Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50048802
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rat)
Suntory Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50103634(CL-287389 | FK-235 | Nilvadipine | Nivadipine | SK...)
Affinity DataIC50: 1nMAssay Description:Inhibition of [3H]nitrendipine binding to L-type calcium channels of rat cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2019
Entry Details Article
PubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rat)
Suntory Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50227967(CHEMBL78973)
Affinity DataIC50: 2.10nMAssay Description:Inhibition of [3H]- Nitrendipine binding to L-type calcium channels of rat cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2019
Entry Details Article
PubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rat)
Suntory Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50101817(CHEBI:7565 | Adalat | Adalat Cc | Afeditab Cr | BA...)
Affinity DataIC50: 2.5nMAssay Description:Inhibition of [3H]nitrendipine binding to L-type calcium channels of rat cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2019
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rat)
Suntory Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50101815(CHEBI:7550 | Nicardipine)
Affinity DataIC50: 2.70nMAssay Description:Inhibition of [3H]nitrendipine binding to L-type calcium channels of rat cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2019
Entry Details Article
PubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rat)
Suntory Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50227968(CHEMBL310953)
Affinity DataIC50: 7.10nMAssay Description:Inhibition of [3H]- Nitrendipine binding to L-type calcium channels of rat cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2019
Entry Details Article
PubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rat)
Suntory Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50227969(CV-4093 | CHEMBL312176)
Affinity DataIC50: 8.70nMAssay Description:Inhibition of [3H]- Nitrendipine binding to L-type calcium channels of rat cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2019
Entry Details Article
PubMed