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Found 26 Enz. Inhib. hit(s) with all data for entry = 50001717
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50017543((6aR,9R,10aR)-9-Methylsulfanylmethyl-7-propyl-4,6,...)
Affinity DataIC50:  1.60nMAssay Description:Inhibitory activity against Dopamine receptor D2 in rat corpus striatum using [3H]-Apomorphine as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(BOVINE)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50017543((6aR,9R,10aR)-9-Methylsulfanylmethyl-7-propyl-4,6,...)
Affinity DataIC50:  48nMAssay Description:Inhibitory activity against Dopamine receptor D2 in calf corpus striatum using [3H]-Spiperone as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50017539(CHEMBL80414 | Propyl-(4,5,6,7-tetrahydro-2H-indazo...)
Affinity DataIC50:  65nMAssay Description:Inhibitory activity against dopamine receptor D2 in rat corpus striatum using [3H]-Apomorphine as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50017542(CHEMBL80437 | Phenethyl-propyl-(4,5,6,7-tetrahydro...)
Affinity DataIC50:  140nMAssay Description:Inhibitory activity against dopamine receptor D2 in rat corpus striatum using [3H]-Apomorphine as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50017547(CHEMBL421512 | Propyl-(4,5,6,7-tetrahydro-2H-indaz...)
Affinity DataIC50:  160nMAssay Description:Inhibitory activity against dopamine receptor D2 in rat corpus striatum using [3H]-Apomorphine as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50017550(CHEMBL76399 | N*6*-Propyl-4,5,6,7-tetrahydro-benzo...)
Affinity DataIC50:  280nMAssay Description:Inhibitory activity against dopamine receptor D2 in rat corpus striatum using [3H]-Apomorphine as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50017551((3-Methylsulfanyl-propyl)-propyl-(4,5,6,7-tetrahyd...)
Affinity DataIC50:  310nMAssay Description:Inhibitory activity against dopamine receptor D2 in rat corpus striatum using [3H]-Apomorphine as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50017541(Butyl-propyl-(4,5,6,7-tetrahydro-2H-indazol-5-yl)-...)
Affinity DataIC50:  330nMAssay Description:Inhibitory activity against Dopamine receptor D2 in rat corpus striatum using [3H]-Apomorphine as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50017544(CHEMBL77421 | Ethyl-(4,5,6,7-tetrahydro-2H-indazol...)
Affinity DataIC50:  610nMAssay Description:Inhibitory activity against dopamine receptor D2 in rat corpus striatum using [3H]-Apomorphine as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(BOVINE)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50017550(CHEMBL76399 | N*6*-Propyl-4,5,6,7-tetrahydro-benzo...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibitory activity against dopamine receptor D2 in calf corpus striatum using [3H]-Spiperone as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(BOVINE)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50017542(CHEMBL80437 | Phenethyl-propyl-(4,5,6,7-tetrahydro...)
Affinity DataIC50:  1.06E+3nMAssay Description:Inhibitory activity against dopamine receptor D2 in calf corpus striatum using [3H]-Spiperone as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50017546(CHEMBL311225 | Methyl-propyl-(4,5,6,7-tetrahydro-2...)
Affinity DataIC50:  1.23E+3nMAssay Description:Inhibitory activity against Dopamine receptor D2 in rat corpus striatum using [3H]-Apomorphine as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(BOVINE)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50017547(CHEMBL421512 | Propyl-(4,5,6,7-tetrahydro-2H-indaz...)
Affinity DataIC50:  1.41E+3nMAssay Description:Inhibitory activity against dopamine receptor D2 in calf corpus striatum using [3H]-Spiperone as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50017540((3-Methylsulfanyl-propyl)-(4,5,6,7-tetrahydro-2H-i...)
Affinity DataIC50:  2.03E+3nMAssay Description:Inhibitory activity against dopamine receptor D2 in rat corpus striatum using [3H]-Apomorphine as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(BOVINE)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50017551((3-Methylsulfanyl-propyl)-propyl-(4,5,6,7-tetrahyd...)
Affinity DataIC50:  3.99E+3nMAssay Description:Inhibitory activity against dopamine receptor D2 in calf corpus striatum using [3H]-Spiperone as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(BOVINE)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50017546(CHEMBL311225 | Methyl-propyl-(4,5,6,7-tetrahydro-2...)
Affinity DataIC50:  8.33E+3nMAssay Description:Inhibitory activity against Dopamine receptor D2 in calf corpus striatum using [3H]-Spiperone as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50017545((4,5,6,7-Tetrahydro-2H-indazol-5-yl)-(2-thiophen-2...)
Affinity DataIC50:  9.16E+3nMAssay Description:Inhibitory activity against dopamine receptor D2 in rat corpus striatum using [3H]-Apomorphine as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(BOVINE)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50017549(Butyl-(4,5,6,7-tetrahydro-2H-indazol-5-yl)-amine |...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibitory activity against dopamine receptor D2 in calf corpus striatum using [3H]-Spiperone as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(BOVINE)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50017548(CHEMBL81400 | Phenethyl-(4,5,6,7-tetrahydro-2H-ind...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibitory activity against dopamine receptor D2 in calf corpus striatum using [3H]-Spiperone as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(BOVINE)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50017541(Butyl-propyl-(4,5,6,7-tetrahydro-2H-indazol-5-yl)-...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibitory activity against Dopamine receptor D2 in calf corpus striatum using [3H]-Spiperone as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(BOVINE)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50017545((4,5,6,7-Tetrahydro-2H-indazol-5-yl)-(2-thiophen-2...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibitory activity against dopamine receptor D2 in calf corpus striatum using [3H]-Spiperone as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(BOVINE)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50017540((3-Methylsulfanyl-propyl)-(4,5,6,7-tetrahydro-2H-i...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibitory activity against dopamine receptor D2 in calf corpus striatum using [3H]-Spiperone as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50017549(Butyl-(4,5,6,7-tetrahydro-2H-indazol-5-yl)-amine |...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibitory activity against dopamine receptor D2 in rat corpus striatum using [3H]-Apomorphine as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(BOVINE)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50017544(CHEMBL77421 | Ethyl-(4,5,6,7-tetrahydro-2H-indazol...)
Affinity DataIC50:  1.16E+4nMAssay Description:Inhibitory activity against dopamine receptor D2 in calf corpus striatum using [3H]-Spiperone as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(BOVINE)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50017539(CHEMBL80414 | Propyl-(4,5,6,7-tetrahydro-2H-indazo...)
Affinity DataIC50:  1.52E+4nMAssay Description:Inhibitory activity against dopamine receptor D2 in calf corpus striatum using [3H]-Spiperone as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50017548(CHEMBL81400 | Phenethyl-(4,5,6,7-tetrahydro-2H-ind...)
Affinity DataIC50:  1.53E+4nMAssay Description:Inhibitory activity against dopamine receptor D2 in rat corpus striatum using [3H]-Apomorphine as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed