Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) with all data for entry = 50046007 Sort by
TargetGlycogen synthase kinase-3 beta(Human)
Chiba University

Curated by ChEMBL
LigandPNGBDBM50090908(CHEMBL1774404 | CHEBI:67291)
Affinity DataIC50: 3.00E+3nMAssay Description:Activation of GSK-3beta in HEK293 cells assessed as suppression of TCF/beta-catenin transcriptional activity after 24 hrs by SuperTOPFlash reporter g...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Chiba University

Curated by ChEMBL
LigandPNGBDBM50090907(CHEMBL444160 | CHEBI:66041)
Affinity DataIC50: 6.80E+3nMAssay Description:Activation of GSK-3beta in HEK293 cells assessed as suppression of TCF/beta-catenin transcriptional activity after 24 hrs by SuperTOPFlash reporter g...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Chiba University

Curated by ChEMBL
LigandPNGBDBM50090909(CHEMBL3120496)
Affinity DataIC50: 1.16E+4nMAssay Description:Activation of GSK-3beta in HEK293 cells assessed as suppression of TCF/beta-catenin transcriptional activity after 24 hrs by SuperTOPFlash reporter g...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed