Compile Data Set for Download or QSAR
Report error Found 15 Enz. Inhib. hit(s) with all data for entry = 50045734
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
The University of Arizona

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50078775BDBM50078775(CHEMBL3416149)
Affinity DataIC50: 15nMAssay Description:Inhibition of FLT3 (unknown origin) using FAM-EPLYWSFPA as substrate preincubated for 60 mins followed by substrate addition by microfluidics assay i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2016
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
The University of Arizona

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50078840BDBM50078840(CHEMBL3416157)
Affinity DataIC50: 16nMAssay Description:Inhibition of FLT3 (unknown origin) using FAM-EPLYWSFPA as substrate preincubated for 60 mins followed by substrate addition by microfluidics assay i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2016
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
The University of Arizona

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50300690BDBM50300690(CHEMBL576982 | N-(5-tert-Butyl-isoxazol-3-yl)-N'-{...)
Affinity DataIC50: 39nMAssay Description:Inhibition of FLT3 (unknown origin) using FAM-EPLYWSFPA as substrate preincubated for 60 mins followed by substrate addition by microfluidics assay i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2016
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
The University of Arizona

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50078836BDBM50078836(CHEMBL3416153)
Affinity DataIC50: 41nMAssay Description:Inhibition of FLT3 (unknown origin) using FAM-EPLYWSFPA as substrate preincubated for 60 mins followed by substrate addition by microfluidics assay i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2016
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
The University of Arizona

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50078774BDBM50078774(CHEMBL3416147)
Affinity DataIC50: 51nMAssay Description:Inhibition of FLT3 (unknown origin) using FAM-EPLYWSFPA as substrate preincubated for 60 mins followed by substrate addition by microfluidics assay i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2016
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
The University of Arizona

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50078843BDBM50078843(CHEMBL3416161)
Affinity DataIC50: 78nMAssay Description:Inhibition of FLT3 (unknown origin) using FAM-EPLYWSFPA as substrate preincubated for 60 mins followed by substrate addition by microfluidics assay i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2016
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
The University of Arizona

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50078780BDBM50078780(CHEMBL3416152)
Affinity DataIC50: 160nMAssay Description:Inhibition of FLT3 (unknown origin) using FAM-EPLYWSFPA as substrate preincubated for 60 mins followed by substrate addition by microfluidics assay i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2016
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
The University of Arizona

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50078777BDBM50078777(CHEMBL3416151)
Affinity DataIC50: 190nMAssay Description:Inhibition of FLT3 (unknown origin) using FAM-EPLYWSFPA as substrate preincubated for 60 mins followed by substrate addition by microfluidics assay i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2016
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
The University of Arizona

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50078837BDBM50078837(CHEMBL3416154)
Affinity DataIC50: 230nMAssay Description:Inhibition of FLT3 (unknown origin) using FAM-EPLYWSFPA as substrate preincubated for 60 mins followed by substrate addition by microfluidics assay i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2016
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
The University of Arizona

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50078839BDBM50078839(CHEMBL3416156)
Affinity DataIC50: 300nMAssay Description:Inhibition of FLT3 (unknown origin) using FAM-EPLYWSFPA as substrate preincubated for 60 mins followed by substrate addition by microfluidics assay i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2016
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
The University of Arizona

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50078841BDBM50078841(CHEMBL3416159)
Affinity DataIC50: 430nMAssay Description:Inhibition of FLT3 (unknown origin) using FAM-EPLYWSFPA as substrate preincubated for 60 mins followed by substrate addition by microfluidics assay i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2016
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
The University of Arizona

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50078842BDBM50078842(CHEMBL3416160)
Affinity DataIC50: 440nMAssay Description:Inhibition of FLT3 (unknown origin) using FAM-EPLYWSFPA as substrate preincubated for 60 mins followed by substrate addition by microfluidics assay i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2016
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
The University of Arizona

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50078776BDBM50078776(CHEMBL3416150)
Affinity DataIC50: 470nMAssay Description:Inhibition of FLT3 (unknown origin) using FAM-EPLYWSFPA as substrate preincubated for 60 mins followed by substrate addition by microfluidics assay i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2016
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
The University of Arizona

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50078773BDBM50078773(CHEMBL3416141)
Affinity DataIC50: 480nMAssay Description:Inhibition of FLT3 (unknown origin) using FAM-EPLYWSFPA as substrate preincubated for 60 mins followed by substrate addition by microfluidics assay i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2016
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
The University of Arizona

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50078838BDBM50078838(CHEMBL3416155)
Affinity DataIC50: 550nMAssay Description:Inhibition of FLT3 (unknown origin) using FAM-EPLYWSFPA as substrate preincubated for 60 mins followed by substrate addition by microfluidics assay i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2016
Entry Details Article
PubMed