BindingDB PrimarySearch

Found 15 Enz. Inhib. hit(s) with all data for entry = 50046324

Dual specificity tyrosine-phosphorylation-regulated kinase 2(Homo sapiens (Human))
India Academy Of Scientific & Innovative Research (Acsir)

Curated by ChEMBL

BDBM50105913(CHEMBL3597991)

IC50: 40nMAssay Description:Inhibition of human recombinant GST-fused Dyrk2 expressed in Escherichia coli using Woodtide as substrate after 15 mins by P81 membrane assay in pres...More data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
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Dual specificity tyrosine-phosphorylation-regulated kinase 1B(Homo sapiens (Human))
India Academy Of Scientific & Innovative Research (Acsir)

Curated by ChEMBL

BDBM50105913(CHEMBL3597991)

IC50: 70nMAssay Description:Inhibition of human recombinant Dyrk1B using Woodtide as substrate after 15 mins by P81 membrane assay in presence of [33P]-g-ATPMore data for this Ligand-Target Pair

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Dual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
India Academy Of Scientific & Innovative Research (Acsir)

Curated by ChEMBL

BDBM100152(7-methoxy-1-methyl-9H-beta-carboline;hydrochloride...)

IC50: 80nMAssay Description:Inhibition of Dyrk1A (unknown origin) using dynatide 3 as substrate after 10 mins by P81 membrane assay in presence of [33P]-g-ATPMore data for this Ligand-Target Pair

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3D Structure (crystal)

Dual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
India Academy Of Scientific & Innovative Research (Acsir)

Curated by ChEMBL

BDBM50105913(CHEMBL3597991)

IC50: 100nMAssay Description:Inhibition of human recombinant His6-tagged Dyrk1A expressed in Escherichia coli using Woodtide as substrate after 15 mins by P81 membrane assay in p...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
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Dual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
India Academy Of Scientific & Innovative Research (Acsir)

Curated by ChEMBL

BDBM50445253(CHEMBL1232500)

IC50: 240nMAssay Description:Inhibition of Dyrk1A (unknown origin)More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
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3D Structure (crystal)

Dual specificity tyrosine-phosphorylation-regulated kinase 1A(RAT)
India Academy Of Scientific & Innovative Research (Acsir)

Curated by ChEMBL

BDBM50070942((-)-Epigallocatechin gallate | (-)-Epigallocatechi...)

IC50: 330nMAssay Description:Inhibition of rat Dyrk1A using Woodtide as substrate after 40 mins by P81 membrane assay in presence of [33P]-g-ATPMore data for this Ligand-Target Pair

PDB Reactome pathway
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Dual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
India Academy Of Scientific & Innovative Research (Acsir)

Curated by ChEMBL

BDBM50105912(CHEMBL3133762)

IC50: 500nMAssay Description:Inhibition of Dyrk1A (unknown origin) using Woodtide as substrate after 30 mins by P81 membrane assay in presence of [33P]-g-ATPMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
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Dual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
India Academy Of Scientific & Innovative Research (Acsir)

Curated by ChEMBL

BDBM50105918(CHEMBL3426272)

IC50: 530nMAssay Description:Inhibition of Dyrk1A (unknown origin) using Woodtide as substrate after 30 mins by P81 membrane assay in presence of [33P]-g-ATPMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

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Dual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
India Academy Of Scientific & Innovative Research (Acsir)

Curated by ChEMBL

BDBM50105916(CHEMBL3133768)

IC50: 830nMAssay Description:Inhibition of Dyrk1A (unknown origin) using Woodtide as substrate after 30 mins by P81 membrane assay in presence of [33P]-g-ATPMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
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Dual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
India Academy Of Scientific & Innovative Research (Acsir)

Curated by ChEMBL

BDBM50026622(CHEMBL408982)

IC50: 930nMAssay Description:Inhibition of Dyrk1A (unknown origin)More data for this Ligand-Target Pair

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Dual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
India Academy Of Scientific & Innovative Research (Acsir)

Curated by ChEMBL

BDBM50105914(CHEMBL3133776)

IC50: 1.30E+3nMAssay Description:Inhibition of Dyrk1A (unknown origin) using Woodtide as substrate after 30 mins by P81 membrane assay in presence of [33P]-g-ATPMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
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Details Article PubMed

Dual specificity tyrosine-phosphorylation-regulated kinase 2(Homo sapiens (Human))
India Academy Of Scientific & Innovative Research (Acsir)

Curated by ChEMBL

BDBM50105912(CHEMBL3133762)

IC50: 1.40E+3nMAssay Description:Inhibition of Dyrk2 (unknown origin) using Woodtide as substrate after 30 mins by P81 membrane assay in presence of [33P]-g-ATPMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

CHEMBL PC cid PC sid Similars

Details Article PubMed

Dual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
India Academy Of Scientific & Innovative Research (Acsir)

Curated by ChEMBL

BDBM50105917(CHEMBL3133771)

IC50: 1.80E+3nMAssay Description:Inhibition of Dyrk1A (unknown origin) using Woodtide as substrate after 30 mins by P81 membrane assay in presence of [33P]-g-ATPMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
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Dual specificity tyrosine-phosphorylation-regulated kinase 3(Homo sapiens (Human))
India Academy Of Scientific & Innovative Research (Acsir)

Curated by ChEMBL

BDBM50105912(CHEMBL3133762)

IC50: 2.20E+3nMAssay Description:Inhibition of Dyrk3 (unknown origin) using Woodtide as substrate after 30 mins by P81 membrane assay in presence of [33P]-g-ATPMore data for this Ligand-Target Pair

PDB KEGG
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Dual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
India Academy Of Scientific & Innovative Research (Acsir)

Curated by ChEMBL

BDBM50105915(CHEMBL3133767)

IC50: 3.10E+3nMAssay Description:Inhibition of Dyrk1A (unknown origin) using Woodtide as substrate after 30 mins by P81 membrane assay in presence of [33P]-g-ATPMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

CHEMBL PC cid PC sid Similars

Details Article PubMed