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Found 77 Enz. Inhib. hit(s) with all data for entry = 50046480
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50114806(CHEMBL3609752)
Affinity DataKi:  1.90E+3nMAssay Description:Binding affinity to human ERG expressed in HEK293 cells by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50114807(CHEMBL3608385)
Affinity DataKi:  2.00E+3nMAssay Description:Binding affinity to human ERG expressed in HEK293 cells by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50114800(CHEMBL3609749)
Affinity DataKi:  2.90E+3nMAssay Description:Binding affinity to human ERG expressed in HEK293 cells by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50114836(CHEMBL3608387)
Affinity DataKi:  3.30E+3nMAssay Description:Binding affinity to human ERG expressed in HEK293 cells by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50114805(CHEMBL3608384)
Affinity DataKi:  3.60E+3nMAssay Description:Binding affinity to human ERG expressed in HEK293 cells by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50114837(CHEMBL3609755)
Affinity DataKi:  6.50E+3nMAssay Description:Binding affinity to human ERG expressed in HEK293 cells by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50114810(CHEMBL3609754)
Affinity DataKi:  8.30E+3nMAssay Description:Binding affinity to human ERG expressed in HEK293 cells by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50114845(CHEMBL3609759)
Affinity DataKi:  1.90E+4nMAssay Description:Binding affinity to human ERG expressed in HEK293 cells by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50114798(CHEMBL3608381)
Affinity DataIC50:  8nMAssay Description:Modulation of gamma-secretase in human SH-SY5Y cells overexpressing APP C-terminal fragment SPA4CT assessed as inhibition of intracellular amyloid be...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50114806(CHEMBL3609752)
Affinity DataIC50:  11nMAssay Description:Modulation of gamma-secretase in human SH-SY5Y cells overexpressing APP C-terminal fragment SPA4CT assessed as inhibition of intracellular amyloid be...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50114837(CHEMBL3609755)
Affinity DataIC50:  13nMAssay Description:Modulation of gamma-secretase in human SH-SY5Y cells overexpressing APP C-terminal fragment SPA4CT assessed as inhibition of intracellular amyloid be...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50114798(CHEMBL3608381)
Affinity DataIC50:  18nMAssay Description:Modulation of gamma-secretase in human SH-SY5Y cells overexpressing APP C-terminal fragment SPA4CT assessed as inhibition of intracellular amyloid be...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50114793(CHEMBL3608392)
Affinity DataIC50:  26nMAssay Description:Modulation of gamma-secretase in human SH-SY5Y cells overexpressing APP C-terminal fragment SPA4CT assessed as inhibition of intracellular amyloid be...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50114796(CHEMBL3608380)
Affinity DataIC50:  28nMAssay Description:Modulation of gamma-secretase in human SH-SY5Y cells overexpressing APP C-terminal fragment SPA4CT assessed as inhibition of intracellular amyloid be...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50114803(CHEMBL3608383)
Affinity DataIC50:  28nMAssay Description:Modulation of gamma-secretase in human SH-SY5Y cells overexpressing APP C-terminal fragment SPA4CT assessed as inhibition of intracellular amyloid be...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50114842(CHEMBL3608390)
Affinity DataIC50:  29nMAssay Description:Modulation of gamma-secretase in human SH-SY5Y cells overexpressing APP C-terminal fragment SPA4CT assessed as inhibition of intracellular amyloid be...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50114800(CHEMBL3609749)
Affinity DataIC50:  31nMAssay Description:Modulation of gamma-secretase in human SH-SY5Y cells overexpressing APP C-terminal fragment SPA4CT assessed as inhibition of intracellular amyloid be...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50114836(CHEMBL3608387)
Affinity DataIC50:  36nMAssay Description:Modulation of gamma-secretase in human SH-SY5Y cells overexpressing APP C-terminal fragment SPA4CT assessed as inhibition of intracellular amyloid be...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50114802(CHEMBL3609750)
Affinity DataIC50:  38nMAssay Description:Modulation of gamma-secretase in human SH-SY5Y cells overexpressing APP C-terminal fragment SPA4CT assessed as inhibition of intracellular amyloid be...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50114845(CHEMBL3609759)
Affinity DataIC50:  42nMAssay Description:Modulation of gamma-secretase in human SH-SY5Y cells overexpressing APP C-terminal fragment SPA4CT assessed as inhibition of intracellular amyloid be...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50114791(CHEMBL3609748)
Affinity DataIC50:  45nMAssay Description:Modulation of gamma-secretase in human SKNBE-2 cells assessed as inhibition of intracellular amyloid beta 42 production after 6 hrs by sandwich ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50114839(CHEMBL3609756)
Affinity DataIC50:  50nMAssay Description:Modulation of gamma-secretase in human SH-SY5Y cells overexpressing APP C-terminal fragment SPA4CT assessed as inhibition of intracellular amyloid be...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50114804(CHEMBL3609751)
Affinity DataIC50:  56nMAssay Description:Modulation of gamma-secretase in human SH-SY5Y cells overexpressing APP C-terminal fragment SPA4CT assessed as inhibition of intracellular amyloid be...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50114810(CHEMBL3609754)
Affinity DataIC50:  58nMAssay Description:Modulation of gamma-secretase in human SH-SY5Y cells overexpressing APP C-terminal fragment SPA4CT assessed as inhibition of intracellular amyloid be...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50114844(CHEMBL3608391)
Affinity DataIC50:  62nMAssay Description:Modulation of gamma-secretase in human SH-SY5Y cells overexpressing APP C-terminal fragment SPA4CT assessed as inhibition of intracellular amyloid be...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50114789(CHEMBL3609747)
Affinity DataIC50:  67nMAssay Description:Modulation of gamma-secretase in human H4 cells expressing wild type APP751 assessed as inhibition of intracellular amyloid beta 42 production after ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50114805(CHEMBL3608384)
Affinity DataIC50:  70nMAssay Description:Modulation of gamma-secretase in human SH-SY5Y cells overexpressing APP C-terminal fragment SPA4CT assessed as inhibition of intracellular amyloid be...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50114796(CHEMBL3608380)
Affinity DataIC50:  70nMAssay Description:Modulation of gamma-secretase in human SH-SY5Y cells overexpressing APP C-terminal fragment SPA4CT assessed as inhibition of intracellular amyloid be...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50114806(CHEMBL3609752)
Affinity DataIC50:  73nMAssay Description:Modulation of gamma-secretase in human SH-SY5Y cells overexpressing APP C-terminal fragment SPA4CT assessed as inhibition of intracellular amyloid be...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50114809(CHEMBL3608386)
Affinity DataIC50:  78nMAssay Description:Modulation of gamma-secretase in human SH-SY5Y cells overexpressing APP C-terminal fragment SPA4CT assessed as inhibition of intracellular amyloid be...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50114807(CHEMBL3608385)
Affinity DataIC50:  78nMAssay Description:Modulation of gamma-secretase in human SH-SY5Y cells overexpressing APP C-terminal fragment SPA4CT assessed as inhibition of intracellular amyloid be...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50364033(CHEMBL1224151)
Affinity DataIC50:  85nMAssay Description:Modulation of gamma-secretase in HEK293 cells expressing Swedish mutant APP assessed as inhibition of intracellular amyloid beta 42 production after ...More data for this Ligand-Target Pair
LigandPNGBDBM50114837(CHEMBL3609755)
Affinity DataIC50:  100nMAssay Description:Modulation of gamma-secretase in human SH-SY5Y cells overexpressing APP C-terminal fragment SPA4CT assessed as inhibition of intracellular amyloid be...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50114803(CHEMBL3608383)
Affinity DataIC50:  110nMAssay Description:Modulation of gamma-secretase in human SH-SY5Y cells overexpressing APP C-terminal fragment SPA4CT assessed as inhibition of intracellular amyloid be...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50114801(CHEMBL3608382)
Affinity DataIC50:  110nMAssay Description:Modulation of gamma-secretase in human SH-SY5Y cells overexpressing APP C-terminal fragment SPA4CT assessed as inhibition of intracellular amyloid be...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50114792(CHEMBL2169963)
Affinity DataIC50:  120nMAssay Description:Modulation of gamma-secretase in HEK293 cells transfected with APPsw-6myc assessed as inhibition of intracellular amyloid beta 42 production after 16...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50114793(CHEMBL3608392)
Affinity DataIC50:  120nMAssay Description:Modulation of gamma-secretase in human SH-SY5Y cells overexpressing APP C-terminal fragment SPA4CT assessed as inhibition of intracellular amyloid be...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50114800(CHEMBL3609749)
Affinity DataIC50:  130nMAssay Description:Modulation of gamma-secretase in human SH-SY5Y cells overexpressing APP C-terminal fragment SPA4CT assessed as inhibition of intracellular amyloid be...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50114799(CHEMBL3608395)
Affinity DataIC50:  145nMAssay Description:Modulation of gamma-secretase in human SH-SY5Y cells overexpressing APP C-terminal fragment SPA4CT assessed as inhibition of intracellular amyloid be...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50114842(CHEMBL3608390)
Affinity DataIC50:  170nMAssay Description:Modulation of gamma-secretase in human SH-SY5Y cells overexpressing APP C-terminal fragment SPA4CT assessed as inhibition of intracellular amyloid be...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50114790(CHEMBL2151284)
Affinity DataIC50:  200nMAssay Description:Modulation of gamma-secretase in human SKNBE-2 cells transfected with wild type APP assessed as inhibition of intracellular amyloid beta 42 productio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50114808(CHEMBL3609753)
Affinity DataIC50:  210nMAssay Description:Modulation of gamma-secretase in human SH-SY5Y cells overexpressing APP C-terminal fragment SPA4CT assessed as inhibition of intracellular amyloid be...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50114836(CHEMBL3608387)
Affinity DataIC50:  230nMAssay Description:Modulation of gamma-secretase in human SH-SY5Y cells overexpressing APP C-terminal fragment SPA4CT assessed as inhibition of intracellular amyloid be...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50114843(CHEMBL3609758)
Affinity DataIC50:  260nMAssay Description:Modulation of gamma-secretase in human SH-SY5Y cells overexpressing APP C-terminal fragment SPA4CT assessed as inhibition of intracellular amyloid be...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50114797(CHEMBL3608394)
Affinity DataIC50:  270nMAssay Description:Modulation of gamma-secretase in human SH-SY5Y cells overexpressing APP C-terminal fragment SPA4CT assessed as inhibition of intracellular amyloid be...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50114845(CHEMBL3609759)
Affinity DataIC50:  290nMAssay Description:Modulation of gamma-secretase in human SH-SY5Y cells overexpressing APP C-terminal fragment SPA4CT assessed as inhibition of intracellular amyloid be...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50114840(CHEMBL3608389)
Affinity DataIC50:  310nMAssay Description:Modulation of gamma-secretase in human SH-SY5Y cells overexpressing APP C-terminal fragment SPA4CT assessed as inhibition of intracellular amyloid be...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50114802(CHEMBL3609750)
Affinity DataIC50:  310nMAssay Description:Modulation of gamma-secretase in human SH-SY5Y cells overexpressing APP C-terminal fragment SPA4CT assessed as inhibition of intracellular amyloid be...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50114838(CHEMBL3608388)
Affinity DataIC50:  350nMAssay Description:Modulation of gamma-secretase in human SH-SY5Y cells overexpressing APP C-terminal fragment SPA4CT assessed as inhibition of intracellular amyloid be...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50114844(CHEMBL3608391)
Affinity DataIC50:  380nMAssay Description:Modulation of gamma-secretase in human SH-SY5Y cells overexpressing APP C-terminal fragment SPA4CT assessed as inhibition of intracellular amyloid be...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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