Compile Data Set for Download or QSAR
maximum 50k data
Found 7 Enz. Inhib. hit(s) with all data for entry = 50006479
TargetLipoprotein lipase(Bos taurus)
Ume£

Curated by ChEMBL
LigandPNGBDBM50500148(CHEMBL3746381)
Affinity DataEC50:  6.60E+3nMAssay Description:Induction of bovine LPL stabilization using intralipid as substrate preincubated for 10 mins with human recombinant ANGPTL4 followed by substrate add...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLipoprotein lipase(Bos taurus)
Ume£

Curated by ChEMBL
LigandPNGBDBM50500149(CHEMBL3747367)
Affinity DataEC50:  5.00E+3nMAssay Description:Induction of bovine LPL stabilization using intralipid as substrate preincubated for 10 mins with human recombinant ANGPTL4 followed by substrate add...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBile acid receptor(Homo sapiens (Human))
Ume£

Curated by ChEMBL
LigandPNGBDBM50500150(CHEMBL3746821)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at FXR (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLipoprotein lipase(Bos taurus)
Ume£

Curated by ChEMBL
LigandPNGBDBM50500150(CHEMBL3746821)
Affinity DataEC50:  6.00E+3nMAssay Description:Induction of bovine LPL stabilization using intralipid as substrate preincubated for 10 mins with human recombinant ANGPTL4 followed by substrate add...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Ume£

Curated by ChEMBL
LigandPNGBDBM50500150(CHEMBL3746821)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at PPARgamma (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Ume£

Curated by ChEMBL
LigandPNGBDBM50500150(CHEMBL3746821)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at RXRalpha (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Ume£

Curated by ChEMBL
LigandPNGBDBM50500150(CHEMBL3746821)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at PPARalpha (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed