Compile Data Set for Download or QSAR
Report error Found 39 Enz. Inhib. hit(s) with all data for entry = 50006342
TargetDNA gyrase subunit B(Staphylococcus aureus)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50499015BDBM50499015(CHEMBL3736321)
Affinity DataIC50: 8nMAssay Description:Inhibition of Staphylococcus aureus DNA GyraseB ATPase activity using linear pBR322 DNA as substrate incubated for 30 mins by fluorescence polarizati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetDNA gyrase subunit B(Staphylococcus aureus)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50499034BDBM50499034(CHEMBL3736385)
Affinity DataIC50: 9nMAssay Description:Inhibition of Staphylococcus aureus DNA GyraseB ATPase activity using linear pBR322 DNA as substrate incubated for 30 mins by fluorescence polarizati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetDNA gyrase subunit B(Staphylococcus aureus)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50499014BDBM50499014(CHEMBL3735341)
Affinity DataIC50: 10nMAssay Description:Inhibition of Staphylococcus aureus DNA GyraseB ATPase activity using linear pBR322 DNA as substrate incubated for 30 mins by fluorescence polarizati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetDNA gyrase subunit B(Staphylococcus aureus)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50499047BDBM50499047(CHEMBL3735577)
Affinity DataIC50: 12nMAssay Description:Inhibition of Staphylococcus aureus DNA GyraseB ATPase activity using linear pBR322 DNA as substrate incubated for 30 mins by fluorescence polarizati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetDNA gyrase subunit B(Staphylococcus aureus)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50499028BDBM50499028(CHEMBL3736056)
Affinity DataIC50: 13nMAssay Description:Inhibition of Staphylococcus aureus DNA GyraseB ATPase activity using linear pBR322 DNA as substrate incubated for 30 mins by fluorescence polarizati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetDNA gyrase subunit B(Staphylococcus aureus)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50499020BDBM50499020(CHEMBL3735121)
Affinity DataIC50: 15nMAssay Description:Inhibition of Staphylococcus aureus DNA GyraseB ATPase activity using linear pBR322 DNA as substrate incubated for 30 mins by fluorescence polarizati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetDNA gyrase subunit B(Staphylococcus aureus)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50499022BDBM50499022(CHEMBL3735336)
Affinity DataIC50: 18nMAssay Description:Inhibition of Staphylococcus aureus DNA GyraseB ATPase activity using linear pBR322 DNA as substrate incubated for 30 mins by fluorescence polarizati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetDNA gyrase subunit B(Staphylococcus aureus)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50499027BDBM50499027(CHEMBL3736376)
Affinity DataIC50: 25nMAssay Description:Inhibition of Staphylococcus aureus DNA GyraseB ATPase activity using linear pBR322 DNA as substrate incubated for 30 mins by fluorescence polarizati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetDNA gyrase subunit B(Staphylococcus aureus)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50499012BDBM50499012(CHEMBL3736517)
Affinity DataIC50: 42nMAssay Description:Inhibition of Staphylococcus aureus DNA GyraseB ATPase activity using linear pBR322 DNA as substrate incubated for 30 mins by fluorescence polarizati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetDNA gyrase subunit B(Staphylococcus aureus)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50499048BDBM50499048(CHEMBL3736023)
Affinity DataIC50: 46nMAssay Description:Inhibition of Staphylococcus aureus DNA GyraseB ATPase activity using linear pBR322 DNA as substrate incubated for 30 mins by fluorescence polarizati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetDNA gyrase subunit B(Staphylococcus aureus)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50499045BDBM50499045(CHEMBL3736253)
Affinity DataIC50: 48nMAssay Description:Inhibition of Staphylococcus aureus DNA GyraseB ATPase activity using linear pBR322 DNA as substrate incubated for 30 mins by fluorescence polarizati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetDNA gyrase subunit B(Staphylococcus aureus)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50499033BDBM50499033(CHEMBL3736147)
Affinity DataIC50: 64nMAssay Description:Inhibition of Staphylococcus aureus DNA GyraseB ATPase activity using linear pBR322 DNA as substrate incubated for 30 mins by fluorescence polarizati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetDNA gyrase subunit B(Staphylococcus aureus)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50499042BDBM50499042(CHEMBL3735435)
Affinity DataIC50: 71nMAssay Description:Inhibition of Staphylococcus aureus DNA GyraseB ATPase activity using linear pBR322 DNA as substrate incubated for 30 mins by fluorescence polarizati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetDNA gyrase subunit B(Staphylococcus aureus)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50499019BDBM50499019(CHEMBL3735826)
Affinity DataIC50: 79nMAssay Description:Inhibition of Staphylococcus aureus DNA GyraseB ATPase activity using linear pBR322 DNA as substrate incubated for 30 mins by fluorescence polarizati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetDNA gyrase subunit B(Staphylococcus aureus)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50499021BDBM50499021(CHEMBL3734860)
Affinity DataIC50: 92nMAssay Description:Inhibition of Staphylococcus aureus DNA GyraseB ATPase activity using linear pBR322 DNA as substrate incubated for 30 mins by fluorescence polarizati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetDNA gyrase subunit B(Staphylococcus aureus)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50499029BDBM50499029(CHEMBL3735238)
Affinity DataIC50: 94nMAssay Description:Inhibition of Staphylococcus aureus DNA GyraseB ATPase activity using linear pBR322 DNA as substrate incubated for 30 mins by fluorescence polarizati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetDNA gyrase subunit B(Staphylococcus aureus)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50499016BDBM50499016(CHEMBL3735130)
Affinity DataIC50: 127nMAssay Description:Inhibition of Staphylococcus aureus DNA GyraseB ATPase activity using linear pBR322 DNA as substrate incubated for 30 mins by fluorescence polarizati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetDNA gyrase subunit B(Staphylococcus aureus)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50499031BDBM50499031(CHEMBL3735134)
Affinity DataIC50: 128nMAssay Description:Inhibition of Staphylococcus aureus DNA GyraseB ATPase activity using linear pBR322 DNA as substrate incubated for 30 mins by fluorescence polarizati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetDNA gyrase subunit B(Staphylococcus aureus)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50499018BDBM50499018(CHEMBL3736222)
Affinity DataIC50: 140nMAssay Description:Inhibition of Staphylococcus aureus DNA GyraseB ATPase activity using linear pBR322 DNA as substrate incubated for 30 mins by fluorescence polarizati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetDNA gyrase subunit B(Staphylococcus aureus)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50499036BDBM50499036(CHEMBL3735737)
Affinity DataIC50: 140nMAssay Description:Inhibition of Staphylococcus aureus DNA GyraseB ATPase activity using linear pBR322 DNA as substrate incubated for 30 mins by fluorescence polarizati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetDNA gyrase subunit B(Staphylococcus aureus)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50499037BDBM50499037(CHEMBL3736246)
Affinity DataIC50: 143nMAssay Description:Inhibition of Staphylococcus aureus DNA GyraseB ATPase activity using linear pBR322 DNA as substrate incubated for 30 mins by fluorescence polarizati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetDNA gyrase subunit B(Staphylococcus aureus)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50499043BDBM50499043(CHEMBL3736504)
Affinity DataIC50: 240nMAssay Description:Inhibition of Staphylococcus aureus DNA GyraseB ATPase activity using linear pBR322 DNA as substrate incubated for 30 mins by fluorescence polarizati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetDNA gyrase subunit B(Staphylococcus aureus)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50499049BDBM50499049(CHEMBL3735875)
Affinity DataIC50: 262nMAssay Description:Inhibition of Staphylococcus aureus DNA GyraseB ATPase activity using linear pBR322 DNA as substrate incubated for 30 mins by fluorescence polarizati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetDNA gyrase subunit B(Staphylococcus aureus)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50499026BDBM50499026(CHEMBL3735188)
Affinity DataIC50: 280nMAssay Description:Inhibition of Staphylococcus aureus DNA GyraseB ATPase activity using linear pBR322 DNA as substrate incubated for 30 mins by fluorescence polarizati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetDNA gyrase subunit B(Staphylococcus aureus)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50499025BDBM50499025(CHEMBL3735216)
Affinity DataIC50: 350nMAssay Description:Inhibition of Staphylococcus aureus DNA GyraseB ATPase activity using linear pBR322 DNA as substrate incubated for 30 mins by fluorescence polarizati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetDNA gyrase subunit B(Staphylococcus aureus)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50499046BDBM50499046(CHEMBL3735055)
Affinity DataIC50: 430nMAssay Description:Inhibition of Staphylococcus aureus DNA GyraseB ATPase activity using linear pBR322 DNA as substrate incubated for 30 mins by fluorescence polarizati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetDNA gyrase subunit B(Staphylococcus aureus)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50499032BDBM50499032(CHEMBL3736233)
Affinity DataIC50: 1.13E+3nMAssay Description:Inhibition of Staphylococcus aureus DNA GyraseB ATPase activity using linear pBR322 DNA as substrate incubated for 30 mins by fluorescence polarizati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetDNA gyrase subunit B(Staphylococcus aureus)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50499044BDBM50499044(CHEMBL3735073)
Affinity DataIC50: 1.22E+3nMAssay Description:Inhibition of Staphylococcus aureus DNA GyraseB ATPase activity using linear pBR322 DNA as substrate incubated for 30 mins by fluorescence polarizati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetDNA gyrase subunit B(Staphylococcus aureus)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50499023BDBM50499023(CHEMBL3735099)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of Staphylococcus aureus DNA GyraseB ATPase activity using linear pBR322 DNA as substrate incubated for 30 mins by fluorescence polarizati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetDNA gyrase subunit B(Staphylococcus aureus)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50499035BDBM50499035(CHEMBL3734929)
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of Staphylococcus aureus DNA GyraseB ATPase activity using linear pBR322 DNA as substrate incubated for 30 mins by fluorescence polarizati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetDNA gyrase subunit B(Staphylococcus aureus)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50499024BDBM50499024(CHEMBL3735471)
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of Staphylococcus aureus DNA GyraseB ATPase activity using linear pBR322 DNA as substrate incubated for 30 mins by fluorescence polarizati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetDNA gyrase subunit B(Staphylococcus aureus)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50499041BDBM50499041(CHEMBL3735431)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of Staphylococcus aureus DNA GyraseB ATPase activity using linear pBR322 DNA as substrate incubated for 30 mins by fluorescence polarizati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetDNA gyrase subunit B(Staphylococcus aureus)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50499013BDBM50499013(CHEMBL3736371)
Affinity DataIC50: 3.20E+3nMAssay Description:Inhibition of Staphylococcus aureus DNA GyraseB ATPase activity using linear pBR322 DNA as substrate incubated for 30 mins by fluorescence polarizati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetDNA gyrase subunit B(Staphylococcus aureus)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50499039BDBM50499039(CHEMBL3734950)
Affinity DataIC50: 5.29E+3nMAssay Description:Inhibition of Staphylococcus aureus DNA GyraseB ATPase activity using linear pBR322 DNA as substrate incubated for 30 mins by fluorescence polarizati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetDNA gyrase subunit B(Staphylococcus aureus)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50499030BDBM50499030(CHEMBL3736029)
Affinity DataIC50: 5.80E+3nMAssay Description:Inhibition of Staphylococcus aureus DNA GyraseB ATPase activity using linear pBR322 DNA as substrate incubated for 30 mins by fluorescence polarizati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetDNA gyrase subunit B(Staphylococcus aureus)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50499040BDBM50499040(CHEMBL3735112)
Affinity DataIC50: 6.06E+3nMAssay Description:Inhibition of Staphylococcus aureus DNA GyraseB ATPase activity using linear pBR322 DNA as substrate incubated for 30 mins by fluorescence polarizati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetDNA gyrase subunit B(Staphylococcus aureus)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50499017BDBM50499017(CHEMBL3735006)
Affinity DataIC50: 6.42E+3nMAssay Description:Inhibition of Staphylococcus aureus DNA GyraseB ATPase activity using linear pBR322 DNA as substrate incubated for 30 mins by fluorescence polarizati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetDNA gyrase subunit B(Staphylococcus aureus)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50499011BDBM50499011(CHEMBL3735833)
Affinity DataIC50: 6.50E+3nMAssay Description:Inhibition of Staphylococcus aureus DNA GyraseB ATPase activity using linear pBR322 DNA as substrate incubated for 30 mins by fluorescence polarizati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetDNA gyrase subunit B(Staphylococcus aureus)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50499038BDBM50499038(CHEMBL3736232)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of Staphylococcus aureus DNA GyraseB ATPase activity using linear pBR322 DNA as substrate incubated for 30 mins by fluorescence polarizati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed