TargetSterol regulatory element-binding protein 2(Homo sapiens (Human))
Catabasis Pharmaceuticals
Curated by ChEMBL
Catabasis Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 1.70E+4nMAssay Description:Inhibition of SREBP2 in human HepG2 cells assessed as reduction of PCSK9 secretion after 16 hrs by ELISAMore data for this Ligand-Target Pair
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Catabasis Pharmaceuticals
Curated by ChEMBL
Catabasis Pharmaceuticals
Curated by ChEMBL
Affinity DataEC50: 730nMAssay Description:Activation of GPR109A in human A431 cells assessed as suppression of forskolin-induced cAMP production after 30 minsMore data for this Ligand-Target Pair