Compile Data Set for Download or QSAR
maximum 50k data
Found 13 Enz. Inhib. hit(s) with all data for entry = 50045476
TargetEndothelin-1 receptor(RAT)
Southeast University

Curated by ChEMBL
LigandPNGBDBM50064000(CHEMBL3400988)
Affinity DataIC50:  3.30nMAssay Description:Displacement of PD156707 from rat ETA receptor after 1 hr by Lowry methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
Southeast University

Curated by ChEMBL
LigandPNGBDBM50063998(CHEMBL3400989)
Affinity DataIC50:  3.90nMAssay Description:Displacement of [125I]ET-1 from rat ETA receptor after 1 hr by Lowry methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
Southeast University

Curated by ChEMBL
LigandPNGBDBM50061101(4-(1,1-Dimethylethyl)-N-(6-(2-hydroxyethoxy)-5-(2-...)
Affinity DataIC50:  4.70nMAssay Description:Displacement of [125I]ET-1 from rat ETA receptor after 1 hr by Lowry methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
Southeast University

Curated by ChEMBL
LigandPNGBDBM50063997(CHEMBL3400996)
Affinity DataIC50:  5.5nMAssay Description:Displacement of [125I]ET-1 from rat ETA receptor after 1 hr by Lowry methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
Southeast University

Curated by ChEMBL
LigandPNGBDBM50063999(CHEMBL3400984)
Affinity DataIC50:  12nMAssay Description:Displacement of [125I]ET-1 from rat ETA receptor after 1 hr by Lowry methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
Southeast University

Curated by ChEMBL
LigandPNGBDBM50063996(CHEMBL3400998)
Affinity DataIC50:  19nMAssay Description:Displacement of [125I]ET-1 from rat ETA receptor after 1 hr by Lowry methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
Southeast University

Curated by ChEMBL
LigandPNGBDBM50029352(CHEMBL336033 | [(5S,8S,11R,14S,16aR)-8-(1H-Indol-3...)
Affinity DataIC50:  28nMAssay Description:Displacement of [125I]ET-1 from rat ETA receptor after 1 hr by Lowry methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(RAT)
Southeast University

Curated by ChEMBL
LigandPNGBDBM50061101(4-(1,1-Dimethylethyl)-N-(6-(2-hydroxyethoxy)-5-(2-...)
Affinity DataIC50:  95nMAssay Description:Displacement of [125I]ET-1 from rat ETB receptor after 1 hr by Lowry methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(RAT)
Southeast University

Curated by ChEMBL
LigandPNGBDBM50063997(CHEMBL3400996)
Affinity DataIC50:  183nMAssay Description:Displacement of [125I]ET-1 from rat ETB receptor after 1 hr by Lowry methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(RAT)
Southeast University

Curated by ChEMBL
LigandPNGBDBM50063998(CHEMBL3400989)
Affinity DataIC50:  198nMAssay Description:Displacement of [125I]ET-1 from rat ETB receptor after 1 hr by Lowry methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(RAT)
Southeast University

Curated by ChEMBL
LigandPNGBDBM50064000(CHEMBL3400988)
Affinity DataIC50:  260nMAssay Description:Displacement of S6c from rat ETB receptor after 1 hr by Lowry methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(RAT)
Southeast University

Curated by ChEMBL
LigandPNGBDBM50063996(CHEMBL3400998)
Affinity DataIC50:  340nMAssay Description:Displacement of [125I]ET-1 from rat ETB receptor after 1 hr by Lowry methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(RAT)
Southeast University

Curated by ChEMBL
LigandPNGBDBM50063999(CHEMBL3400984)
Affinity DataIC50:  453nMAssay Description:Displacement of [125I]ET-1 from rat ETB receptor after 1 hr by Lowry methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed