Compile Data Set for Download or QSAR
Report error Found 71 Enz. Inhib. hit(s) with all data for entry = 50006493
TargetVitamin D3 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50200182((1S,3R,5Z,7E)-9,10-secocholesta-5,7,10(19)-triene-...)
Affinity DataIC50: 1.10nMAssay Description:Binding affinity to vitamin D3 receptor (unknown origin) after 4 hrs using fluormone VDR red by polar screen VDR competitor assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50500270(CHEMBL3747703)
Affinity DataEC50:  2.30nMAssay Description:Agonist activity at vitamin D3 receptor in human HL-60 cells assessed as induction of cell differentiation after 96 hrs by NBT dye-based microscopic ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50441900(CHEMBL2434990)
Affinity DataEC50:  8.5nMAssay Description:Agonist activity at vitamin D3 receptor in human HL-60 cells assessed as induction of cell differentiation after 96 hrs by NBT dye-based microscopic ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50200182((1S,3R,5Z,7E)-9,10-secocholesta-5,7,10(19)-triene-...)
Affinity DataEC50:  9nMAssay Description:Agonist activity at vitamin D3 receptor in human HL-60 cells assessed as induction of cell differentiation after 96 hrs by NBT dye-based microscopic ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50500264(CHEMBL3747394)
Affinity DataEC50:  10nMAssay Description:Agonist activity at vitamin D3 receptor in human HL-60 cells assessed as induction of cell differentiation after 96 hrs by NBT dye-based microscopic ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50500260(CHEMBL3747184)
Affinity DataEC50:  10nMAssay Description:Agonist activity at vitamin D3 receptor in human HL-60 cells assessed as induction of cell differentiation after 96 hrs by NBT dye-based microscopic ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50500291(CHEMBL3746520)
Affinity DataEC50:  14nMAssay Description:Agonist activity at vitamin D3 receptor in human HL-60 cells assessed as induction of cell differentiation after 96 hrs by NBT dye-based microscopic ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50500259(CHEMBL3746013)
Affinity DataEC50:  18nMAssay Description:Agonist activity at vitamin D3 receptor in human HL-60 cells assessed as induction of cell differentiation after 96 hrs by NBT dye-based microscopic ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50500267(CHEMBL3747341)
Affinity DataEC50:  22nMAssay Description:Agonist activity at vitamin D3 receptor in human HL-60 cells assessed as induction of cell differentiation after 96 hrs by NBT dye-based microscopic ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50500283(CHEMBL3747296)
Affinity DataEC50:  26nMAssay Description:Agonist activity at vitamin D3 receptor in human HL-60 cells assessed as induction of cell differentiation after 96 hrs by NBT dye-based microscopic ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50500268(CHEMBL3746465)
Affinity DataEC50:  37nMAssay Description:Agonist activity at vitamin D3 receptor in human HL-60 cells assessed as induction of cell differentiation after 96 hrs by NBT dye-based microscopic ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50500269(CHEMBL3747730)
Affinity DataEC50:  66nMAssay Description:Agonist activity at vitamin D3 receptor in human HL-60 cells assessed as induction of cell differentiation after 96 hrs by NBT dye-based microscopic ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50500269(CHEMBL3747730)
Affinity DataIC50: 71nMAssay Description:Binding affinity to vitamin D3 receptor (unknown origin) after 4 hrs using fluormone VDR red by polar screen VDR competitor assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50500279(CHEMBL3747383)
Affinity DataEC50:  77nMAssay Description:Agonist activity at vitamin D3 receptor in human HL-60 cells assessed as induction of cell differentiation after 96 hrs by NBT dye-based microscopic ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50500251(CHEMBL3746078)
Affinity DataEC50:  91nMAssay Description:Agonist activity at vitamin D3 receptor in human HL-60 cells assessed as induction of cell differentiation after 96 hrs by NBT dye-based microscopic ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50500282(CHEMBL3747675)
Affinity DataEC50:  96nMAssay Description:Agonist activity at vitamin D3 receptor in human HL-60 cells assessed as induction of cell differentiation after 96 hrs by NBT dye-based microscopic ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50500287(CHEMBL3746404)
Affinity DataEC50:  97nMAssay Description:Agonist activity at vitamin D3 receptor in human HL-60 cells assessed as induction of cell differentiation after 96 hrs by NBT dye-based microscopic ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50233329(CHEMBL3747640)
Affinity DataEC50:  110nMAssay Description:Agonist activity at vitamin D3 receptor in human HL-60 cells assessed as induction of cell differentiation after 96 hrs by NBT dye-based microscopic ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50500286(CHEMBL3747314)
Affinity DataEC50:  120nMAssay Description:Agonist activity at vitamin D3 receptor in human HL-60 cells assessed as induction of cell differentiation after 96 hrs by NBT dye-based microscopic ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50500292(CHEMBL3746222)
Affinity DataEC50:  130nMAssay Description:Agonist activity at vitamin D3 receptor in human HL-60 cells assessed as induction of cell differentiation after 96 hrs by NBT dye-based microscopic ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50500272(CHEMBL3747213)
Affinity DataEC50:  130nMAssay Description:Agonist activity at vitamin D3 receptor in human HL-60 cells assessed as induction of cell differentiation after 96 hrs by NBT dye-based microscopic ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50500258(CHEMBL3747642)
Affinity DataEC50:  150nMAssay Description:Agonist activity at vitamin D3 receptor in human HL-60 cells assessed as induction of cell differentiation after 96 hrs by NBT dye-based microscopic ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50500260(CHEMBL3747184)
Affinity DataIC50: 194nMAssay Description:Binding affinity to vitamin D3 receptor (unknown origin) after 4 hrs using fluormone VDR red by polar screen VDR competitor assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50500268(CHEMBL3746465)
Affinity DataIC50: 197nMAssay Description:Binding affinity to vitamin D3 receptor (unknown origin) after 4 hrs using fluormone VDR red by polar screen VDR competitor assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50500262(CHEMBL3747246)
Affinity DataEC50:  200nMAssay Description:Agonist activity at vitamin D3 receptor in human HL-60 cells assessed as induction of cell differentiation after 96 hrs by NBT dye-based microscopic ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50500297(CHEMBL3746415)
Affinity DataEC50:  210nMAssay Description:Agonist activity at vitamin D3 receptor in human HL-60 cells assessed as induction of cell differentiation after 96 hrs by NBT dye-based microscopic ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50500276(CHEMBL3747701)
Affinity DataEC50:  210nMAssay Description:Agonist activity at vitamin D3 receptor in human HL-60 cells assessed as induction of cell differentiation after 96 hrs by NBT dye-based microscopic ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50500278(CHEMBL3747218)
Affinity DataEC50:  240nMAssay Description:Agonist activity at vitamin D3 receptor in human HL-60 cells assessed as induction of cell differentiation after 96 hrs by NBT dye-based microscopic ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50500273(CHEMBL3747293)
Affinity DataEC50:  240nMAssay Description:Agonist activity at vitamin D3 receptor in human HL-60 cells assessed as induction of cell differentiation after 96 hrs by NBT dye-based microscopic ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50500280(CHEMBL3746576)
Affinity DataEC50:  380nMAssay Description:Agonist activity at vitamin D3 receptor in human HL-60 cells assessed as induction of cell differentiation after 96 hrs by NBT dye-based microscopic ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50500270(CHEMBL3747703)
Affinity DataIC50: 389nMAssay Description:Binding affinity to vitamin D3 receptor (unknown origin) after 4 hrs using fluormone VDR red by polar screen VDR competitor assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50500264(CHEMBL3747394)
Affinity DataIC50: 564nMAssay Description:Binding affinity to vitamin D3 receptor (unknown origin) after 4 hrs using fluormone VDR red by polar screen VDR competitor assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50500288(CHEMBL3746116)
Affinity DataEC50:  590nMAssay Description:Agonist activity at vitamin D3 receptor in human HL-60 cells assessed as induction of cell differentiation after 96 hrs by NBT dye-based microscopic ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM36720(LG190155)
Affinity DataEC50:  590nMAssay Description:Agonist activity at vitamin D3 receptor in human HL-60 cells assessed as induction of cell differentiation after 96 hrs by NBT dye-based microscopic ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50500255(CHEMBL3747395)
Affinity DataEC50:  630nMAssay Description:Agonist activity at vitamin D3 receptor in human HL-60 cells assessed as induction of cell differentiation after 96 hrs by NBT dye-based microscopic ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50500265(CHEMBL3746880)
Affinity DataEC50:  740nMAssay Description:Agonist activity at vitamin D3 receptor in human HL-60 cells assessed as induction of cell differentiation after 96 hrs by NBT dye-based microscopic ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50500267(CHEMBL3747341)
Affinity DataIC50: 863nMAssay Description:Binding affinity to vitamin D3 receptor (unknown origin) after 4 hrs using fluormone VDR red by polar screen VDR competitor assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50500290(CHEMBL3747768)
Affinity DataEC50:  870nMAssay Description:Agonist activity at vitamin D3 receptor in human HL-60 cells assessed as induction of cell differentiation after 96 hrs by NBT dye-based microscopic ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50500286(CHEMBL3747314)
Affinity DataIC50: 1.01E+3nMAssay Description:Binding affinity to vitamin D3 receptor (unknown origin) after 4 hrs using fluormone VDR red by polar screen VDR competitor assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50500263(CHEMBL3747284)
Affinity DataEC50:  1.03E+3nMAssay Description:Agonist activity at vitamin D3 receptor in human HL-60 cells assessed as induction of cell differentiation after 96 hrs by NBT dye-based microscopic ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50500259(CHEMBL3746013)
Affinity DataIC50: 1.19E+3nMAssay Description:Binding affinity to vitamin D3 receptor (unknown origin) after 4 hrs using fluormone VDR red by polar screen VDR competitor assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50500293(CHEMBL3746130)
Affinity DataEC50:  1.39E+3nMAssay Description:Agonist activity at vitamin D3 receptor in human HL-60 cells assessed as induction of cell differentiation after 96 hrs by NBT dye-based microscopic ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50500281(CHEMBL3746290)
Affinity DataEC50:  1.90E+3nMAssay Description:Agonist activity at vitamin D3 receptor in human HL-60 cells assessed as induction of cell differentiation after 96 hrs by NBT dye-based microscopic ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50500302(CHEMBL3745792)
Affinity DataEC50:  1.96E+3nMAssay Description:Agonist activity at vitamin D3 receptor in human HL-60 cells assessed as induction of cell differentiation after 96 hrs by NBT dye-based microscopic ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50500289(CHEMBL3746676)
Affinity DataEC50:  2.20E+3nMAssay Description:Agonist activity at vitamin D3 receptor in human HL-60 cells assessed as induction of cell differentiation after 96 hrs by NBT dye-based microscopic ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50500295(CHEMBL3746829)
Affinity DataEC50:  2.32E+3nMAssay Description:Agonist activity at vitamin D3 receptor in human HL-60 cells assessed as induction of cell differentiation after 96 hrs by NBT dye-based microscopic ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50500273(CHEMBL3747293)
Affinity DataIC50: 3.52E+3nMAssay Description:Binding affinity to vitamin D3 receptor (unknown origin) after 4 hrs using fluormone VDR red by polar screen VDR competitor assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50500285(CHEMBL3746653)
Affinity DataEC50:  3.95E+3nMAssay Description:Agonist activity at vitamin D3 receptor in human HL-60 cells assessed as induction of cell differentiation after 96 hrs by NBT dye-based microscopic ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50500256(CHEMBL3746817)
Affinity DataEC50:  5.10E+3nMAssay Description:Agonist activity at vitamin D3 receptor in human HL-60 cells assessed as induction of cell differentiation after 96 hrs by NBT dye-based microscopic ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50500258(CHEMBL3747642)
Affinity DataIC50: 5.24E+3nMAssay Description:Binding affinity to vitamin D3 receptor (unknown origin) after 4 hrs using fluormone VDR red by polar screen VDR competitor assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
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