Affinity DataKi: 2.40nMAssay Description:Binding affinity to human histamine H4 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 4.5nMAssay Description:Binding affinity to human histamine H4 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 4.80nMAssay Description:Binding affinity to human histamine H4 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 5.30nMAssay Description:Displacement of [3H]histamine from mouse recombinant histamine H4 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Binding affinity to guinea pig histamine H4 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 6.20nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in HEK293T cellsMore data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Binding affinity to histamine H4 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Displacement of [3H]histamine from human recombinant histamine H4 receptorMore data for this Ligand-Target Pair
TargetHistamine H4 receptor(Rattus norvegicus (rat))
Janssen Research And Development
Curated by ChEMBL
Janssen Research And Development
Curated by ChEMBL
Affinity DataKi: 12nMAssay Description:Displacement of [3H]histamine from rat histamine H4 receptor expressed in HEK293T cellsMore data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Binding affinity to histamine H3 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 21nMAssay Description:Displacement of [3H]histamine from mouse histamine H4 receptor expressed in HEK293T cellsMore data for this Ligand-Target Pair
Affinity DataKi: 42nMAssay Description:Binding affinity to mouse histamine H4 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 123nMAssay Description:Displacement of [3H]histamine from guinea pig histamine H4 receptor expressed in HEK293T cellsMore data for this Ligand-Target Pair
TargetHistamine H4 receptor(Rattus norvegicus (rat))
Janssen Research And Development
Curated by ChEMBL
Janssen Research And Development
Curated by ChEMBL
Affinity DataKi: 136nMAssay Description:Binding affinity to rat histamine H4 receptorMore data for this Ligand-Target Pair
TargetHistamine H4 receptor(Rattus norvegicus (rat))
Janssen Research And Development
Curated by ChEMBL
Janssen Research And Development
Curated by ChEMBL
Affinity DataKi: 188nMAssay Description:Displacement of [3H]histamine from rat recombinant histamine H4 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 306nMAssay Description:Displacement of [3H]histamine from guinea pig recombinant histamine H4 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.11E+3nMAssay Description:Binding affinity to human histamine H4 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 5.00E+3nMAssay Description:Binding affinity to histamine H2 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 6.00E+3nMAssay Description:Binding affinity to histamine H1 receptor (unknown origin)More data for this Ligand-Target Pair