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Report error Found 23 Enz. Inhib. hit(s) with all data for entry = 6775
TargetAdenosine receptor A1(Rat)
North-West University

LigandPNGBDBM50393880(CHEMBL2158245)
Affinity DataKi:  369nMAssay Description:For the A2a receptor binding study, the incubation contained 10 mg of the original tissue weight of the striatal membranes, 4 nM [3H]NECA, 50 nM CPA,...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A1(Rat)
North-West University

LigandPNGBDBM50393884(CHEMBL2158241)
Affinity DataKi:  548nMAssay Description:For the A2a receptor binding study, the incubation contained 10 mg of the original tissue weight of the striatal membranes, 4 nM [3H]NECA, 50 nM CPA,...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A1(Rat)
North-West University

LigandPNGBDBM50393884(CHEMBL2158241)
Affinity DataKi:  595nMAssay Description:For the A2a receptor binding study, the incubation contained 10 mg of the original tissue weight of the striatal membranes, 4 nM [3H]NECA, 50 nM CPA,...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A1(Rat)
North-West University

LigandPNGBDBM50393879(CHEMBL2158246)
Affinity DataKi:  648nMAssay Description:For the A2a receptor binding study, the incubation contained 10 mg of the original tissue weight of the striatal membranes, 4 nM [3H]NECA, 50 nM CPA,...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A1(Rat)
North-West University

LigandPNGBDBM50393876(CHEMBL2158249)
Affinity DataKi:  649nMAssay Description:For the A2a receptor binding study, the incubation contained 10 mg of the original tissue weight of the striatal membranes, 4 nM [3H]NECA, 50 nM CPA,...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A1(Rat)
North-West University

LigandPNGBDBM50393882(CHEMBL2158243)
Affinity DataKi:  676nMAssay Description:For the A2a receptor binding study, the incubation contained 10 mg of the original tissue weight of the striatal membranes, 4 nM [3H]NECA, 50 nM CPA,...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A2a(Rat)
North-West University

LigandPNGBDBM50393884(CHEMBL2158241)
Affinity DataKi:  980nMAssay Description:For the A2a receptor binding study, the incubation contained 10 mg of the original tissue weight of the striatal membranes, 4 nM [3H]NECA, 50 nM CPA,...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A1(Rat)
North-West University

LigandPNGBDBM50393880(CHEMBL2158245)
Affinity DataKi:  1.73E+3nMAssay Description:For the A2a receptor binding study, the incubation contained 10 mg of the original tissue weight of the striatal membranes, 4 nM [3H]NECA, 50 nM CPA,...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A1(Rat)
North-West University

LigandPNGBDBM50393876(CHEMBL2158249)
Affinity DataKi:  1.88E+3nMAssay Description:For the A2a receptor binding study, the incubation contained 10 mg of the original tissue weight of the striatal membranes, 4 nM [3H]NECA, 50 nM CPA,...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A1(Rat)
North-West University

LigandPNGBDBM50350641(CHEMBL342357)
Affinity DataKi:  4.67E+3nMAssay Description:For the A2a receptor binding study, the incubation contained 10 mg of the original tissue weight of the striatal membranes, 4 nM [3H]NECA, 50 nM CPA,...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A1(Rat)
North-West University

LigandPNGBDBM50393881(CHEMBL2158244)
Affinity DataKi:  6.30E+3nMAssay Description:For the A2a receptor binding study, the incubation contained 10 mg of the original tissue weight of the striatal membranes, 4 nM [3H]NECA, 50 nM CPA,...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A1(Rat)
North-West University

LigandPNGBDBM50393879(CHEMBL2158246)
Affinity DataKi:  7.72E+3nMAssay Description:For the A2a receptor binding study, the incubation contained 10 mg of the original tissue weight of the striatal membranes, 4 nM [3H]NECA, 50 nM CPA,...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A1(Rat)
North-West University

LigandPNGBDBM50334284(5-Benzyloxyisatin | CHEMBL1642670)
Affinity DataKi:  9.79E+3nMAssay Description:For the A2a receptor binding study, the incubation contained 10 mg of the original tissue weight of the striatal membranes, 4 nM [3H]NECA, 50 nM CPA,...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A2a(Rat)
North-West University

LigandPNGBDBM50393881(CHEMBL2158244)
Affinity DataKi:  1.27E+4nMAssay Description:For the A2a receptor binding study, the incubation contained 10 mg of the original tissue weight of the striatal membranes, 4 nM [3H]NECA, 50 nM CPA,...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A2a(Rat)
North-West University

LigandPNGBDBM50393876(CHEMBL2158249)
Affinity DataKi:  1.70E+4nMAssay Description:For the A2a receptor binding study, the incubation contained 10 mg of the original tissue weight of the striatal membranes, 4 nM [3H]NECA, 50 nM CPA,...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A1(Rat)
North-West University

LigandPNGBDBM50393881(CHEMBL2158244)
Affinity DataKi:  3.67E+4nMAssay Description:For the A2a receptor binding study, the incubation contained 10 mg of the original tissue weight of the striatal membranes, 4 nM [3H]NECA, 50 nM CPA,...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAmine oxidase [flavin-containing] B(Human)
North-West University

LigandPNGBDBM50393881(CHEMBL2158244)
Affinity DataIC50:  290nMpH: 7.4Assay Description:The enzymatic reactions were carried out at pH 7.4 (K2HPO4/KH2PO4 100 mM, made isotonic with KCl) to a final volume of 500 無. The reactions containe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAmine oxidase [flavin-containing] B(Human)
North-West University

LigandPNGBDBM50393877(CHEMBL2158248)
Affinity DataIC50:  443nMpH: 7.4Assay Description:The enzymatic reactions were carried out at pH 7.4 (K2HPO4/KH2PO4 100 mM, made isotonic with KCl) to a final volume of 500 無. The reactions containe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAmine oxidase [flavin-containing] B(Human)
North-West University

LigandPNGBDBM50393883(CHEMBL2158242)
Affinity DataIC50:  460nMpH: 7.4Assay Description:The enzymatic reactions were carried out at pH 7.4 (K2HPO4/KH2PO4 100 mM, made isotonic with KCl) to a final volume of 500 無. The reactions containe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAmine oxidase [flavin-containing] B(Human)
North-West University

LigandPNGBDBM50393878(CHEMBL2158247)
Affinity DataIC50:  1.39E+3nMpH: 7.4Assay Description:The enzymatic reactions were carried out at pH 7.4 (K2HPO4/KH2PO4 100 mM, made isotonic with KCl) to a final volume of 500 無. The reactions containe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAmine oxidase [flavin-containing] B(Human)
North-West University

LigandPNGBDBM50393884(CHEMBL2158241)
Affinity DataIC50:  1.88E+3nMpH: 7.4Assay Description:The enzymatic reactions were carried out at pH 7.4 (K2HPO4/KH2PO4 100 mM, made isotonic with KCl) to a final volume of 500 無. The reactions containe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAmine oxidase [flavin-containing] B(Human)
North-West University

LigandPNGBDBM50393876(CHEMBL2158249)
Affinity DataIC50:  3.90E+3nMpH: 7.4Assay Description:The enzymatic reactions were carried out at pH 7.4 (K2HPO4/KH2PO4 100 mM, made isotonic with KCl) to a final volume of 500 無. The reactions containe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAmine oxidase [flavin-containing] B(Human)
North-West University

LigandPNGBDBM50393879(CHEMBL2158246)
Affinity DataIC50:  9.17E+3nMpH: 7.4Assay Description:The enzymatic reactions were carried out at pH 7.4 (K2HPO4/KH2PO4 100 mM, made isotonic with KCl) to a final volume of 500 無. The reactions containe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed