Compile Data Set for Download or QSAR
maximum 50k data
Found 32 Enz. Inhib. hit(s) with all data for entry = 50045400
TargetNociceptin receptor(Homo sapiens (Human))
West Chester University

Curated by ChEMBL
LigandPNGBDBM50060848(CHEMBL3394751)
Affinity DataIC50:  3.90nMAssay Description:Displacement of [125I]-Tyr14-nociceptin from human ORL1 expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
West Chester University

Curated by ChEMBL
LigandPNGBDBM50060837(CHEMBL3394744)
Affinity DataIC50:  4.20nMAssay Description:Displacement of [125I]-Tyr14-nociceptin from human ORL1 expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
West Chester University

Curated by ChEMBL
LigandPNGBDBM50060843(CHEMBL3394748)
Affinity DataIC50:  8nMAssay Description:Displacement of [125I]-Tyr14-nociceptin from human ORL1 expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
West Chester University

Curated by ChEMBL
LigandPNGBDBM50060893(CHEMBL3394753)
Affinity DataIC50:  8.80nMAssay Description:Displacement of [125I]-Tyr14-nociceptin from human ORL1 expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
West Chester University

Curated by ChEMBL
LigandPNGBDBM50060844(CHEMBL3394749)
Affinity DataIC50:  14nMAssay Description:Displacement of [125I]-Tyr14-nociceptin from human ORL1 expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
West Chester University

Curated by ChEMBL
LigandPNGBDBM50060903(CHEMBL3394756)
Affinity DataIC50:  18nMAssay Description:Displacement of [125I]-Tyr14-nociceptin from human ORL1 expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
West Chester University

Curated by ChEMBL
LigandPNGBDBM50060846(CHEMBL3394750)
Affinity DataIC50:  26nMAssay Description:Displacement of [125I]-Tyr14-nociceptin from human ORL1 expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
West Chester University

Curated by ChEMBL
LigandPNGBDBM50060836(CHEMBL3394743)
Affinity DataIC50:  29nMAssay Description:Displacement of [3H]DAMGO from human Mu opioid receptor expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
West Chester University

Curated by ChEMBL
LigandPNGBDBM50060842(CHEMBL3394747)
Affinity DataIC50:  29nMAssay Description:Displacement of [3H]DAMGO from human Mu opioid receptor expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
West Chester University

Curated by ChEMBL
LigandPNGBDBM50060904(CHEMBL3394742)
Affinity DataIC50:  34nMAssay Description:Displacement of [125I]-Tyr14-nociceptin from human ORL1 expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
West Chester University

Curated by ChEMBL
LigandPNGBDBM50060838(CHEMBL3394745)
Affinity DataIC50:  36nMAssay Description:Displacement of [3H]DAMGO from human Mu opioid receptor expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
West Chester University

Curated by ChEMBL
LigandPNGBDBM50060897(CHEMBL3394754)
Affinity DataIC50:  37nMAssay Description:Displacement of [125I]-Tyr14-nociceptin from human ORL1 expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
West Chester University

Curated by ChEMBL
LigandPNGBDBM50060863(CHEMBL3394752)
Affinity DataIC50:  41nMAssay Description:Displacement of [125I]-Tyr14-nociceptin from human ORL1 expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
West Chester University

Curated by ChEMBL
LigandPNGBDBM50060841(CHEMBL3394746)
Affinity DataIC50:  47nMAssay Description:Displacement of [3H]DAMGO from human Mu opioid receptor expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
West Chester University

Curated by ChEMBL
LigandPNGBDBM50060863(CHEMBL3394752)
Affinity DataIC50:  57nMAssay Description:Displacement of [3H]DAMGO from human Mu opioid receptor expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
West Chester University

Curated by ChEMBL
LigandPNGBDBM50060836(CHEMBL3394743)
Affinity DataIC50:  61nMAssay Description:Displacement of [125I]-Tyr14-nociceptin from human ORL1 expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
West Chester University

Curated by ChEMBL
LigandPNGBDBM50060844(CHEMBL3394749)
Affinity DataIC50:  69nMAssay Description:Displacement of [3H]DAMGO from human Mu opioid receptor expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
West Chester University

Curated by ChEMBL
LigandPNGBDBM50060848(CHEMBL3394751)
Affinity DataIC50:  79nMAssay Description:Displacement of [3H]DAMGO from human Mu opioid receptor expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
West Chester University

Curated by ChEMBL
LigandPNGBDBM50060843(CHEMBL3394748)
Affinity DataIC50:  80nMAssay Description:Displacement of [3H]DAMGO from human Mu opioid receptor expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
West Chester University

Curated by ChEMBL
LigandPNGBDBM50060902(CHEMBL3394755)
Affinity DataIC50:  82nMAssay Description:Displacement of [125I]-Tyr14-nociceptin from human ORL1 expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
West Chester University

Curated by ChEMBL
LigandPNGBDBM50060838(CHEMBL3394745)
Affinity DataIC50:  100nMAssay Description:Displacement of [125I]-Tyr14-nociceptin from human ORL1 expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
West Chester University

Curated by ChEMBL
LigandPNGBDBM50060846(CHEMBL3394750)
Affinity DataIC50:  103nMAssay Description:Displacement of [3H]DAMGO from human Mu opioid receptor expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
West Chester University

Curated by ChEMBL
LigandPNGBDBM50060837(CHEMBL3394744)
Affinity DataIC50:  110nMAssay Description:Displacement of [3H]DAMGO from human Mu opioid receptor expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
West Chester University

Curated by ChEMBL
LigandPNGBDBM50060842(CHEMBL3394747)
Affinity DataIC50:  160nMAssay Description:Displacement of [125I]-Tyr14-nociceptin from human ORL1 expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
West Chester University

Curated by ChEMBL
LigandPNGBDBM50060841(CHEMBL3394746)
Affinity DataIC50:  166nMAssay Description:Displacement of [125I]-Tyr14-nociceptin from human ORL1 expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
West Chester University

Curated by ChEMBL
LigandPNGBDBM50060893(CHEMBL3394753)
Affinity DataIC50:  200nMAssay Description:Displacement of [3H]U69,593 from human kappa opioid receptor expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
West Chester University

Curated by ChEMBL
LigandPNGBDBM50060904(CHEMBL3394742)
Affinity DataIC50:  240nMAssay Description:Displacement of [3H]U69,593 from human kappa opioid receptor expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
West Chester University

Curated by ChEMBL
LigandPNGBDBM50060897(CHEMBL3394754)
Affinity DataIC50:  540nMAssay Description:Displacement of [3H]DAMGO from human Mu opioid receptor expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
West Chester University

Curated by ChEMBL
LigandPNGBDBM50060903(CHEMBL3394756)
Affinity DataIC50:  820nMAssay Description:Displacement of [3H]DAMGO from human Mu opioid receptor expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
West Chester University

Curated by ChEMBL
LigandPNGBDBM50060893(CHEMBL3394753)
Affinity DataIC50:  990nMAssay Description:Displacement of [3H]DAMGO from human Mu opioid receptor expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
West Chester University

Curated by ChEMBL
LigandPNGBDBM50060904(CHEMBL3394742)
Affinity DataIC50:  1.19E+3nMAssay Description:Displacement of [3H]DAMGO from human Mu opioid receptor expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
West Chester University

Curated by ChEMBL
LigandPNGBDBM50060902(CHEMBL3394755)
Affinity DataIC50:  2.60E+3nMAssay Description:Displacement of [3H]DAMGO from human Mu opioid receptor expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed