Compile Data Set for Download or QSAR
Report error Found 15 Enz. Inhib. hit(s) with all data for entry = 50046020
TargetNischarin(Rat)
University of Camerino

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50091345BDBM50091345(CHEMBL2092861)
Affinity DataKi:  1.10nMAssay Description:Displacement of [125I]-p-iodoclonidin from I1-imidazoline receptor in rat PC12 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2016
Entry Details Article
PubMed
TargetNischarin(Rat)
University of Camerino

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50091347BDBM50091347(CHEMBL71429)
Affinity DataKi:  5nMAssay Description:Displacement of [125I]-p-iodoclonidin from I1-imidazoline receptor in rat PC12 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2016
Entry Details Article
PubMed
TargetNischarin(Rat)
University of Camerino

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50091336BDBM50091336(CHEMBL3582266)
Affinity DataKi:  13nMAssay Description:Displacement of [125I]-p-iodoclonidin from I1-imidazoline receptor in rat PC12 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2016
Entry Details Article
PubMed
TargetNischarin(Rat)
University of Camerino

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50091338BDBM50091338(CHEMBL3582264)
Affinity DataKi:  23nMAssay Description:Displacement of [125I]-p-iodoclonidin from I1-imidazoline receptor in rat PC12 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2016
Entry Details Article
PubMed
TargetNischarin(Rat)
University of Camerino

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50091341BDBM50091341(CHEMBL3582261)
Affinity DataKi:  63nMAssay Description:Displacement of [125I]-p-iodoclonidin from I1-imidazoline receptor in rat PC12 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2016
Entry Details Article
PubMed
TargetNischarin(Rat)
University of Camerino

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50091342BDBM50091342(CHEMBL3582260)
Affinity DataKi:  98nMAssay Description:Displacement of [125I]-p-iodoclonidin from I1-imidazoline receptor in rat PC12 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2016
Entry Details Article
PubMed
TargetNischarin(Rat)
University of Camerino

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50412250BDBM50412250(CHEMBL128168)
Affinity DataKi:  126nMAssay Description:Displacement of [125I]-p-iodoclonidin from I1-imidazoline receptor in rat PC12 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2016
Entry Details Article
PubMed
TargetNischarin(Rat)
University of Camerino

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50091344BDBM50091344(CHEMBL3582258)
Affinity DataKi:  155nMAssay Description:Displacement of [125I]-p-iodoclonidin from I1-imidazoline receptor in rat PC12 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2016
Entry Details Article
PubMed
TargetNischarin(Rat)
University of Camerino

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50091335BDBM50091335(CHEMBL3582267)
Affinity DataKi:  195nMAssay Description:Displacement of [125I]-p-iodoclonidin from I1-imidazoline receptor in rat PC12 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2016
Entry Details Article
PubMed
TargetNischarin(Rat)
University of Camerino

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50412260BDBM50412260(CHEMBL273485)
Affinity DataKi:  309nMAssay Description:Displacement of [125I]-p-iodoclonidin from I1-imidazoline receptor in rat PC12 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2016
Entry Details Article
PubMed
TargetNischarin(Rat)
University of Camerino

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50091340BDBM50091340(CHEMBL3582262)
Affinity DataKi: <1.00E+3nMAssay Description:Displacement of [125I]-p-iodoclonidin from I1-imidazoline receptor in rat PC12 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2016
Entry Details Article
PubMed
TargetNischarin(Rat)
University of Camerino

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50091339BDBM50091339(CHEMBL3582263)
Affinity DataKi: <1.00E+3nMAssay Description:Displacement of [125I]-p-iodoclonidin from I1-imidazoline receptor in rat PC12 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2016
Entry Details Article
PubMed
TargetNischarin(Rat)
University of Camerino

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50091337BDBM50091337(CHEMBL3582265)
Affinity DataKi:  1.05E+3nMAssay Description:Displacement of [125I]-p-iodoclonidin from I1-imidazoline receptor in rat PC12 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2016
Entry Details Article
PubMed
TargetNischarin(Rat)
University of Camerino

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50091343BDBM50091343(CHEMBL3582259)
Affinity DataKi:  2.24E+3nMAssay Description:Displacement of [125I]-p-iodoclonidin from I1-imidazoline receptor in rat PC12 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2016
Entry Details Article
PubMed
TargetNischarin(Rat)
University of Camerino

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50091346BDBM50091346(CHEMBL1907832)
Affinity DataKi:  6.31E+3nMAssay Description:Displacement of [125I]-p-iodoclonidin from I1-imidazoline receptor in rat PC12 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2016
Entry Details Article
PubMed