comple...More data for this Ligand-Target Pair
Affinity DataEC50: 150nMAssay Description:Agonist activity at human CB2R expressed in CHO cells assessed as reduction in forskolin-induced cAMP accumulation by beta-galactosidase based comple...More data for this Ligand-Target Pair
Affinity DataKi: 155nMAssay Description:Displacement of [3H]WIN-55212-2 from human CB2R expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 160nMAssay Description:Agonist activity at human CB2R expressed in CHO cells assessed as reduction in forskolin-induced cAMP accumulation by beta-galactosidase based comple...More data for this Ligand-Target Pair
Affinity DataEC50: 181nMAssay Description:Agonist activity at human CB2R expressed in CHO cells assessed as reduction in forskolin-induced cAMP accumulation by beta-galactosidase based comple...More data for this Ligand-Target Pair
Affinity DataEC50: 214nMAssay Description:Agonist activity at human CB2R expressed in CHO cells assessed as reduction in forskolin-induced cAMP accumulation by beta-galactosidase based comple...More data for this Ligand-Target Pair
Affinity DataKi: 215nMAssay Description:Displacement of [3H]WIN-55212-2 from human CB2R expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 231nMAssay Description:Agonist activity at human CB2R expressed in CHO cells assessed as reduction in forskolin-induced cAMP accumulation by beta-galactosidase based comple...More data for this Ligand-Target Pair
Affinity DataKi: 235nMAssay Description:Displacement of [3H]WIN-55212-2 from human CB2R expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 270nMAssay Description:Agonist activity at human CB2R expressed in CHO cells assessed as reduction in forskolin-induced cAMP accumulation by beta-galactosidase based comple...More data for this Ligand-Target Pair
Affinity DataKi: 275nMAssay Description:Displacement of [3H]CP55940 from human CB1R expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 290nMAssay Description:Displacement of [3H]WIN-55212-2 from human CB2R expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 296nMAssay Description:Agonist activity at human CB2R expressed in CHO cells assessed as reduction in forskolin-induced cAMP accumulation by beta-galactosidase based comple...More data for this Ligand-Target Pair
Affinity DataKi: 300nMAssay Description:Displacement of [3H]WIN-55212-2 from human CB2R expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 320nMAssay Description:Displacement of [3H]WIN-55212-2 from human CB2R expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 355nMAssay Description:Displacement of [3H]WIN-55212-2 from human CB2R expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 360nMAssay Description:Displacement of [3H]WIN-55212-2 from human CB2R expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 380nMAssay Description:Displacement of [3H]WIN-55212-2 from human CB2R expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 450nMAssay Description:Displacement of [3H]WIN-55212-2 from human CB2R expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 490nMAssay Description:Displacement of [3H]WIN-55212-2 from human CB2R expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 617nMAssay Description:Agonist activity at human CB2R expressed in CHO cells assessed as reduction in forskolin-induced cAMP accumulation by beta-galactosidase based comple...More data for this Ligand-Target Pair
Affinity DataEC50: 674nMAssay Description:Agonist activity at human CB2R expressed in CHO cells assessed as reduction in forskolin-induced cAMP accumulation by beta-galactosidase based comple...More data for this Ligand-Target Pair
Affinity DataEC50: 850nMAssay Description:Agonist activity at human CB2R expressed in CHO cells assessed as reduction in forskolin-induced cAMP accumulation by beta-galactosidase based comple...More data for this Ligand-Target Pair
Affinity DataEC50: 1.55E+3nMAssay Description:Agonist activity at human CB1R expressed in CHO cells assessed as reduction in forskolin-induced cAMP accumulation by beta-galactosidase based comple...More data for this Ligand-Target Pair
Affinity DataEC50: 1.76E+3nMAssay Description:Agonist activity at human CB2R expressed in CHO cells assessed as reduction in forskolin-induced cAMP accumulation by beta-galactosidase based comple...More data for this Ligand-Target Pair
Affinity DataEC50: 2.19E+3nMAssay Description:Agonist activity at human CB2R expressed in CHO cells assessed as reduction in forskolin-induced cAMP accumulation by beta-galactosidase based comple...More data for this Ligand-Target Pair
Affinity DataEC50: >3.00E+3nMAssay Description:Agonist activity at human CB2R expressed in CHO cells assessed as reduction in forskolin-induced cAMP accumulation by beta-galactosidase based comple...More data for this Ligand-Target Pair






















3D Structure (crystal)









