TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Wayne State University
Curated by ChEMBL
Wayne State University
Curated by ChEMBL
Affinity DataKi: 0.710nMAssay Description:Inhibition of [1,2-3H]serotonin reuptake in rat cerebral cortex SERTMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Wayne State University
Curated by ChEMBL
Wayne State University
Curated by ChEMBL
Affinity DataKi: 2.70nMAssay Description:Inhibition of [1,2-3H]serotonin reuptake in rat cerebral cortex SERTMore data for this Ligand-Target Pair
Affinity DataKi: 4.80nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat cerebral cortex NETMore data for this Ligand-Target Pair
Affinity DataKi: 4.90nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat cerebral cortex NETMore data for this Ligand-Target Pair
Affinity DataKi: 5.90nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat cerebral cortex NETMore data for this Ligand-Target Pair
Affinity DataKi: 7.40nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat cerebral cortex NETMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wayne State University
Curated by ChEMBL
Wayne State University
Curated by ChEMBL
Affinity DataKi: 8.90nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat striatum DATMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Wayne State University
Curated by ChEMBL
Wayne State University
Curated by ChEMBL
Affinity DataKi: 9nMAssay Description:Inhibition of [1,2-3H]serotonin reuptake in rat cerebral cortex SERTMore data for this Ligand-Target Pair
Affinity DataKi: 9.30nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat cerebral cortex NETMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat cerebral cortex NETMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wayne State University
Curated by ChEMBL
Wayne State University
Curated by ChEMBL
Affinity DataKi: 13nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat striatum DATMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat cerebral cortex NETMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wayne State University
Curated by ChEMBL
Wayne State University
Curated by ChEMBL
Affinity DataKi: 17nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat striatum DATMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wayne State University
Curated by ChEMBL
Wayne State University
Curated by ChEMBL
Affinity DataKi: 20nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat striatum DATMore data for this Ligand-Target Pair
Affinity DataKi: 25nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat cerebral cortex NETMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wayne State University
Curated by ChEMBL
Wayne State University
Curated by ChEMBL
Affinity DataKi: 26nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat striatum DATMore data for this Ligand-Target Pair
Affinity DataKi: 26nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat cerebral cortex NETMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Wayne State University
Curated by ChEMBL
Wayne State University
Curated by ChEMBL
Affinity DataKi: 27nMAssay Description:Inhibition of [1,2-3H]serotonin reuptake in rat cerebral cortex SERTMore data for this Ligand-Target Pair
Affinity DataKi: 27nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat cerebral cortex NETMore data for this Ligand-Target Pair
Affinity DataKi: 28nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat cerebral cortex NETMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wayne State University
Curated by ChEMBL
Wayne State University
Curated by ChEMBL
Affinity DataKi: 29nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat striatum DATMore data for this Ligand-Target Pair
Affinity DataKi: 29nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat cerebral cortex NETMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wayne State University
Curated by ChEMBL
Wayne State University
Curated by ChEMBL
Affinity DataKi: 29nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat striatum DATMore data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat cerebral cortex NETMore data for this Ligand-Target Pair
Affinity DataKi: 34nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat cerebral cortex NETMore data for this Ligand-Target Pair
Affinity DataKi: 34nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat cerebral cortex NETMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wayne State University
Curated by ChEMBL
Wayne State University
Curated by ChEMBL
Affinity DataKi: 37nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat striatum DATMore data for this Ligand-Target Pair
Affinity DataKi: 38nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat cerebral cortex NETMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Wayne State University
Curated by ChEMBL
Wayne State University
Curated by ChEMBL
Affinity DataKi: 42nMAssay Description:Inhibition of [1,2-3H]serotonin reuptake in rat cerebral cortex SERTMore data for this Ligand-Target Pair
Affinity DataKi: 42nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat cerebral cortex NETMore data for this Ligand-Target Pair
Affinity DataKi: 44nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat cerebral cortex NETMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wayne State University
Curated by ChEMBL
Wayne State University
Curated by ChEMBL
Affinity DataKi: 44nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat striatum DATMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wayne State University
Curated by ChEMBL
Wayne State University
Curated by ChEMBL
Affinity DataKi: 48nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat striatum DATMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wayne State University
Curated by ChEMBL
Wayne State University
Curated by ChEMBL
Affinity DataKi: 52nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat striatum DATMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Wayne State University
Curated by ChEMBL
Wayne State University
Curated by ChEMBL
Affinity DataKi: 54nMAssay Description:Inhibition of [1,2-3H]serotonin reuptake in rat cerebral cortex SERTMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wayne State University
Curated by ChEMBL
Wayne State University
Curated by ChEMBL
Affinity DataKi: 57nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat striatum DATMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wayne State University
Curated by ChEMBL
Wayne State University
Curated by ChEMBL
Affinity DataKi: 59nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat striatum DATMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Wayne State University
Curated by ChEMBL
Wayne State University
Curated by ChEMBL
Affinity DataKi: 64nMAssay Description:Inhibition of [1,2-3H]serotonin reuptake in rat cerebral cortex SERTMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Wayne State University
Curated by ChEMBL
Wayne State University
Curated by ChEMBL
Affinity DataKi: 68nMAssay Description:Inhibition of [1,2-3H]serotonin reuptake in rat cerebral cortex SERTMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wayne State University
Curated by ChEMBL
Wayne State University
Curated by ChEMBL
Affinity DataKi: 82nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat striatum DATMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Wayne State University
Curated by ChEMBL
Wayne State University
Curated by ChEMBL
Affinity DataKi: 107nMAssay Description:Inhibition of [1,2-3H]serotonin reuptake in rat cerebral cortex SERTMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Wayne State University
Curated by ChEMBL
Wayne State University
Curated by ChEMBL
Affinity DataKi: 129nMAssay Description:Inhibition of [1,2-3H]serotonin reuptake in rat cerebral cortex SERTMore data for this Ligand-Target Pair
Affinity DataKi: 152nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat cerebral cortex NETMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wayne State University
Curated by ChEMBL
Wayne State University
Curated by ChEMBL
Affinity DataKi: 167nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat striatum DATMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wayne State University
Curated by ChEMBL
Wayne State University
Curated by ChEMBL
Affinity DataKi: 209nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat striatum DATMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Wayne State University
Curated by ChEMBL
Wayne State University
Curated by ChEMBL
Affinity DataKi: 223nMAssay Description:Inhibition of [1,2-3H]serotonin reuptake in rat cerebral cortex SERTMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wayne State University
Curated by ChEMBL
Wayne State University
Curated by ChEMBL
Affinity DataKi: 234nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat striatum DATMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Wayne State University
Curated by ChEMBL
Wayne State University
Curated by ChEMBL
Affinity DataKi: 258nMAssay Description:Inhibition of [1,2-3H]serotonin reuptake in rat cerebral cortex SERTMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wayne State University
Curated by ChEMBL
Wayne State University
Curated by ChEMBL
Affinity DataKi: 259nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat striatum DATMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Wayne State University
Curated by ChEMBL
Wayne State University
Curated by ChEMBL
Affinity DataKi: 281nMAssay Description:Inhibition of [1,2-3H]serotonin reuptake in rat cerebral cortex SERTMore data for this Ligand-Target Pair