Compile Data Set for Download or QSAR
maximum 50k data
Found 15 Enz. Inhib. hit(s) with all data for entry = 50045461
TargetCollagenase 3(Homo sapiens (Human))
University Of Catania

Curated by ChEMBL
LigandPNGBDBM50359900(CHEMBL260125)
Affinity DataIC50:  158nMAssay Description:Inhibition of MMP13 catalytic domain (unknown origin) assessed as reduction in hydrolysis of Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 substrate measured f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
University Of Catania

Curated by ChEMBL
LigandPNGBDBM50359901(CHEMBL260886)
Affinity DataIC50:  3.15E+3nMAssay Description:Inhibition of MMP3 catalytic domain (unknown origin) assessed as reduction in hydrolysis of Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 substrate measured fo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
University Of Catania

Curated by ChEMBL
LigandPNGBDBM50359898(CHEMBL412064)
Affinity DataIC50:  5.06E+3nMAssay Description:Inhibition of MMP3 catalytic domain (unknown origin) assessed as reduction in hydrolysis of Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 substrate measured fo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
University Of Catania

Curated by ChEMBL
LigandPNGBDBM50359897(CHEMBL264164)
Affinity DataIC50:  6.19E+3nMAssay Description:Inhibition of MMP3 catalytic domain (unknown origin) assessed as reduction in hydrolysis of Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 substrate measured fo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
University Of Catania

Curated by ChEMBL
LigandPNGBDBM50359900(CHEMBL260125)
Affinity DataIC50:  1.04E+4nMAssay Description:Inhibition of MMP3 catalytic domain (unknown origin) assessed as reduction in hydrolysis of Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 substrate measured fo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
University Of Catania

Curated by ChEMBL
LigandPNGBDBM50359899(CHEMBL263909)
Affinity DataIC50:  2.50E+4nMAssay Description:Inhibition of MMP13 catalytic domain (unknown origin) assessed as reduction in hydrolysis of Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 substrate measured f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
University Of Catania

Curated by ChEMBL
LigandPNGBDBM50063580(CHEMBL3398611)
Affinity DataIC50:  2.69E+4nMAssay Description:Inhibition of MMP13 catalytic domain (unknown origin) assessed as reduction in hydrolysis of Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 substrate measured f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
University Of Catania

Curated by ChEMBL
LigandPNGBDBM50359903(CHEMBL409502)
Affinity DataIC50:  3.20E+4nMAssay Description:Inhibition of MMP13 catalytic domain (unknown origin) assessed as reduction in hydrolysis of Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 substrate measured f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
University Of Catania

Curated by ChEMBL
LigandPNGBDBM50359894(CHEMBL407151)
Affinity DataIC50:  4.30E+4nMAssay Description:Inhibition of MMP3 catalytic domain (unknown origin) assessed as reduction in hydrolysis of Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 substrate measured fo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
University Of Catania

Curated by ChEMBL
LigandPNGBDBM50359896(CHEMBL410649)
Affinity DataIC50:  5.59E+4nMAssay Description:Inhibition of MMP13 catalytic domain (unknown origin) assessed as reduction in hydrolysis of Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 substrate measured f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
University Of Catania

Curated by ChEMBL
LigandPNGBDBM50359895(CHEMBL261267)
Affinity DataIC50:  5.59E+4nMAssay Description:Inhibition of MMP13 catalytic domain (unknown origin) assessed as reduction in hydrolysis of Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 substrate measured f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
University Of Catania

Curated by ChEMBL
LigandPNGBDBM50359894(CHEMBL407151)
Affinity DataIC50:  6.40E+4nMAssay Description:Inhibition of MMP13 catalytic domain (unknown origin) assessed as reduction in hydrolysis of Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 substrate measured f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
University Of Catania

Curated by ChEMBL
LigandPNGBDBM50359899(CHEMBL263909)
Affinity DataIC50:  6.50E+4nMAssay Description:Inhibition of MMP3 catalytic domain (unknown origin) assessed as reduction in hydrolysis of Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 substrate measured fo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
University Of Catania

Curated by ChEMBL
LigandPNGBDBM50359897(CHEMBL264164)
Affinity DataIC50:  8.94E+4nMAssay Description:Inhibition of MMP13 catalytic domain (unknown origin) assessed as reduction in hydrolysis of Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 substrate measured f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
University Of Catania

Curated by ChEMBL
LigandPNGBDBM50063579(CHEMBL3398610)
Affinity DataIC50:  9.74E+4nMAssay Description:Inhibition of MMP3 catalytic domain (unknown origin) assessed as reduction in hydrolysis of Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 substrate measured fo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed