Compile Data Set for Download or QSAR
Report error Found 7 Enz. Inhib. hit(s) with all data for entry = 50046783
TargetMuscarinic acetylcholine receptor M1(Human)
Sumitomo Dainippon Pharma

Curated by ChEMBL
LigandPNGBDBM50130927(CHEMBL3633184)
Affinity DataEC50:  14nMAssay Description:Agonist activity at human muscarinic M1 acetylcholine receptor expressed in CHO cells assessed as calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2016
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M4(Human)
Sumitomo Dainippon Pharma

Curated by ChEMBL
LigandPNGBDBM50130927(CHEMBL3633184)
Affinity DataEC50:  86nMAssay Description:Partial agonist activity at human muscarinic M4 acetylcholine receptor expressed in CHO cells co-expressing Galpha16 assessed as calcium mobilization...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2016
Entry Details Article
PubMed
TargetCytochrome P450 2C9(Human)
Sumitomo Dainippon Pharma

Curated by ChEMBL
LigandPNGBDBM50130927(CHEMBL3633184)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of CYP2C9 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2016
Entry Details Article
PubMed
TargetCytochrome P450 2C19(Human)
Sumitomo Dainippon Pharma

Curated by ChEMBL
LigandPNGBDBM50130927(CHEMBL3633184)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of CYP2C19 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2016
Entry Details Article
PubMed
TargetCytochrome P450 1A2(Human)
Sumitomo Dainippon Pharma

Curated by ChEMBL
LigandPNGBDBM50130927(CHEMBL3633184)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of CYP1A2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2016
Entry Details Article
PubMed
TargetCytochrome P450 2D6(Human)
Sumitomo Dainippon Pharma

Curated by ChEMBL
LigandPNGBDBM50130927(CHEMBL3633184)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of CYP2D6 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2016
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Sumitomo Dainippon Pharma

Curated by ChEMBL
LigandPNGBDBM50130927(CHEMBL3633184)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of CYP3A4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2016
Entry Details Article
PubMed