Compile Data Set for Download or QSAR
Report error Found 72 Enz. Inhib. hit(s) with all data for entry = 50022525
TargetNeutrophil elastase(Human)TBA
LigandPNGBDBM50652827(CHEMBL5661917)
Affinity DataIC50: 0.0240nMAssay Description:Inhibition of human neutrophil elastase using MeOSuc-AAPV-MCA as substrate measured at 60 mins interval for up to several hrs by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetNeutrophil elastase(Human)TBA
LigandPNGBDBM50120437(CHEMBL3617973 | US12415819, Compound 54)
Affinity DataIC50: 0.0650nMAssay Description:Inhibition of human neutrophil elastase using MeOSuc-AAPV-MCA as substrate measured at 60 mins interval for up to several hrs by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetNeutrophil elastase(Human)TBA
LigandPNGBDBM50120437(CHEMBL3617973 | US12415819, Compound 54)
Affinity DataKi:  0.0800nMAssay Description:Competitive inhibition of human neutrophil elastase using varying levels of MeOSuc-AAPV-MCA as substrate measured at 60 mins interval for up to sever...More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetNeutrophil elastase(Human)TBA
LigandPNGBDBM50652828(CHEMBL5661855)
Affinity DataIC50: 0.25nMAssay Description:Inhibition of human neutrophil elastase using MeOSuc-AAPV-MCA as substrate measured at 60 mins interval for up to several hrs by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetNeutrophil elastase(Human)TBA
LigandPNGBDBM50120436(CHEMBL3617972)
Affinity DataIC50: 0.540nMAssay Description:Inhibition of human neutrophil elastase using MeOSuc-AAPV-MCA as substrate measured at 60 mins interval for up to several hrs by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetNeutrophil elastase(Human)TBA
LigandPNGBDBM50652826(CHEMBL5661860)
Affinity DataIC50: 0.600nMAssay Description:Inhibition of human neutrophil elastase using MeOSuc-AAPV-MCA as substrate measured at 60 mins interval for up to several hrs by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetNeutrophil elastase(Human)TBA
LigandPNGBDBM50652821(CHEMBL5661868)
Affinity DataIC50: 1nMAssay Description:Inhibition of human neutrophil elastase using MeOSuc-AAPV-MCA as substrate measured at 60 mins interval for up to several hrs by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetNeutrophil elastase(Human)TBA
LigandPNGBDBM50652817(CHEMBL5661928)
Affinity DataIC50: 1nMAssay Description:Inhibition of human neutrophil elastase using MeOSuc-AAPV-MCA as substrate measured at 60 mins interval for up to several hrs by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetNeutrophil elastase(Human)TBA
LigandPNGBDBM50652825(CHEMBL5661871)
Affinity DataIC50: 1.60nMAssay Description:Inhibition of human neutrophil elastase using MeOSuc-AAPV-MCA as substrate measured at 60 mins interval for up to several hrs by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetNeutrophil elastase(Human)TBA
LigandPNGBDBM50652818(CHEMBL5661863)
Affinity DataIC50: 2.10nMAssay Description:Inhibition of human neutrophil elastase using MeOSuc-AAPV-MCA as substrate measured at 60 mins interval for up to several hrs by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetNeutrophil elastase(Human)TBA
LigandPNGBDBM50120425(CHEMBL3617969)
Affinity DataIC50: 3.5nMAssay Description:Inhibition of human neutrophil elastase using MeOSuc-AAPV-MCA as substrate measured at 60 mins interval for up to several hrs by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetNeutrophil elastase(Human)TBA
LigandPNGBDBM50652819(CHEMBL1738716)
Affinity DataIC50: 4.30nMAssay Description:Inhibition of human neutrophil elastase using MeOSuc-AAPV-MCA as substrate measured at 60 mins interval for up to several hrs by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetNeutrophil elastase(Human)TBA
LigandPNGBDBM50652822(CHEMBL5661856)
Affinity DataIC50: 4.70nMAssay Description:Inhibition of human neutrophil elastase using MeOSuc-AAPV-MCA as substrate measured at 60 mins interval for up to several hrs by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetNeutrophil elastase(Human)TBA
LigandPNGBDBM50652824(CHEMBL5661846)
Affinity DataIC50: 5nMAssay Description:Inhibition of human neutrophil elastase using MeOSuc-AAPV-MCA as substrate measured at 60 mins interval for up to several hrs by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In Depth
Date in BDB:
TBA
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetNeutrophil elastase(Mouse)TBA
LigandPNGBDBM50120437(CHEMBL3617973 | US12415819, Compound 54)
Affinity DataKi:  6nMAssay Description:Competitive inhibition of mouse neutrophil elastase using varying levels of MeOSuc-AAPV-MCA as substrate measured at 60 mins interval for up to sever...More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetNeutrophil elastase(Human)TBA
LigandPNGBDBM50652820(CHEMBL5661879)
Affinity DataIC50: 13nMAssay Description:Inhibition of human neutrophil elastase using MeOSuc-AAPV-MCA as substrate measured at 60 mins interval for up to several hrs by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetNeutrophil elastase(Human)TBA
LigandPNGBDBM50120426(CHEMBL3617968)
Affinity DataKi:  15nMAssay Description:Competitive inhibition of human neutrophil elastase using varying levels of MeOSuc-AAPV-MCA as substrate measured at 60 mins interval for up to sever...More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetNeutrophil elastase(Human)TBA
LigandPNGBDBM50120426(CHEMBL3617968)
Affinity DataIC50: 20nMAssay Description:Inhibition of human neutrophil elastase using MeOSuc-AAPV-MCA as substrate measured at 60 mins interval for up to several hrs by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetNeutrophil elastase(Human)TBA
LigandPNGBDBM50652811(CHEMBL5661905)
Affinity DataIC50: 20nMAssay Description:Inhibition of human neutrophil elastase using MeOSuc-AAPV-MCA as substrate measured at 60 mins interval for up to several hrs by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetNeutrophil elastase(Human)TBA
LigandPNGBDBM50652815(CHEMBL5661897)
Affinity DataIC50: 20nMAssay Description:Inhibition of human neutrophil elastase using MeOSuc-AAPV-MCA as substrate measured at 60 mins interval for up to several hrs by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetNeutrophil elastase(Human)TBA
LigandPNGBDBM50652823(CHEMBL5661882)
Affinity DataIC50: 25nMAssay Description:Inhibition of human neutrophil elastase using MeOSuc-AAPV-MCA as substrate measured at 60 mins interval for up to several hrs by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetNeutrophil elastase(Human)TBA
LigandPNGBDBM50652816(CHEMBL5661864)
Affinity DataIC50: 27nMAssay Description:Inhibition of human neutrophil elastase using MeOSuc-AAPV-MCA as substrate measured at 60 mins interval for up to several hrs by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetNeutrophil elastase(Human)TBA
LigandPNGBDBM50652812(CHEMBL5661832)
Affinity DataIC50: 40nMAssay Description:Inhibition of human neutrophil elastase using MeOSuc-AAPV-MCA as substrate measured at 60 mins interval for up to several hrs by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetNeutrophil elastase(Human)TBA
LigandPNGBDBM50652813(CHEMBL5661875)
Affinity DataIC50: 50nMAssay Description:Inhibition of human neutrophil elastase using MeOSuc-AAPV-MCA as substrate measured at 60 mins interval for up to several hrs by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetNeutrophil elastase(Human)TBA
LigandPNGBDBM50652814(CHEMBL5661851)
Affinity DataIC50: 70nMAssay Description:Inhibition of human neutrophil elastase using MeOSuc-AAPV-MCA as substrate measured at 60 mins interval for up to several hrs by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetNeutrophil elastase(Human)TBA
LigandPNGBDBM50120437(CHEMBL3617973 | US12415819, Compound 54)
Affinity DataIC50: 140nMAssay Description:Inhibition of human neutrophil elastase using MeOSuc-AAPV-MCA as substrate measured at 60 mins interval for up to several hrs in presence of hydrogen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetNeutrophil elastase(Human)TBA
LigandPNGBDBM50652810(CHEMBL5661893)
Affinity DataIC50: 200nMAssay Description:Inhibition of human neutrophil elastase using MeOSuc-AAPV-MCA as substrate measured at 60 mins interval for up to several hrs by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetNeutrophil elastase(Human)TBA
LigandPNGBDBM50652809(CHEMBL5661839)
Affinity DataIC50: 200nMAssay Description:Inhibition of human neutrophil elastase using MeOSuc-AAPV-MCA as substrate measured at 60 mins interval for up to several hrs by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetNeutrophil elastase(Human)TBA
LigandPNGBDBM50652807(CHEMBL5661903)
Affinity DataIC50: 200nMAssay Description:Inhibition of human neutrophil elastase using MeOSuc-AAPV-MCA as substrate measured at 60 mins interval for up to several hrs by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetNeutrophil elastase(Mouse)TBA
LigandPNGBDBM50120426(CHEMBL3617968)
Affinity DataKi:  700nMAssay Description:Competitive inhibition of mouse neutrophil elastase using varying levels of MeOSuc-AAPV-MCA as substrate measured at 60 mins interval for up to sever...More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetNeutrophil elastase(Human)TBA
LigandPNGBDBM50487991(CHEMBL5275929)
Affinity DataIC50: 900nMAssay Description:Inhibition of human neutrophil elastase using MeOSuc-AAPV-MCA as substrate measured at 60 mins interval for up to several hrs by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetNeutrophil elastase(Human)TBA
LigandPNGBDBM50652808(CHEMBL5661854)
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of human neutrophil elastase using MeOSuc-AAPV-MCA as substrate measured at 60 mins interval for up to several hrs by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetCoagulation factor VII(Human)TBA
LigandPNGBDBM50120426(CHEMBL3617968)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of FVIIa (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetCoagulation factor X(Human)TBA
LigandPNGBDBM50120437(CHEMBL3617973 | US12415819, Compound 54)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of FXa (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetCoagulation factor X(Human)TBA
LigandPNGBDBM50120426(CHEMBL3617968)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of FXa (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProthrombin(Human)TBA
LigandPNGBDBM50120437(CHEMBL3617973 | US12415819, Compound 54)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of thrombin (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetCoagulation factor XI(Human)TBA
LigandPNGBDBM50120426(CHEMBL3617968)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of FXIa (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetCoagulation factor IX(Human)TBA
LigandPNGBDBM50120437(CHEMBL3617973 | US12415819, Compound 54)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of FIXa (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetCoagulation factor IX(Human)TBA
LigandPNGBDBM50120426(CHEMBL3617968)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of FIXa (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetCoagulation factor VII(Human)TBA
LigandPNGBDBM50120437(CHEMBL3617973 | US12415819, Compound 54)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of FVIIa (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetPlasminogen(Human)TBA
LigandPNGBDBM50120437(CHEMBL3617973 | US12415819, Compound 54)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of plasmin (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetPlasminogen(Human)TBA
LigandPNGBDBM50120426(CHEMBL3617968)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of plasmin (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetCoagulation factor XI(Human)TBA
LigandPNGBDBM50120437(CHEMBL3617973 | US12415819, Compound 54)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of FXIa (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetKallikrein-1(Human)TBA
LigandPNGBDBM50120426(CHEMBL3617968)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of kallikrein-1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProlyl endopeptidase FAP(Human)TBA
LigandPNGBDBM50120437(CHEMBL3617973 | US12415819, Compound 54)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of FAP (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProlyl endopeptidase FAP(Human)TBA
LigandPNGBDBM50120426(CHEMBL3617968)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of FAP (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50120437(CHEMBL3617973 | US12415819, Compound 54)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of urokinase (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetKallikrein-5(Human)TBA
LigandPNGBDBM50120426(CHEMBL3617968)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of kallikrein-5 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetKallikrein-4(Human)TBA
LigandPNGBDBM50120437(CHEMBL3617973 | US12415819, Compound 54)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of kallikrein-4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetKallikrein-4(Human)TBA
LigandPNGBDBM50120426(CHEMBL3617968)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of kallikrein-4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
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