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Found 7 Enz. Inhib. hit(s) with all data for entry = 50006514
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Chongqing University

Curated by ChEMBL
LigandPNGBDBM50066974(7-Benzyl-2,3-dihydroxy-6-methyl-4-propyl-naphthale...)
Affinity DataKi:  8.00E+3nMAssay Description:Inhibition of human LDHA using pyruvate as substrate assessed as disappearance of NADHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Chongqing University

Curated by ChEMBL
LigandPNGBDBM23222(Oxalamic acid | Oxamate | Oxamate, 3 | Oxamidic Ac...)
Affinity DataKi:  1.38E+5nMAssay Description:Inhibition of human LDHA using pyruvate as substrate assessed as disappearance of NADHMore data for this Ligand-Target Pair
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Chongqing University

Curated by ChEMBL
LigandPNGBDBM50500509(CHEMBL3747506)
Affinity DataIC50:  250nMAssay Description:Inhibition of human LDHA using pyruvate as substrate assessed as disappearance of NADH preincubated for 10 mins followed by substrate addition every ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Chongqing University

Curated by ChEMBL
LigandPNGBDBM50500507(CHEMBL3746581)
Affinity DataIC50:  2.30E+3nMAssay Description:Inhibition of human LDHA using pyruvate as substrate assessed as disappearance of NADH preincubated for 10 mins followed by substrate addition every ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Chongqing University

Curated by ChEMBL
LigandPNGBDBM50500508(CHEMBL3746496)
Affinity DataIC50:  3.50E+3nMAssay Description:Inhibition of human LDHA using pyruvate as substrate assessed as disappearance of NADH preincubated for 10 mins followed by substrate addition every ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Chongqing University

Curated by ChEMBL
LigandPNGBDBM50500505(CHEMBL3746548)
Affinity DataIC50:  4.80E+3nMAssay Description:Inhibition of human LDHA using pyruvate as substrate assessed as disappearance of NADH preincubated for 10 mins followed by substrate addition every ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Chongqing University

Curated by ChEMBL
LigandPNGBDBM50500506(CHEMBL3746363)
Affinity DataIC50:  7.80E+3nMAssay Description:Inhibition of human LDHA using pyruvate as substrate assessed as disappearance of NADH preincubated for 10 mins followed by substrate addition every ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed