Compile Data Set for Download or QSAR
Report error Found 13 Enz. Inhib. hit(s) with all data for entry = 50046846
TargetUrea transporter 2(Rat)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50134204BDBM50134204(CHEMBL3740772)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of rat UT-A1 expressed in MDCK-UT-A1-AQP1-YFP cells after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/23/2017
Entry Details Article
PubMed
TargetUrea transporter 2(Rat)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50135099BDBM50135099(CHEMBL3739636)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of rat UT-A1 expressed in MDCK-UT-A1-AQP1-YFP cells after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/23/2017
Entry Details Article
PubMed
TargetUrea transporter 2(Rat)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50135098BDBM50135098(CHEMBL3741585)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of rat UT-A1 expressed in MDCK-UT-A1-AQP1-YFP cells after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/23/2017
Entry Details Article
PubMed
TargetUrea transporter 2(Rat)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50134208BDBM50134208(CHEMBL3742039)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of rat UT-A1 expressed in MDCK-UT-A1-AQP1-YFP cells after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/23/2017
Entry Details Article
PubMed
TargetUrea transporter 2(Rat)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50134205BDBM50134205(CHEMBL3741102)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of rat UT-A1 expressed in MDCK-UT-A1-AQP1-YFP cells after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/23/2017
Entry Details Article
PubMed
TargetUrea transporter 2(Rat)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50135104BDBM50135104(CHEMBL3741981)
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibition of rat UT-A1 expressed in MDCK-UT-A1-AQP1-YFP cells after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/23/2017
Entry Details Article
PubMed
TargetUrea transporter 2(Rat)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50134206BDBM50134206(CHEMBL3742032)
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibition of rat UT-A1 expressed in MDCK-UT-A1-AQP1-YFP cells after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/23/2017
Entry Details Article
PubMed
TargetUrea transporter 1(Rat)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50135101BDBM50135101(CHEMBL3739701)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of UT-B in rat whole blood after 15 mins by RBC lysis assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/23/2017
Entry Details Article
PubMed
TargetUrea transporter 2(Rat)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50135103BDBM50135103(CHEMBL3741231)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of rat UT-A1 expressed in MDCK-UT-A1-AQP1-YFP cells after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/23/2017
Entry Details Article
PubMed
TargetUrea transporter 1(Rat)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50135106BDBM50135106(CHEMBL3739646)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of UT-B in rat whole blood after 15 mins by RBC lysis assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/23/2017
Entry Details Article
PubMed
TargetUrea transporter 2(Rat)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50134207BDBM50134207(CHEMBL3741384)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of rat UT-A1 expressed in MDCK-UT-A1-AQP1-YFP cells after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/23/2017
Entry Details Article
PubMed
TargetUrea transporter 2(Rat)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50134203BDBM50134203(CHEMBL2442435)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of rat UT-A1 expressed in MDCK-UT-A1-AQP1-YFP cells after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/23/2017
Entry Details Article
PubMed
TargetUrea transporter 2(Rat)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50134202BDBM50134202(CHEMBL424175)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of rat UT-A1 expressed in MDCK-UT-A1-AQP1-YFP cells after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/23/2017
Entry Details Article
PubMed