Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50046064
LigandPNGBDBM50324735(CHEMBL568150 | AS605240 | (5E)-5-(QUINOXALIN-6-YLM...)
Affinity DataIC50: 9nMAssay Description:Inhibition of human recombinant GST-tagged PI3Kgamma incubated for 180 mins using [33P]gamma-ATP by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2016
Entry Details Article
PubMed
TargetAldo-keto reductase family 1 member B1(Human)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50334175(2-(2,4-dioxo-5-(4-phenoxybenzylidene)thiazolidin-3...)
Affinity DataIC50: 130nMAssay Description:Inhibition of aldose reductase (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2016
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50093478(CHEMBL3585578)
Affinity DataIC50: 190nMAssay Description:Agonist activity at PPARgamma (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2016
Entry Details Article
PubMed
LigandPNGBDBM50403077(CHEMBL2216899)
Affinity DataIC50: 250nMAssay Description:Inhibition of human recombinant GST-tagged PI3Kgamma incubated for 180 mins using [33P]gamma-ATP by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2016
Entry Details Article
PubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Human)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50093477(CHEMBL3585579)
Affinity DataIC50: 690nMAssay Description:Inhibition of GST-tagged PTP1B (unknown origin) by pNPP catalysis based colorimetric high throughput assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2016
Entry Details Article
PubMed
TargetAldo-keto reductase family 1 member B1(Human)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50093476(CHEMBL1645385)
Affinity DataIC50: 6.14E+3nMAssay Description:Inhibition of aldose reductase (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2016
Entry Details Article
PubMed