Compile Data Set for Download or QSAR
Report error Found 15 Enz. Inhib. hit(s) with all data for entry = 50045016 Sort by
LigandPNGBDBM50041679(CHEMBL3358892)
Affinity DataKd:  1.90E+3nMAssay Description:Binding affinity to human MCL1 (173 to 329 aa) by isothermal titration calorimetryMore data for this Ligand-Target Pair
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PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM50041679(CHEMBL3358892)
Affinity DataKd:  6.00E+3nMAssay Description:Binding affinity to human MCL1 (173 to 329 aa) by 19F NMR spectroscopyMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM50013867(CHEMBL3265299)
Affinity DataIC50: 180nMAssay Description:Inhibition of MCL1 (unknown origin)More data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50041687(CHEMBL3358899)
Affinity DataIC50: 4.10E+3nMAssay Description:Binding affinity to human MCL1 (173 to 329 aa) using TAMRA-labeled Noxa peptide preincubated for 30 mins by fluorescent polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50041679(CHEMBL3358892)
Affinity DataIC50: 4.50E+3nMAssay Description:Binding affinity to human MCL1 (173 to 329 aa) using TAMRA-labeled Noxa peptide preincubated for 30 mins by fluorescent polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM50041674(CHEMBL3358901)
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity to human MCL1 (173 to 329 aa) using TAMRA-labeled Noxa peptide preincubated for 30 mins by fluorescent polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50041690(CHEMBL3358900)
Affinity DataIC50: 2.13E+4nMAssay Description:Binding affinity to human MCL1 (173 to 329 aa) using TAMRA-labeled Noxa peptide preincubated for 30 mins by fluorescent polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50041680(CHEMBL3358893)
Affinity DataIC50: 2.50E+4nMAssay Description:Binding affinity to human MCL1 (173 to 329 aa) using TAMRA-labeled Noxa peptide preincubated for 30 mins by fluorescent polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50041686(CHEMBL3358898)
Affinity DataIC50: 2.50E+4nMAssay Description:Binding affinity to human MCL1 (173 to 329 aa) using TAMRA-labeled Noxa peptide preincubated for 30 mins by fluorescent polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50041675(CHEMBL3358902)
Affinity DataIC50: 5.00E+4nMAssay Description:Binding affinity to human MCL1 (173 to 329 aa) using TAMRA-labeled Noxa peptide preincubated for 30 mins by fluorescent polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50041678(CHEMBL3358903)
Affinity DataIC50: 5.00E+4nMAssay Description:Binding affinity to human MCL1 (173 to 329 aa) using TAMRA-labeled Noxa peptide preincubated for 30 mins by fluorescent polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50041681(CHEMBL3358894)
Affinity DataIC50: 5.00E+4nMAssay Description:Binding affinity to human MCL1 (173 to 329 aa) using TAMRA-labeled Noxa peptide preincubated for 30 mins by fluorescent polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50041682(CHEMBL3358895)
Affinity DataIC50: 5.00E+4nMAssay Description:Binding affinity to human MCL1 (173 to 329 aa) using TAMRA-labeled Noxa peptide preincubated for 30 mins by fluorescent polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50041684(CHEMBL3358896)
Affinity DataIC50: 5.00E+4nMAssay Description:Binding affinity to human MCL1 (173 to 329 aa) using TAMRA-labeled Noxa peptide preincubated for 30 mins by fluorescent polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50041685(CHEMBL3358897)
Affinity DataIC50: 5.00E+4nMAssay Description:Binding affinity to human MCL1 (173 to 329 aa) using TAMRA-labeled Noxa peptide preincubated for 30 mins by fluorescent polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed