Compile Data Set for Download or QSAR
maximum 50k data
Found 59 Enz. Inhib. hit(s) with all data for entry = 50046833
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50133685(CHEMBL3633663)
Affinity DataIC50:  4.16E+3nMAssay Description:Antagonist activity at human muscarinic M3 receptor expressed in HEK293 cells assessed as inhibition of carbachol-induced inositol monophosphate accu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50133685(CHEMBL3633663)
Affinity DataIC50:  4.17E+3nMAssay Description:Antagonist activity at human muscarinic M3 receptor expressed in HEK293 cells assessed as inhibition of carbachol-induced inositol monophosphate accu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor family C group 6 member A(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50133685(CHEMBL3633663)
Affinity DataIC50:  5.50E+3nMAssay Description:Antagonist activity at mouse GPRC6A receptor expressed in HEK293 cells assessed as inhibition of L-ornithine-induced inositol monophosphate accumulat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor family C group 6 member A(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50133685(CHEMBL3633663)
Affinity DataIC50:  5.50E+3nMAssay Description:Antagonist activity at mouse GPRC6A receptor expressed in HEK293 cells assessed as inhibition of L-ornithine-induced inositol monophosphate accumulat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor family C group 6 member A(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50133679(CHEMBL3633665)
Affinity DataIC50:  6.17E+3nMAssay Description:Antagonist activity at mouse GPRC6A receptor expressed in HEK293 cells assessed as inhibition of L-ornithine-induced inositol monophosphate accumulat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor family C group 6 member A(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50133679(CHEMBL3633665)
Affinity DataIC50:  6.17E+3nMAssay Description:Antagonist activity at mouse GPRC6A receptor expressed in HEK293 cells assessed as inhibition of L-ornithine-induced inositol monophosphate accumulat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor family C group 6 member A(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50133682(CHEMBL3633656)
Affinity DataIC50:  9.33E+3nMAssay Description:Antagonist activity at mouse GPRC6A receptor expressed in HEK293 cells assessed as inhibition of L-ornithine-induced inositol monophosphate accumulat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor family C group 6 member A(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50133682(CHEMBL3633656)
Affinity DataIC50:  9.33E+3nMAssay Description:Antagonist activity at mouse GPRC6A receptor expressed in HEK293 cells assessed as inhibition of L-ornithine-induced inositol monophosphate accumulat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor family C group 6 member A(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50133681(CHEMBL3633655)
Affinity DataIC50:  2.13E+4nMAssay Description:Antagonist activity at mouse GPRC6A receptor expressed in HEK293 cells assessed as inhibition of L-ornithine-induced inositol monophosphate accumulat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor family C group 6 member A(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50133681(CHEMBL3633655)
Affinity DataIC50:  2.14E+4nMAssay Description:Antagonist activity at mouse GPRC6A receptor expressed in HEK293 cells assessed as inhibition of L-ornithine-induced inositol monophosphate accumulat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor family C group 6 member A(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50133676(CHEMBL3633650)
Affinity DataIC50:  2.19E+4nMAssay Description:Antagonist activity at mouse GPRC6A receptor expressed in HEK293 cells assessed as inhibition of L-ornithine-induced inositol monophosphate accumulat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor family C group 6 member A(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50133676(CHEMBL3633650)
Affinity DataIC50:  2.19E+4nMAssay Description:Antagonist activity at mouse GPRC6A receptor expressed in HEK293 cells assessed as inhibition of L-ornithine-induced inositol monophosphate accumulat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50133676(CHEMBL3633650)
Affinity DataIC50:  2.75E+4nMAssay Description:Antagonist activity at human muscarinic M3 receptor expressed in HEK293 cells assessed as inhibition of carbachol-induced inositol monophosphate accu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50133676(CHEMBL3633650)
Affinity DataIC50:  2.75E+4nMAssay Description:Antagonist activity at human muscarinic M3 receptor expressed in HEK293 cells assessed as inhibition of carbachol-induced inositol monophosphate accu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor family C group 6 member A(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50133677(CHEMBL3633651)
Affinity DataIC50:  3.98E+4nMAssay Description:Antagonist activity at mouse GPRC6A receptor expressed in HEK293 cells assessed as inhibition of L-ornithine-induced inositol monophosphate accumulat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor family C group 6 member A(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50133677(CHEMBL3633651)
Affinity DataIC50:  3.98E+4nMAssay Description:Antagonist activity at mouse GPRC6A receptor expressed in HEK293 cells assessed as inhibition of L-ornithine-induced inositol monophosphate accumulat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50133682(CHEMBL3633656)
Affinity DataIC50:  4.17E+4nMAssay Description:Antagonist activity at rat mGluR5 expressed in CHO cells assessed as inhibition of L-glutamate-induced inositol monophosphate accumulation after 1 hr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50133682(CHEMBL3633656)
Affinity DataIC50:  4.17E+4nMAssay Description:Antagonist activity at rat mGluR5 expressed in CHO cells assessed as inhibition of L-glutamate-induced inositol monophosphate accumulation after 1 hr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50133679(CHEMBL3633665)
Affinity DataIC50:  5.12E+4nMAssay Description:Antagonist activity at human muscarinic M3 receptor expressed in HEK293 cells assessed as inhibition of carbachol-induced inositol monophosphate accu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50133682(CHEMBL3633656)
Affinity DataIC50:  5.13E+4nMAssay Description:Antagonist activity at human 5HT2C receptor expressed in HEK293 cells assessed as inhibition of serotonin-induced inositol monophosphate accumulation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50133679(CHEMBL3633665)
Affinity DataIC50:  5.13E+4nMAssay Description:Antagonist activity at human muscarinic M3 receptor expressed in HEK293 cells assessed as inhibition of carbachol-induced inositol monophosphate accu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50133682(CHEMBL3633656)
Affinity DataIC50:  5.13E+4nMAssay Description:Antagonist activity at human 5HT2C receptor expressed in HEK293 cells assessed as inhibition of serotonin-induced inositol monophosphate accumulation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Rattus norvegicus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50133682(CHEMBL3633656)
Affinity DataIC50:  5.62E+4nMAssay Description:Antagonist activity at rat CaSR expressed in HEK293 cells assessed as inhibition of Ca2+-induced inositol monophosphate accumulation after 1 hr by FR...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Rattus norvegicus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50133682(CHEMBL3633656)
Affinity DataIC50:  5.62E+4nMAssay Description:Antagonist activity at rat CaSR expressed in HEK293 cells assessed as inhibition of Ca2+-induced inositol monophosphate accumulation after 1 hr by FR...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor family C group 6 member A(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50133686(CHEMBL3633664)
Affinity DataIC50:  5.73E+4nMAssay Description:Antagonist activity at mouse GPRC6A receptor expressed in HEK293 cells assessed as inhibition of L-ornithine-induced inositol monophosphate accumulat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50133682(CHEMBL3633656)
Affinity DataIC50:  5.75E+4nMAssay Description:Antagonist activity at human muscarinic M3 receptor expressed in HEK293 cells assessed as inhibition of carbachol-induced inositol monophosphate accu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor family C group 6 member A(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50133686(CHEMBL3633664)
Affinity DataIC50:  5.75E+4nMAssay Description:Antagonist activity at mouse GPRC6A receptor expressed in HEK293 cells assessed as inhibition of L-ornithine-induced inositol monophosphate accumulat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50133682(CHEMBL3633656)
Affinity DataIC50:  5.75E+4nMAssay Description:Antagonist activity at human muscarinic M3 receptor expressed in HEK293 cells assessed as inhibition of carbachol-induced inositol monophosphate accu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor family C group 6 member A(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50133680(CHEMBL3633654)
Affinity DataIC50:  6.61E+4nMAssay Description:Antagonist activity at mouse GPRC6A receptor expressed in HEK293 cells assessed as inhibition of L-ornithine-induced inositol monophosphate accumulat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor family C group 6 member A(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50133680(CHEMBL3633654)
Affinity DataIC50:  6.61E+4nMAssay Description:Antagonist activity at mouse GPRC6A receptor expressed in HEK293 cells assessed as inhibition of L-ornithine-induced inositol monophosphate accumulat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor family C group 6 member A(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50133678(CHEMBL3633653)
Affinity DataIC50:  1.32E+5nMAssay Description:Antagonist activity at mouse GPRC6A receptor expressed in HEK293 cells assessed as inhibition of L-ornithine-induced inositol monophosphate accumulat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor family C group 6 member A(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50133678(CHEMBL3633653)
Affinity DataIC50:  1.32E+5nMAssay Description:Antagonist activity at mouse GPRC6A receptor expressed in HEK293 cells assessed as inhibition of L-ornithine-induced inositol monophosphate accumulat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50133685(CHEMBL3633663)
Affinity DataIC50:  2.09E+5nMAssay Description:Antagonist activity at human 5HT2C receptor expressed in HEK293 cells assessed as inhibition of serotonin-induced inositol monophosphate accumulation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50133685(CHEMBL3633663)
Affinity DataIC50:  2.09E+5nMAssay Description:Antagonist activity at human 5HT2C receptor expressed in HEK293 cells assessed as inhibition of serotonin-induced inositol monophosphate accumulation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50133676(CHEMBL3633650)
Affinity DataIC50:  2.14E+5nMAssay Description:Antagonist activity at human 5HT2C receptor expressed in HEK293 cells assessed as inhibition of serotonin-induced inositol monophosphate accumulation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50133676(CHEMBL3633650)
Affinity DataIC50:  2.14E+5nMAssay Description:Antagonist activity at human 5HT2C receptor expressed in HEK293 cells assessed as inhibition of serotonin-induced inositol monophosphate accumulation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50133676(CHEMBL3633650)
Affinity DataIC50:  2.24E+5nMAssay Description:Antagonist activity at rat mGluR5 expressed in CHO cells assessed as inhibition of L-glutamate-induced inositol monophosphate accumulation after 1 hr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50133676(CHEMBL3633650)
Affinity DataIC50:  2.24E+5nMAssay Description:Antagonist activity at rat mGluR5 expressed in CHO cells assessed as inhibition of L-glutamate-induced inositol monophosphate accumulation after 1 hr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Rattus norvegicus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50133685(CHEMBL3633663)
Affinity DataIC50:  2.40E+5nMAssay Description:Antagonist activity at rat CaSR expressed in HEK293 cells assessed as inhibition of Ca2+-induced inositol monophosphate accumulation after 1 hr by FR...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Rattus norvegicus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50133685(CHEMBL3633663)
Affinity DataIC50:  2.40E+5nMAssay Description:Antagonist activity at rat CaSR expressed in HEK293 cells assessed as inhibition of Ca2+-induced inositol monophosphate accumulation after 1 hr by FR...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor family C group 6 member A(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50133683(CHEMBL3633657)
Affinity DataIC50:  2.45E+5nMAssay Description:Antagonist activity at mouse GPRC6A receptor expressed in HEK293 cells assessed as inhibition of L-ornithine-induced inositol monophosphate accumulat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor family C group 6 member A(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50133683(CHEMBL3633657)
Affinity DataIC50:  2.48E+5nMAssay Description:Antagonist activity at mouse GPRC6A receptor expressed in HEK293 cells assessed as inhibition of L-ornithine-induced inositol monophosphate accumulat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor family C group 6 member A(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50133684(CHEMBL3633662)
Affinity DataIC50:  2.56E+5nMAssay Description:Antagonist activity at mouse GPRC6A receptor expressed in HEK293 cells assessed as inhibition of L-ornithine-induced inositol monophosphate accumulat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor family C group 6 member A(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50133684(CHEMBL3633662)
Affinity DataIC50:  2.57E+5nMAssay Description:Antagonist activity at mouse GPRC6A receptor expressed in HEK293 cells assessed as inhibition of L-ornithine-induced inositol monophosphate accumulat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50133685(CHEMBL3633663)
Affinity DataIC50:  2.63E+5nMAssay Description:Antagonist activity at rat mGluR5 expressed in CHO cells assessed as inhibition of L-glutamate-induced inositol monophosphate accumulation after 1 hr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50133685(CHEMBL3633663)
Affinity DataIC50:  2.63E+5nMAssay Description:Antagonist activity at rat mGluR5 expressed in CHO cells assessed as inhibition of L-glutamate-induced inositol monophosphate accumulation after 1 hr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50133679(CHEMBL3633665)
Affinity DataIC50:  2.69E+5nMAssay Description:Antagonist activity at human 5HT2C receptor expressed in HEK293 cells assessed as inhibition of serotonin-induced inositol monophosphate accumulation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50133679(CHEMBL3633665)
Affinity DataIC50:  2.69E+5nMAssay Description:Antagonist activity at rat mGluR5 expressed in CHO cells assessed as inhibition of L-glutamate-induced inositol monophosphate accumulation after 1 hr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50133679(CHEMBL3633665)
Affinity DataIC50:  2.69E+5nMAssay Description:Antagonist activity at human 5HT2C receptor expressed in HEK293 cells assessed as inhibition of serotonin-induced inositol monophosphate accumulation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50133679(CHEMBL3633665)
Affinity DataIC50:  2.69E+5nMAssay Description:Antagonist activity at rat mGluR5 expressed in CHO cells assessed as inhibition of L-glutamate-induced inositol monophosphate accumulation after 1 hr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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