Compile Data Set for Download or QSAR
Report error Found 43 Enz. Inhib. hit(s) with all data for entry = 50046542
TargetMelatonin receptor type 1A(Human)
University of Urbino

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50117886BDBM50117886(CHEMBL3612603)
Affinity DataKi:  0.0300nMAssay Description:Displacement of 2-[125I]-Iodomelatonin from human MT1 receptor transfected in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2016
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
University of Urbino

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50117899BDBM50117899(CHEMBL3612604)
Affinity DataKi:  0.700nMAssay Description:Displacement of 2-[125I]-Iodomelatonin from human MT1 receptor transfected in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2016
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
University of Urbino

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50117899BDBM50117899(CHEMBL3612604)
Affinity DataEC50:  0.900nMAssay Description:Intrinsic activity at human MT1 receptor transfected in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2016
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
University of Urbino

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50117907BDBM50117907(CHEMBL3612608)
Affinity DataKi:  1.60nMAssay Description:Displacement of 2-[125I]-Iodomelatonin from human MT1 receptor transfected in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2016
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
University of Urbino

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50117886BDBM50117886(CHEMBL3612603)
Affinity DataEC50:  1.70nMAssay Description:Intrinsic activity at human MT1 receptor transfected in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2016
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
University of Urbino

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50117902BDBM50117902(CHEMBL3612606)
Affinity DataEC50:  2nMAssay Description:Intrinsic activity at human MT1 receptor transfected in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2016
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
University of Urbino

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50117879BDBM50117879(CHEMBL3612461)
Affinity DataKi:  5nMAssay Description:Displacement of 2-[125I]-Iodomelatonin from human MT1 receptor transfected in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2016
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
University of Urbino

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50117880BDBM50117880(CHEMBL3612462)
Affinity DataKi:  5.30nMAssay Description:Displacement of 2-[125I]-Iodomelatonin from human MT1 receptor transfected in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2016
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
University of Urbino

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50117902BDBM50117902(CHEMBL3612606)
Affinity DataKi:  5.80nMAssay Description:Displacement of 2-[125I]-Iodomelatonin from human MT1 receptor transfected in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2016
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
University of Urbino

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50117907BDBM50117907(CHEMBL3612608)
Affinity DataEC50:  6.20nMAssay Description:Intrinsic activity at human MT1 receptor transfected in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2016
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
University of Urbino

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50117876BDBM50117876(CHEMBL3612456)
Affinity DataKi:  13nMAssay Description:Displacement of 2-[125I]-Iodomelatonin from human MT1 receptor transfected in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2016
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
University of Urbino

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50117882BDBM50117882(CHEMBL3612464)
Affinity DataKi:  17nMAssay Description:Displacement of 2-[125I]-Iodomelatonin from human MT1 receptor transfected in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2016
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
University of Urbino

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50117908BDBM50117908(CHEMBL3612609)
Affinity DataKi:  22nMAssay Description:Displacement of 2-[125I]-Iodomelatonin from human MT1 receptor transfected in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2016
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
University of Urbino

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50117884BDBM50117884(CHEMBL3612468)
Affinity DataEC50:  31nMAssay Description:Intrinsic activity at human MT1 receptor transfected in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2016
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
University of Urbino

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50117883BDBM50117883(CHEMBL3612467)
Affinity DataEC50:  36nMAssay Description:Intrinsic activity at human MT1 receptor transfected in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2016
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
University of Urbino

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50117883BDBM50117883(CHEMBL3612467)
Affinity DataKi:  37nMAssay Description:Displacement of 2-[125I]-Iodomelatonin from human MT1 receptor transfected in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2016
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
University of Urbino

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50117884BDBM50117884(CHEMBL3612468)
Affinity DataKi:  45nMAssay Description:Displacement of 2-[125I]-Iodomelatonin from human MT1 receptor transfected in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2016
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
University of Urbino

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50117885BDBM50117885(CHEMBL3612469)
Affinity DataKi:  45nMAssay Description:Displacement of 2-[125I]-Iodomelatonin from human MT1 receptor transfected in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2016
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
University of Urbino

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50117875BDBM50117875(CHEMBL3612455)
Affinity DataKi:  57nMAssay Description:Displacement of 2-[125I]-Iodomelatonin from human MT1 receptor transfected in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2016
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
University of Urbino

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50117880BDBM50117880(CHEMBL3612462)
Affinity DataEC50:  110nMAssay Description:Intrinsic activity at human MT1 receptor transfected in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2016
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
University of Urbino

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50117877BDBM50117877(CHEMBL3612458)
Affinity DataKi:  115nMAssay Description:Displacement of 2-[125I]-Iodomelatonin from human MT1 receptor transfected in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2016
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
University of Urbino

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50117919BDBM50117919(CHEMBL3612470)
Affinity DataKi:  122nMAssay Description:Displacement of 2-[125I]-Iodomelatonin from human MT1 receptor transfected in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2016
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
University of Urbino

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50117881BDBM50117881(CHEMBL3612463)
Affinity DataKi:  132nMAssay Description:Displacement of 2-[125I]-Iodomelatonin from human MT1 receptor transfected in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2016
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
University of Urbino

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50117879BDBM50117879(CHEMBL3612461)
Affinity DataEC50:  160nMAssay Description:Intrinsic activity at human MT1 receptor transfected in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2016
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
University of Urbino

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50117926BDBM50117926(CHEMBL3612605)
Affinity DataKi:  171nMAssay Description:Displacement of 2-[125I]-Iodomelatonin from human MT1 receptor transfected in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2016
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
University of Urbino

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50117882BDBM50117882(CHEMBL3612464)
Affinity DataEC50:  177nMAssay Description:Intrinsic activity at human MT1 receptor transfected in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2016
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
University of Urbino

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50117917BDBM50117917(CHEMBL3612465)
Affinity DataKi:  186nMAssay Description:Displacement of 2-[125I]-Iodomelatonin from human MT1 receptor transfected in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2016
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
University of Urbino

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50117885BDBM50117885(CHEMBL3612469)
Affinity DataEC50:  192nMAssay Description:Intrinsic activity at human MT1 receptor transfected in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2016
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
University of Urbino

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50117918BDBM50117918(CHEMBL3612466)
Affinity DataKi:  214nMAssay Description:Displacement of 2-[125I]-Iodomelatonin from human MT1 receptor transfected in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2016
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
University of Urbino

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50117876BDBM50117876(CHEMBL3612456)
Affinity DataEC50:  242nMAssay Description:Intrinsic activity at human MT1 receptor transfected in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2016
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
University of Urbino

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50117920BDBM50117920(CHEMBL3612471)
Affinity DataKi:  291nMAssay Description:Displacement of 2-[125I]-Iodomelatonin from human MT1 receptor transfected in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2016
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
University of Urbino

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50117878BDBM50117878(CHEMBL3612460)
Affinity DataKi:  305nMAssay Description:Displacement of 2-[125I]-Iodomelatonin from human MT1 receptor transfected in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2016
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
University of Urbino

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50117929BDBM50117929(CHEMBL3612610)
Affinity DataKi:  326nMAssay Description:Displacement of 2-[125I]-Iodomelatonin from human MT1 receptor transfected in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2016
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
University of Urbino

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50117881BDBM50117881(CHEMBL3612463)
Affinity DataEC50:  393nMAssay Description:Intrinsic activity at human MT1 receptor transfected in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2016
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
University of Urbino

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50117915BDBM50117915(CHEMBL3612457)
Affinity DataKi:  480nMAssay Description:Displacement of 2-[125I]-Iodomelatonin from human MT1 receptor transfected in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2016
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
University of Urbino

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50117923BDBM50117923(CHEMBL3612602)
Affinity DataKi:  633nMAssay Description:Displacement of 2-[125I]-Iodomelatonin from human MT1 receptor transfected in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2016
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
University of Urbino

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50117908BDBM50117908(CHEMBL3612609)
Affinity DataEC50:  809nMAssay Description:Intrinsic activity at human MT1 receptor transfected in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2016
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
University of Urbino

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50117875BDBM50117875(CHEMBL3612455)
Affinity DataEC50:  906nMAssay Description:Intrinsic activity at human MT1 receptor transfected in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2016
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
University of Urbino

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50117916BDBM50117916(CHEMBL3612459)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of 2-[125I]-Iodomelatonin from human MT1 receptor transfected in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2016
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
University of Urbino

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50117877BDBM50117877(CHEMBL3612458)
Affinity DataEC50:  2.42E+3nMAssay Description:Intrinsic activity at human MT1 receptor transfected in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2016
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
University of Urbino

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50117878BDBM50117878(CHEMBL3612460)
Affinity DataEC50:  2.66E+3nMAssay Description:Intrinsic activity at human MT1 receptor transfected in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2016
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
University of Urbino

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50117912BDBM50117912(CHEMBL3612611)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of 2-[125I]-Iodomelatonin from human MT1 receptor transfected in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2016
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
University of Urbino

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50117927BDBM50117927(CHEMBL3612607)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of 2-[125I]-Iodomelatonin from human MT1 receptor transfected in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2016
Entry Details Article
PubMed