Compile Data Set for Download or QSAR
maximum 50k data
Found 39 Enz. Inhib. hit(s) with all data for entry = 50046101
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50094910(CHEMBL3589475)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of HTRF binding to N-terminal His-tagged BRD2(2) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide and Cryptate-labe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50094913(CHEMBL3589482)
Affinity DataIC50:  9.00E+3nMAssay Description:Inhibition of HTRF binding to N-terminal His-tagged BRD4(1) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide and Cryptate-labe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50094887(CHEMBL3589478)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of HTRF binding to N-terminal His-tagged BRD2(2) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide and Cryptate-labe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50094896(CHEMBL3589487)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of HTRF binding to N-terminal His-tagged BRD2(2) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide and Cryptate-labe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50094888(CHEMBL3589479)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of HTRF binding to N-terminal His-tagged BRD2(2) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide and Cryptate-labe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50094899(CHEMBL3589471)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibition of HTRF binding to N-terminal His-tagged BRD2(2) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide and Cryptate-labe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50094908(CHEMBL3589473)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibition of HTRF binding to N-terminal His-tagged BRD2(2) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide and Cryptate-labe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50094914(CHEMBL3589483)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibition of HTRF binding to N-terminal His-tagged BRD4(1) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide and Cryptate-labe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50094899(CHEMBL3589471)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibition of HTRF binding to N-terminal His-tagged BRD4(1) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide and Cryptate-labe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50094898(CHEMBL3589470)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibition of HTRF binding to N-terminal His-tagged BRD4(1) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide and Cryptate-labe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50094897(CHEMBL3589469)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibition of HTRF binding to N-terminal His-tagged BRD4(1) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide and Cryptate-labe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50094900(CHEMBL3589472)
Affinity DataIC50:  1.40E+4nMAssay Description:Inhibition of HTRF binding to N-terminal His-tagged BRD4(1) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide and Cryptate-labe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50094908(CHEMBL3589473)
Affinity DataIC50:  1.60E+4nMAssay Description:Inhibition of HTRF binding to N-terminal His-tagged BRD4(1) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide and Cryptate-labe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50094909(CHEMBL3589474)
Affinity DataIC50:  1.80E+4nMAssay Description:Inhibition of HTRF binding to N-terminal His-tagged BRD4(1) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide and Cryptate-labe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50094894(CHEMBL3589485)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibition of HTRF binding to N-terminal His-tagged BRD2(2) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide and Cryptate-labe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50094886(CHEMBL3589468)
Affinity DataIC50:  2.20E+4nMAssay Description:Inhibition of HTRF binding to N-terminal His-tagged BRD2(2) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide and Cryptate-labe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50094897(CHEMBL3589469)
Affinity DataIC50:  2.30E+4nMAssay Description:Inhibition of HTRF binding to N-terminal His-tagged BRD2(2) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide and Cryptate-labe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50094898(CHEMBL3589470)
Affinity DataIC50:  2.40E+4nMAssay Description:Inhibition of HTRF binding to N-terminal His-tagged BRD2(2) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide and Cryptate-labe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50094911(CHEMBL3589476)
Affinity DataIC50:  2.50E+4nMAssay Description:Inhibition of HTRF binding to N-terminal His-tagged BRD4(1) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide and Cryptate-labe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50094910(CHEMBL3589475)
Affinity DataIC50:  2.50E+4nMAssay Description:Inhibition of HTRF binding to N-terminal His-tagged BRD4(1) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide and Cryptate-labe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50094911(CHEMBL3589476)
Affinity DataIC50:  2.50E+4nMAssay Description:Inhibition of HTRF binding to N-terminal His-tagged BRD2(2) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide and Cryptate-labe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50094915(CHEMBL3589484)
Affinity DataIC50:  2.50E+4nMAssay Description:Inhibition of HTRF binding to N-terminal His-tagged BRD4(1) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide and Cryptate-labe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50094886(CHEMBL3589468)
Affinity DataIC50:  2.60E+4nMAssay Description:Inhibition of HTRF binding to N-terminal His-tagged BRD4(1) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide and Cryptate-labe...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50094894(CHEMBL3589485)
Affinity DataIC50:  2.60E+4nMAssay Description:Inhibition of HTRF binding to N-terminal His-tagged BRD4(1) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide and Cryptate-labe...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50094909(CHEMBL3589474)
Affinity DataIC50:  2.60E+4nMAssay Description:Inhibition of HTRF binding to N-terminal His-tagged BRD2(2) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide and Cryptate-labe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50094916(CHEMBL3589486)
Affinity DataIC50:  2.90E+4nMAssay Description:Inhibition of HTRF binding to N-terminal His-tagged BRD4(1) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide and Cryptate-labe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50094912(CHEMBL3589477)
Affinity DataIC50:  3.40E+4nMAssay Description:Inhibition of HTRF binding to N-terminal His-tagged BRD4(1) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide and Cryptate-labe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50094887(CHEMBL3589478)
Affinity DataIC50:  4.00E+4nMAssay Description:Inhibition of HTRF binding to N-terminal His-tagged BRD4(1) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide and Cryptate-labe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50094888(CHEMBL3589479)
Affinity DataIC50:  4.40E+4nMAssay Description:Inhibition of HTRF binding to N-terminal His-tagged BRD4(1) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide and Cryptate-labe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50094896(CHEMBL3589487)
Affinity DataIC50:  4.40E+4nMAssay Description:Inhibition of HTRF binding to N-terminal His-tagged BRD4(1) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide and Cryptate-labe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50094889(CHEMBL3589480)
Affinity DataIC50:  4.60E+4nMAssay Description:Inhibition of HTRF binding to N-terminal His-tagged BRD4(1) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide and Cryptate-labe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50094917(CHEMBL3589488)
Affinity DataIC50:  4.70E+4nMAssay Description:Inhibition of HTRF binding to N-terminal His-tagged BRD4(1) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide and Cryptate-labe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50094918(CHEMBL3589489)
Affinity DataIC50:  4.90E+4nMAssay Description:Inhibition of HTRF binding to N-terminal His-tagged BRD4(1) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide and Cryptate-labe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50094889(CHEMBL3589480)
Affinity DataIC50:  4.90E+4nMAssay Description:Inhibition of HTRF binding to N-terminal His-tagged BRD2(2) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide and Cryptate-labe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50094890(CHEMBL3589481)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of HTRF binding to N-terminal His-tagged BRD2(2) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide and Cryptate-labe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50094900(CHEMBL3589472)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of HTRF binding to N-terminal His-tagged BRD2(2) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide and Cryptate-labe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50094912(CHEMBL3589477)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of HTRF binding to N-terminal His-tagged BRD2(2) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide and Cryptate-labe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50094890(CHEMBL3589481)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of HTRF binding to N-terminal His-tagged BRD4(1) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide and Cryptate-labe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50094919(CHEMBL3589490)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of HTRF binding to N-terminal His-tagged BRD4(1) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide and Cryptate-labe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed