Compile Data Set for Download or QSAR
maximum 50k data
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 50047158
TargetCREB-binding protein(Human)
University of Z£Rich

Curated by ChEMBL
LigandPNGBDBM50150909(CHEMBL3774461)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of human N-terminal His-tagged KDM4A (1 to 359 residues) expressed in Escherichia coli using biotin-H3K9me3 as substrate preincubated for ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCREB-binding protein(Human)
University of Z£Rich

Curated by ChEMBL
LigandPNGBDBM50443249(Ischemin)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of human N-terminal His-tagged KDM4A (1 to 359 residues) expressed in Escherichia coli using biotin-H3K9me3 as substrate preincubated for ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedPDB3D3D Structure (crystal)

TargetCREB-binding protein(Human)
University of Z£Rich

Curated by ChEMBL
LigandPNGBDBM50150939(CHEMBL3775960)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of human N-terminal His-tagged KDM4A (1 to 359 residues) expressed in Escherichia coli using biotin-H3K9me3 as substrate preincubated for ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCREB-binding protein(Human)
University of Z£Rich

Curated by ChEMBL
LigandPNGBDBM50150919(CHEMBL3775048)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human N-terminal His-tagged KDM4A (1 to 359 residues) expressed in Escherichia coli using biotin-H3K9me3 as substrate preincubated for ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCREB-binding protein(Human)
University of Z£Rich

Curated by ChEMBL
LigandPNGBDBM50150938(CHEMBL3775724)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human N-terminal His-tagged KDM4A (1 to 359 residues) expressed in Escherichia coli using biotin-H3K9me3 as substrate preincubated for ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCREB-binding protein(Human)
University of Z£Rich

Curated by ChEMBL
LigandPNGBDBM50150938(CHEMBL3775724)
Affinity DataKd:  1.30E+4nMAssay Description:Inhibition of human N-terminal His-tagged KDM4A (1 to 359 residues) expressed in Escherichia coli using biotin-H3K9me3 as substrate preincubated for ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCREB-binding protein(Human)
University of Z£Rich

Curated by ChEMBL
LigandPNGBDBM50150909(CHEMBL3774461)
Affinity DataKd:  4.20E+3nMAssay Description:Inhibition of human N-terminal His-tagged KDM4A (1 to 359 residues) expressed in Escherichia coli using biotin-H3K9me3 as substrate preincubated for ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCREB-binding protein(Human)
University of Z£Rich

Curated by ChEMBL
LigandPNGBDBM50148552(CHEMBL3770150)
Affinity DataKd:  770nMAssay Description:Inhibition of human N-terminal His-tagged KDM4A (1 to 359 residues) expressed in Escherichia coli using biotin-H3K9me3 as substrate preincubated for ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedPDB3D3D Structure (crystal)

TargetCREB-binding protein(Human)
University of Z£Rich

Curated by ChEMBL
LigandPNGBDBM50148550(CHEMBL3770132)
Affinity DataKd:  2.90E+4nMAssay Description:Inhibition of human N-terminal His-tagged KDM4A (1 to 359 residues) expressed in Escherichia coli using biotin-H3K9me3 as substrate preincubated for ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed