Compile Data Set for Download or QSAR
Report error Found 71 Enz. Inhib. hit(s) with all data for entry = 50045020 Sort by
TargetSphingosine 1-phosphate receptor 5(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50041981(CHEMBL3358955)
Affinity DataEC50:  107nMAssay Description:Agonist activity at human S1P5 receptor by beta-arrestin recruitment assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50041981(CHEMBL3358955)
Affinity DataEC50:  2.5nMAssay Description:Agonist activity at human S1P1 receptor by beta-arrestin recruitment assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50041979(CHEMBL3359520)
Affinity DataEC50:  11nMAssay Description:Agonist activity at human S1P1 receptor by beta-arrestin recruitment assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSphingosine 1-phosphate receptor 2(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50041981(CHEMBL3358955)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human S1P2 receptor by beta-arrestin recruitment assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSphingosine 1-phosphate receptor 2(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50041979(CHEMBL3359520)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human S1P2 receptor by beta-arrestin recruitment assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSphingosine 1-phosphate receptor 3(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50041981(CHEMBL3358955)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human S1P3 receptor by beta-arrestin recruitment assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSphingosine 1-phosphate receptor 3(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50041979(CHEMBL3359520)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human S1P3 receptor by beta-arrestin recruitment assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSphingosine 1-phosphate receptor 4(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50041981(CHEMBL3358955)
Affinity DataEC50:  570nMAssay Description:Agonist activity at human S1P4 receptor by beta-arrestin recruitment assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSphingosine 1-phosphate receptor 4(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50041979(CHEMBL3359520)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human S1P4 receptor by beta-arrestin recruitment assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50041979(CHEMBL3359520)
Affinity DataEC50:  0.150nMAssay Description:Agonist activity at human S1P1 receptor assessed as cAMP accumulation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSphingosine 1-phosphate receptor 5(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50041979(CHEMBL3359520)
Affinity DataEC50:  410nMAssay Description:Agonist activity at human S1P5 receptor by beta-arrestin recruitment assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50041981(CHEMBL3358955)
Affinity DataEC50:  0.0950nMAssay Description:Agonist activity at human S1P1 receptor assessed as cAMP accumulation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50041989(CHEMBL3359514)
Affinity DataEC50:  0.490nMAssay Description:Agonist activity at human S1P1 receptor assessed as cAMP accumulation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50041988(CHEMBL3359515)
Affinity DataEC50:  150nMAssay Description:Agonist activity at human S1P1 receptor assessed as cAMP accumulation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50041987(CHEMBL3359516)
Affinity DataEC50:  83nMAssay Description:Agonist activity at human S1P1 receptor assessed as cAMP accumulation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50041986(CHEMBL3359517)
Affinity DataEC50:  38nMAssay Description:Agonist activity at human S1P1 receptor assessed as cAMP accumulation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50041985(CHEMBL3359518)
Affinity DataEC50:  6.70nMAssay Description:Agonist activity at human S1P1 receptor assessed as cAMP accumulation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50041980(CHEMBL3359519)
Affinity DataEC50:  0.150nMAssay Description:Agonist activity at human S1P1 receptor assessed as cAMP accumulation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSphingosine 1-phosphate receptor 4(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50041981(CHEMBL3358955)
Affinity DataEC50:  570nMAssay Description:Agonist activity at human S1P4 receptor by beta-arrestin recruitment assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSphingosine 1-phosphate receptor 2(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50041981(CHEMBL3358955)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human S1P2 receptor by beta-arrestin recruitment assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSphingosine 1-phosphate receptor 2(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50041980(CHEMBL3359519)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human S1P2 receptor by beta-arrestin recruitment assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSphingosine 1-phosphate receptor 2(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50041980(CHEMBL3359519)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human S1P2 receptor by beta-arrestin recruitment assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSphingosine 1-phosphate receptor 2(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50041979(CHEMBL3359520)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human S1P2 receptor by beta-arrestin recruitment assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSphingosine 1-phosphate receptor 3(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50041981(CHEMBL3358955)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human S1P3 receptor by beta-arrestin recruitment assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSphingosine 1-phosphate receptor 3(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50041980(CHEMBL3359519)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human S1P3 receptor by beta-arrestin recruitment assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSphingosine 1-phosphate receptor 3(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50041980(CHEMBL3359519)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human S1P3 receptor by beta-arrestin recruitment assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSphingosine 1-phosphate receptor 3(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50041979(CHEMBL3359520)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human S1P3 receptor by beta-arrestin recruitment assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50041979(CHEMBL3359520)
Affinity DataEC50:  0.150nMAssay Description:Agonist activity at human S1P1 receptor assessed as cAMP accumulation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSphingosine 1-phosphate receptor 4(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50041980(CHEMBL3359519)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human S1P4 receptor by beta-arrestin recruitment assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSphingosine 1-phosphate receptor 4(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50041980(CHEMBL3359519)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human S1P4 receptor by beta-arrestin recruitment assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSphingosine 1-phosphate receptor 4(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50041979(CHEMBL3359520)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human S1P4 receptor by beta-arrestin recruitment assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSphingosine 1-phosphate receptor 5(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50041981(CHEMBL3358955)
Affinity DataEC50:  107nMAssay Description:Agonist activity at human S1P5 receptor by beta-arrestin recruitment assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSphingosine 1-phosphate receptor 5(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50041980(CHEMBL3359519)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human S1P5 receptor by beta-arrestin recruitment assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSphingosine 1-phosphate receptor 5(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50041980(CHEMBL3359519)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human S1P5 receptor by beta-arrestin recruitment assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSphingosine 1-phosphate receptor 5(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50041979(CHEMBL3359520)
Affinity DataEC50:  410nMAssay Description:Agonist activity at human S1P5 receptor by beta-arrestin recruitment assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50041981(CHEMBL3358955)
Affinity DataEC50:  0.0950nMAssay Description:Agonist activity at human S1P1 receptor assessed as cAMP accumulation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSphingosine 1-phosphate receptor 2(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50041983(CHEMBL3359523)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human S1P2 receptor by beta-arrestin recruitment assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Mouse)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50041983(CHEMBL3359523)
Affinity DataEC50:  0.0640nMAssay Description:Agonist activity at mouse S1P1 receptor assessed as cAMP accumulation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Mouse)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50041982(CHEMBL3359522)
Affinity DataEC50:  0.0500nMAssay Description:Agonist activity at mouse S1P1 receptor assessed as cAMP accumulation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSphingosine 1-phosphate receptor 5(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50041983(CHEMBL3359523)
Affinity DataEC50:  19nMAssay Description:Agonist activity at human S1P5 receptor by beta-arrestin recruitment assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSphingosine 1-phosphate receptor 5(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50041982(CHEMBL3359522)
Affinity DataEC50:  47nMAssay Description:Agonist activity at human S1P5 receptor by beta-arrestin recruitment assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSphingosine 1-phosphate receptor 4(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50041983(CHEMBL3359523)
Affinity DataEC50:  85nMAssay Description:Agonist activity at human S1P4 receptor by beta-arrestin recruitment assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSphingosine 1-phosphate receptor 4(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50041982(CHEMBL3359522)
Affinity DataEC50:  8.60E+3nMAssay Description:Agonist activity at human S1P4 receptor by beta-arrestin recruitment assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSphingosine 1-phosphate receptor 3(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50041983(CHEMBL3359523)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human S1P3 receptor by beta-arrestin recruitment assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSphingosine 1-phosphate receptor 3(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50041982(CHEMBL3359522)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human S1P3 receptor by beta-arrestin recruitment assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Rat)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50041982(CHEMBL3359522)
Affinity DataEC50:  0.0720nMAssay Description:Agonist activity at rat S1P1 receptor assessed as cAMP accumulation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSphingosine 1-phosphate receptor 2(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50041982(CHEMBL3359522)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human S1P2 receptor by beta-arrestin recruitment assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50041981(CHEMBL3358955)
Affinity DataEC50:  0.0410nMAssay Description:Agonist activity at human S1P1 receptor assessed as cAMP accumulation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50041980(CHEMBL3359519)
Affinity DataEC50:  0.640nMAssay Description:Agonist activity at human S1P1 receptor assessed as cAMP accumulation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50041980(CHEMBL3359519)
Affinity DataEC50:  0.150nMAssay Description:Agonist activity at human S1P1 receptor assessed as cAMP accumulation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Displayed 1 to 50 (of 71 total ) | Next | Last >>
Jump to: