TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Umr Cnrs-Universit£
Curated by ChEMBL
Umr Cnrs-Universit£
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Inhibition of B-Raf V600E mutant (unknown origin) assessed as inhibition of phosphorylation of peptide substrateMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Umr Cnrs-Universit£
Curated by ChEMBL
Umr Cnrs-Universit£
Curated by ChEMBL
Affinity DataIC50: 31nMAssay Description:Inhibition of B-Raf V600E mutant (unknown origin) assessed as inhibition of phosphorylation of peptide substrateMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Umr Cnrs-Universit£
Curated by ChEMBL
Umr Cnrs-Universit£
Curated by ChEMBL
Affinity DataIC50: <100nMAssay Description:Inhibition of B-Raf V600E mutant (unknown origin) assessed as inhibition of phosphorylation of peptide substrateMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Umr Cnrs-Universit£
Curated by ChEMBL
Umr Cnrs-Universit£
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of wild type B-Raf (unknown origin) assessed as inhibition of phosphorylation of peptide substrateMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Umr Cnrs-Universit£
Curated by ChEMBL
Umr Cnrs-Universit£
Curated by ChEMBL
Affinity DataIC50: <100nMAssay Description:Inhibition of B-Raf V600E mutant (unknown origin) assessed as inhibition of phosphorylation of peptide substrateMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Umr Cnrs-Universit£
Curated by ChEMBL
Umr Cnrs-Universit£
Curated by ChEMBL
Affinity DataIC50: 160nMAssay Description:Inhibition of wild type B-Raf (unknown origin) assessed as inhibition of phosphorylation of peptide substrateMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Umr Cnrs-Universit£
Curated by ChEMBL
Umr Cnrs-Universit£
Curated by ChEMBL
Affinity DataIC50: <800nMAssay Description:Inhibition of B-Raf V600E mutant in human A375 cells assessed as phosphorylation of ERKMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Umr Cnrs-Universit£
Curated by ChEMBL
Umr Cnrs-Universit£
Curated by ChEMBL
Affinity DataIC50: <1.00E+3nMAssay Description:Inhibition of B-Raf V600E mutant in human A375 cells assessed as phosphorylation of ERKMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Umr Cnrs-Universit£
Curated by ChEMBL
Umr Cnrs-Universit£
Curated by ChEMBL
Affinity DataIC50: <1.00E+3nMAssay Description:Inhibition of B-Raf V600E mutant in human A375 cells assessed as phosphorylation of ERKMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Umr Cnrs-Universit£
Curated by ChEMBL
Umr Cnrs-Universit£
Curated by ChEMBL
Affinity DataKd: 1.41E+3nMAssay Description:Binding affinity to B-Raf V600E mutant (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Umr Cnrs-Universit£
Curated by ChEMBL
Umr Cnrs-Universit£
Curated by ChEMBL
Affinity DataKd: 62nMAssay Description:Binding affinity to wild type B-Raf (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Umr Cnrs-Universit£
Curated by ChEMBL
Umr Cnrs-Universit£
Curated by ChEMBL
Affinity DataKd: 100nMAssay Description:Binding affinity to wild type B-Raf (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Umr Cnrs-Universit£
Curated by ChEMBL
Umr Cnrs-Universit£
Curated by ChEMBL
Affinity DataKd: 400nMAssay Description:Binding affinity to wild type B-Raf (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Umr Cnrs-Universit£
Curated by ChEMBL
Umr Cnrs-Universit£
Curated by ChEMBL
Affinity DataKd: 690nMAssay Description:Binding affinity to wild type B-Raf (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Umr Cnrs-Universit£
Curated by ChEMBL
Umr Cnrs-Universit£
Curated by ChEMBL
Affinity DataKd: 140nMAssay Description:Binding affinity to B-Raf V600E mutant (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Umr Cnrs-Universit£
Curated by ChEMBL
Umr Cnrs-Universit£
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Activation of tumorigenic wild type B-Raf in human IPC-298 cells with Ras mutation assessed as phosphorylation of ERKMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Umr Cnrs-Universit£
Curated by ChEMBL
Umr Cnrs-Universit£
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Activation of tumorigenic wild type B-Raf in human IPC-298 cells with Ras mutation assessed as phosphorylation of ERKMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Umr Cnrs-Universit£
Curated by ChEMBL
Umr Cnrs-Universit£
Curated by ChEMBL
Affinity DataKd: 130nMAssay Description:Binding affinity to B-Raf V600E mutant (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Umr Cnrs-Universit£
Curated by ChEMBL
Umr Cnrs-Universit£
Curated by ChEMBL
Affinity DataKd: 550nMAssay Description:Binding affinity to B-Raf V600E mutant (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Umr Cnrs-Universit£
Curated by ChEMBL
Umr Cnrs-Universit£
Curated by ChEMBL
Affinity DataEC50: <500nMAssay Description:Activation of tumorigenic wild type B-Raf in human IPC-298 cells with Ras mutation assessed as phosphorylation of ERKMore data for this Ligand-Target Pair