Compile Data Set for Download or QSAR
Report error Found 35 Enz. Inhib. hit(s) with all data for entry = 50046820
TargetKappa-type opioid receptor(Rat)
The University of Kansas

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50133217BDBM50133217(CHEMBL3634917)
Affinity DataKi:  29nMAssay Description:Displacement of [3H]diprenorphine from rat kappa-opioid receptor expressed in CHO cells after 90 mins by scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2016
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 224024BDBM224024(Dynorphin A (1-13) | YGGFLRRXRPKLK | BDBM50241435)
Affinity DataEC50:  40nMAssay Description:Agonist activity at kappa-opioid receptor (unknown origin) after 90 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2016
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Rat)
The University of Kansas

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50133220BDBM50133220(CHEMBL3634920)
Affinity DataKi:  44nMAssay Description:Displacement of [3H]diprenorphine from rat kappa-opioid receptor expressed in CHO cells after 90 mins by scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2016
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Rat)
The University of Kansas

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50133221BDBM50133221(CHEMBL3634921)
Affinity DataKi:  62nMAssay Description:Displacement of [3H]diprenorphine from rat kappa-opioid receptor expressed in CHO cells after 90 mins by scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2016
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Rat)
The University of Kansas

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50133260BDBM50133260(CHEMBL3634927)
Affinity DataKi:  69nMAssay Description:Displacement of [3H]diprenorphine from rat kappa-opioid receptor expressed in CHO cells after 90 mins by scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2016
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Rat)
The University of Kansas

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50012153BDBM50012153(zyklophin)
Affinity DataKi:  95nMAssay Description:Displacement of [3H]diprenorphine from rat kappa-opioid receptor expressed in CHO cells after 90 mins by scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2016
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
The University of Kansas

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50133217BDBM50133217(CHEMBL3634917)
Affinity DataKi:  157nMAssay Description:Displacement of [3H]DAMGO from rat mu-opioid receptor expressed in CHO cells after 90 mins by scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2016
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Rat)
The University of Kansas

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50133218BDBM50133218(CHEMBL3634918)
Affinity DataKi:  160nMAssay Description:Displacement of [3H]diprenorphine from rat kappa-opioid receptor expressed in CHO cells after 90 mins by scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2016
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Rat)
The University of Kansas

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50133256BDBM50133256(CHEMBL3632647)
Affinity DataKi:  168nMAssay Description:Displacement of [3H]diprenorphine from rat kappa-opioid receptor expressed in CHO cells after 90 mins by scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2016
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Rat)
The University of Kansas

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50133263BDBM50133263(CHEMBL3634929)
Affinity DataKi:  222nMAssay Description:Displacement of [3H]diprenorphine from rat kappa-opioid receptor expressed in CHO cells after 90 mins by scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2016
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Rat)
The University of Kansas

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50133255BDBM50133255(CHEMBL3634926)
Affinity DataKi:  293nMAssay Description:Displacement of [3H]diprenorphine from rat kappa-opioid receptor expressed in CHO cells after 90 mins by scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2016
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Rat)
The University of Kansas

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50133219BDBM50133219(CHEMBL3634919)
Affinity DataKi:  326nMAssay Description:Displacement of [3H]diprenorphine from rat kappa-opioid receptor expressed in CHO cells after 90 mins by scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2016
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Rat)
The University of Kansas

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50133222BDBM50133222(CHEMBL3634922)
Affinity DataKi:  346nMAssay Description:Displacement of [3H]diprenorphine from rat kappa-opioid receptor expressed in CHO cells after 90 mins by scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2016
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Rat)
The University of Kansas

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50133262BDBM50133262(CHEMBL3634928)
Affinity DataKi:  403nMAssay Description:Displacement of [3H]diprenorphine from rat kappa-opioid receptor expressed in CHO cells after 90 mins by scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2016
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Rat)
The University of Kansas

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50133266BDBM50133266(CHEMBL3634930)
Affinity DataKi:  410nMAssay Description:Displacement of [3H]diprenorphine from rat kappa-opioid receptor expressed in CHO cells after 90 mins by scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2016
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Rat)
The University of Kansas

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50133216BDBM50133216(CHEMBL3634916)
Affinity DataKi:  412nMAssay Description:Displacement of [3H]diprenorphine from rat kappa-opioid receptor expressed in CHO cells after 90 mins by scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2016
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Rat)
The University of Kansas

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50133252BDBM50133252(CHEMBL3634923)
Affinity DataKi:  516nMAssay Description:Displacement of [3H]diprenorphine from rat kappa-opioid receptor expressed in CHO cells after 90 mins by scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2016
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
The University of Kansas

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50133218BDBM50133218(CHEMBL3634918)
Affinity DataKi:  1.49E+3nMAssay Description:Displacement of [3H]DAMGO from rat mu-opioid receptor expressed in CHO cells after 90 mins by scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2016
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Rat)
The University of Kansas

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50133254BDBM50133254(CHEMBL3634925)
Affinity DataKi:  1.75E+3nMAssay Description:Displacement of [3H]diprenorphine from rat kappa-opioid receptor expressed in CHO cells after 90 mins by scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2016
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
The University of Kansas

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50133216BDBM50133216(CHEMBL3634916)
Affinity DataKi:  2.44E+3nMAssay Description:Displacement of [3H]DAMGO from rat mu-opioid receptor expressed in CHO cells after 90 mins by scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2016
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
The University of Kansas

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50133256BDBM50133256(CHEMBL3632647)
Affinity DataKi:  2.55E+3nMAssay Description:Displacement of [3H]DAMGO from rat mu-opioid receptor expressed in CHO cells after 90 mins by scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2016
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
The University of Kansas

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50133266BDBM50133266(CHEMBL3634930)
Affinity DataKi:  2.61E+3nMAssay Description:Displacement of [3H]DAMGO from rat mu-opioid receptor expressed in CHO cells after 90 mins by scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2016
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
The University of Kansas

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50133262BDBM50133262(CHEMBL3634928)
Affinity DataKi:  3.20E+3nMAssay Description:Displacement of [3H]DAMGO from rat mu-opioid receptor expressed in CHO cells after 90 mins by scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2016
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Rat)
The University of Kansas

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50133253BDBM50133253(CHEMBL3634924)
Affinity DataKi:  4.01E+3nMAssay Description:Displacement of [3H]diprenorphine from rat kappa-opioid receptor expressed in CHO cells after 90 mins by scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2016
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
The University of Kansas

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50012153BDBM50012153(zyklophin)
Affinity DataKi:  4.38E+3nMAssay Description:Displacement of [3H]DAMGO from rat mu-opioid receptor expressed in CHO cells after 90 mins by scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2016
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
The University of Kansas

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50133263BDBM50133263(CHEMBL3634929)
Affinity DataKi:  8.26E+3nMAssay Description:Displacement of [3H]DAMGO from rat mu-opioid receptor expressed in CHO cells after 90 mins by scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2016
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
The University of Kansas

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50133221BDBM50133221(CHEMBL3634921)
Affinity DataKi:  8.47E+3nMAssay Description:Displacement of [3H]DAMGO from rat mu-opioid receptor expressed in CHO cells after 90 mins by scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2016
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
The University of Kansas

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50133252BDBM50133252(CHEMBL3634923)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]DAMGO from rat mu-opioid receptor expressed in CHO cells after 90 mins by scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2016
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
The University of Kansas

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50133253BDBM50133253(CHEMBL3634924)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]DAMGO from rat mu-opioid receptor expressed in CHO cells after 90 mins by scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2016
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
The University of Kansas

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50133255BDBM50133255(CHEMBL3634926)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]DAMGO from rat mu-opioid receptor expressed in CHO cells after 90 mins by scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2016
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
The University of Kansas

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50133222BDBM50133222(CHEMBL3634922)
Affinity DataKi:  1.06E+4nMAssay Description:Displacement of [3H]DAMGO from rat mu-opioid receptor expressed in CHO cells after 90 mins by scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2016
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
The University of Kansas

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50133220BDBM50133220(CHEMBL3634920)
Affinity DataKi:  1.09E+4nMAssay Description:Displacement of [3H]DAMGO from rat mu-opioid receptor expressed in CHO cells after 90 mins by scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2016
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
The University of Kansas

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50133219BDBM50133219(CHEMBL3634919)
Affinity DataKi:  1.10E+4nMAssay Description:Displacement of [3H]DAMGO from rat mu-opioid receptor expressed in CHO cells after 90 mins by scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2016
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
The University of Kansas

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50133260BDBM50133260(CHEMBL3634927)
Affinity DataKi:  1.13E+4nMAssay Description:Displacement of [3H]DAMGO from rat mu-opioid receptor expressed in CHO cells after 90 mins by scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2016
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
The University of Kansas

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50133254BDBM50133254(CHEMBL3634925)
Affinity DataKi:  1.15E+4nMAssay Description:Displacement of [3H]DAMGO from rat mu-opioid receptor expressed in CHO cells after 90 mins by scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2016
Entry Details Article
PubMed