Compile Data Set for Download or QSAR
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Found 33 Enz. Inhib. hit(s) with all data for entry = 50045635
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50072313(CHEMBL3408393)
Affinity DataIC50:  1.70nMAssay Description:Inhibition of CHK1 (unknown origin) using FAM-KKKVSRSGLYRSPSMPENLNRPR-COOH peptide substrate incubated for 1 hr by caliper microfluidic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50072316(CHEMBL3408396)
Affinity DataIC50:  2.60nMAssay Description:Inhibition of CHK1 (unknown origin) using FAM-KKKVSRSGLYRSPSMPENLNRPR-COOH peptide substrate incubated for 1 hr by caliper microfluidic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50072315(CHEMBL3408395)
Affinity DataIC50:  3.5nMAssay Description:Inhibition of CHK1 (unknown origin) using FAM-KKKVSRSGLYRSPSMPENLNRPR-COOH peptide substrate incubated for 1 hr by caliper microfluidic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50072314(CHEMBL3408394)
Affinity DataIC50:  4.60nMAssay Description:Inhibition of CHK1 (unknown origin) using FAM-KKKVSRSGLYRSPSMPENLNRPR-COOH peptide substrate incubated for 1 hr by caliper microfluidic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50072312(CHEMBL3408392)
Affinity DataIC50:  7.60nMAssay Description:Inhibition of CHK1 (unknown origin) using FAM-KKKVSRSGLYRSPSMPENLNRPR-COOH peptide substrate incubated for 1 hr by caliper microfluidic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50072281(CHEMBL3408382)
Affinity DataIC50:  9.90nMAssay Description:Inhibition of CHK1 (unknown origin) using FAM-KKKVSRSGLYRSPSMPENLNRPR-COOH peptide substrate incubated for 1 hr by caliper microfluidic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM17054((2S,3R,4R,6R,18R)-18-hydroxy-3-methoxy-2-methyl-4-...)
Affinity DataIC50:  9.90nMAssay Description:Inhibition of CHK1 (unknown origin) using FAM-KKKVSRSGLYRSPSMPENLNRPR-COOH peptide substrate incubated for 1 hr by caliper microfluidic assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50072310(CHEMBL3408390)
Affinity DataIC50:  12nMAssay Description:Inhibition of CHK1 (unknown origin) using FAM-KKKVSRSGLYRSPSMPENLNRPR-COOH peptide substrate incubated for 1 hr by caliper microfluidic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50072309(CHEMBL3408389)
Affinity DataIC50:  13nMAssay Description:Inhibition of CHK1 (unknown origin) using FAM-KKKVSRSGLYRSPSMPENLNRPR-COOH peptide substrate incubated for 1 hr by caliper microfluidic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50072308(CHEMBL3408388)
Affinity DataIC50:  14nMAssay Description:Inhibition of CHK1 (unknown origin) using FAM-KKKVSRSGLYRSPSMPENLNRPR-COOH peptide substrate incubated for 1 hr by caliper microfluidic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50072307(CHEMBL3408387)
Affinity DataIC50:  16nMAssay Description:Inhibition of CHK1 (unknown origin) using FAM-KKKVSRSGLYRSPSMPENLNRPR-COOH peptide substrate incubated for 1 hr by caliper microfluidic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50072306(CHEMBL3408386)
Affinity DataIC50:  17nMAssay Description:Inhibition of CHK1 (unknown origin) using FAM-KKKVSRSGLYRSPSMPENLNRPR-COOH peptide substrate incubated for 1 hr by caliper microfluidic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50072305(CHEMBL3408385)
Affinity DataIC50:  19nMAssay Description:Inhibition of CHK1 (unknown origin) using FAM-KKKVSRSGLYRSPSMPENLNRPR-COOH peptide substrate incubated for 1 hr by caliper microfluidic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50072304(CHEMBL3408384)
Affinity DataIC50:  20nMAssay Description:Inhibition of CHK1 (unknown origin) using FAM-KKKVSRSGLYRSPSMPENLNRPR-COOH peptide substrate incubated for 1 hr by caliper microfluidic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50072303(CHEMBL3408383)
Affinity DataIC50:  22nMAssay Description:Inhibition of CHK1 (unknown origin) using FAM-KKKVSRSGLYRSPSMPENLNRPR-COOH peptide substrate incubated for 1 hr by caliper microfluidic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50072311(CHEMBL3408391)
Affinity DataIC50:  23nMAssay Description:Inhibition of CHK1 (unknown origin) using FAM-KKKVSRSGLYRSPSMPENLNRPR-COOH peptide substrate incubated for 1 hr by caliper microfluidic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50072280(CHEMBL3408381)
Affinity DataIC50:  27nMAssay Description:Inhibition of CHK1 (unknown origin) using FAM-KKKVSRSGLYRSPSMPENLNRPR-COOH peptide substrate incubated for 1 hr by caliper microfluidic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50072313(CHEMBL3408393)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibition of human ERG assessed as reduction in channel current expressed in HEK cells by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50072316(CHEMBL3408396)
Affinity DataIC50:  3.40E+3nMAssay Description:Inhibition of human ERG assessed as reduction in channel current expressed in HEK cells by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50072315(CHEMBL3408395)
Affinity DataIC50:  4.60E+3nMAssay Description:Inhibition of human ERG assessed as reduction in channel current expressed in HEK cells by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50072314(CHEMBL3408394)
Affinity DataIC50:  5.70E+3nMAssay Description:Inhibition of human ERG assessed as reduction in channel current expressed in HEK cells by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50072312(CHEMBL3408392)
Affinity DataIC50:  6.80E+3nMAssay Description:Inhibition of human ERG assessed as reduction in channel current expressed in HEK cells by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50072281(CHEMBL3408382)
Affinity DataIC50:  7.60E+3nMAssay Description:Inhibition of human ERG assessed as reduction in channel current expressed in HEK cells by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50072309(CHEMBL3408389)
Affinity DataIC50:  8.40E+3nMAssay Description:Inhibition of human ERG assessed as reduction in channel current expressed in HEK cells by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50072310(CHEMBL3408390)
Affinity DataIC50:  8.40E+3nMAssay Description:Inhibition of human ERG assessed as reduction in channel current expressed in HEK cells by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50072308(CHEMBL3408388)
Affinity DataIC50:  9.30E+3nMAssay Description:Inhibition of human ERG assessed as reduction in channel current expressed in HEK cells by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50072307(CHEMBL3408387)
Affinity DataIC50:  1.04E+4nMAssay Description:Inhibition of human ERG assessed as reduction in channel current expressed in HEK cells by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50072306(CHEMBL3408386)
Affinity DataIC50:  1.15E+4nMAssay Description:Inhibition of human ERG assessed as reduction in channel current expressed in HEK cells by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50072305(CHEMBL3408385)
Affinity DataIC50:  1.76E+4nMAssay Description:Inhibition of human ERG assessed as reduction in channel current expressed in HEK cells by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50072304(CHEMBL3408384)
Affinity DataIC50:  2.87E+4nMAssay Description:Inhibition of human ERG assessed as reduction in channel current expressed in HEK cells by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50072303(CHEMBL3408383)
Affinity DataIC50:  3.26E+4nMAssay Description:Inhibition of human ERG assessed as reduction in channel current expressed in HEK cells by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50072311(CHEMBL3408391)
Affinity DataIC50:  4.55E+4nMAssay Description:Inhibition of human ERG assessed as reduction in channel current expressed in HEK cells by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50072280(CHEMBL3408381)
Affinity DataIC50:  4.84E+4nMAssay Description:Inhibition of human ERG assessed as reduction in channel current expressed in HEK cells by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed