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Found 153 Enz. Inhib. hit(s) with all data for entry = 50046956
TargetD(3) dopamine receptor(Homo sapiens (Human))
Aptuit

Curated by ChEMBL
LigandPNGBDBM50370572(CHEMBL85606 | SB-277011)
Affinity DataKi:  4nMAssay Description:Antagonist activity at human dopamine D3 receptor expressed in CHO cells after 90 mins by [35S]-GTPgamma S assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Aptuit

Curated by ChEMBL
LigandPNGBDBM50139853(CHEMBL3764143 | US10577361, E14)
Affinity DataKi:  5nMAssay Description:Displacement of [3H]-dofetilide from human ERG potassium channel by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Aptuit

Curated by ChEMBL
LigandPNGBDBM50139853(CHEMBL3764143 | US10577361, E14)
Affinity DataKi:  5.01nMAssay Description:Displacement of [3H]-dofetilide from human ERG potassium channel by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Aptuit

Curated by ChEMBL
LigandPNGBDBM50370572(CHEMBL85606 | SB-277011)
Affinity DataKi:  6.30nMAssay Description:Displacement of [125I]-7-OH-PIPAT from rat brain dopamine D3 receptor after 45 mins by microplate scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Aptuit

Curated by ChEMBL
LigandPNGBDBM50139924(CHEMBL3765266 | US10577361, E30)
Affinity DataKi:  10nMAssay Description:Antagonist activity at human dopamine D3 receptor expressed in CHO cells after 90 mins by [35S]-GTPgamma S assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Aptuit

Curated by ChEMBL
LigandPNGBDBM50139853(CHEMBL3764143 | US10577361, E14)
Affinity DataKi:  10nMAssay Description:Agonist activity at human dopamine D3 receptor expressed in CHO cells after 90 mins by [35S]-GTPgamma S assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Aptuit

Curated by ChEMBL
LigandPNGBDBM50139853(CHEMBL3764143 | US10577361, E14)
Affinity DataKi:  10nMAssay Description:Agonist activity at human dopamine D3 receptor expressed in CHO cells after 90 mins by [35S]-GTPgamma S assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Aptuit

Curated by ChEMBL
LigandPNGBDBM50139923(CHEMBL3765285 | US10577361, E29)
Affinity DataKi:  13nMAssay Description:Antagonist activity at human dopamine D3 receptor expressed in CHO cells after 90 mins by [35S]-GTPgamma S assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Aptuit

Curated by ChEMBL
LigandPNGBDBM50139923(CHEMBL3765285 | US10577361, E29)
Affinity DataKi:  16nMAssay Description:Displacement of [125I]-7-OH-PIPAT from rat brain dopamine D3 receptor after 45 mins by microplate scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Aptuit

Curated by ChEMBL
LigandPNGBDBM50139851(CHEMBL3764306 | US10577361, E20)
Affinity DataKi:  16nMAssay Description:Antagonist activity at human dopamine D3 receptor expressed in CHO cells after 90 mins by [35S]-GTPgamma S assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Aptuit

Curated by ChEMBL
LigandPNGBDBM50139925(CHEMBL3764246 | US10577361, E37)
Affinity DataKi:  16nMAssay Description:Antagonist activity at human dopamine D3 receptor expressed in CHO cells after 90 mins by [35S]-GTPgamma S assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Aptuit

Curated by ChEMBL
LigandPNGBDBM50139891(CHEMBL3764245 | US10577361, E25)
Affinity DataKi:  20nMAssay Description:Antagonist activity at human dopamine D3 receptor expressed in CHO cells after 90 mins by [35S]-GTPgamma S assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Aptuit

Curated by ChEMBL
LigandPNGBDBM50139852(CHEMBL3765426 | US10577361, E11)
Affinity DataKi:  20nMAssay Description:Antagonist activity at human dopamine D3 receptor expressed in CHO cells after 90 mins by [35S]-GTPgamma S assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Aptuit

Curated by ChEMBL
LigandPNGBDBM50139852(CHEMBL3765426 | US10577361, E11)
Affinity DataKi:  20nMAssay Description:Antagonist activity at human dopamine D3 receptor expressed in CHO cells after 90 mins by [35S]-GTPgamma S assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Aptuit

Curated by ChEMBL
LigandPNGBDBM50139895(CHEMBL3765267 | US10577361, E32)
Affinity DataKi:  20nMAssay Description:Displacement of [125I]-7-OH-PIPAT from rat brain dopamine D2 receptor after 45 mins by microplate scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Aptuit

Curated by ChEMBL
LigandPNGBDBM50139850(CHEMBL3763418 | US10577361, E4)
Affinity DataKi:  25nMAssay Description:Antagonist activity at human dopamine D3 receptor expressed in CHO cells after 90 mins by [35S]-GTPgamma S assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Aptuit

Curated by ChEMBL
LigandPNGBDBM50139861(CHEMBL3764557 | US10577361, E7)
Affinity DataKi:  25nMAssay Description:Antagonist activity at human dopamine D3 receptor expressed in CHO cells after 90 mins by [35S]-GTPgamma S assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Aptuit

Curated by ChEMBL
LigandPNGBDBM50139924(CHEMBL3765266 | US10577361, E30)
Affinity DataKi:  25nMAssay Description:Displacement of [125I]-7-OH-PIPAT from rat brain dopamine D3 receptor after 45 mins by microplate scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Aptuit

Curated by ChEMBL
LigandPNGBDBM50139850(CHEMBL3763418 | US10577361, E4)
Affinity DataKi:  25.1nMAssay Description:Displacement of [125I]-7-OH-PIPAT from rat brain dopamine D2 receptor after 45 mins by microplate scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Aptuit

Curated by ChEMBL
LigandPNGBDBM50139852(CHEMBL3765426 | US10577361, E11)
Affinity DataKi:  31.6nMAssay Description:Displacement of [125I]-7-OH-PIPAT from rat brain dopamine D3 receptor after 45 mins by microplate scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Aptuit

Curated by ChEMBL
LigandPNGBDBM50139852(CHEMBL3765426 | US10577361, E11)
Affinity DataKi:  32nMAssay Description:Agonist activity at human dopamine D3 receptor expressed in CHO cells after 90 mins by [35S]-GTPgamma S assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Aptuit

Curated by ChEMBL
LigandPNGBDBM50139851(CHEMBL3764306 | US10577361, E20)
Affinity DataKi:  32nMAssay Description:Displacement of [125I]-7-OH-PIPAT from rat brain dopamine D3 receptor after 45 mins by microplate scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Aptuit

Curated by ChEMBL
LigandPNGBDBM50139891(CHEMBL3764245 | US10577361, E25)
Affinity DataKi:  40nMAssay Description:Displacement of [125I]-7-OH-PIPAT from rat brain dopamine D3 receptor after 45 mins by microplate scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Aptuit

Curated by ChEMBL
LigandPNGBDBM50139921(CHEMBL3764597 | US10577361, E35)
Affinity DataKi:  40nMAssay Description:Agonist activity at human dopamine D3 receptor expressed in CHO cells after 90 mins by [35S]-GTPgamma S assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Aptuit

Curated by ChEMBL
LigandPNGBDBM50139895(CHEMBL3765267 | US10577361, E32)
Affinity DataKi:  63nMAssay Description:Displacement of [125I]-7-OH-PIPAT from rat brain dopamine D3 receptor after 45 mins by microplate scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Aptuit

Curated by ChEMBL
LigandPNGBDBM50139921(CHEMBL3764597 | US10577361, E35)
Affinity DataKi:  63nMAssay Description:Displacement of [125I]-7-OH-PIPAT from rat brain dopamine D3 receptor after 45 mins by microplate scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Aptuit

Curated by ChEMBL
LigandPNGBDBM50139850(CHEMBL3763418 | US10577361, E4)
Affinity DataKi:  79nMAssay Description:Displacement of [125I]-7-OH-PIPAT from rat brain dopamine D3 receptor after 45 mins by microplate scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Aptuit

Curated by ChEMBL
LigandPNGBDBM50139850(CHEMBL3763418 | US10577361, E4)
Affinity DataKi:  79nMAssay Description:Agonist activity at human dopamine D3 receptor expressed in CHO cells after 90 mins by [35S]-GTPgamma S assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Aptuit

Curated by ChEMBL
LigandPNGBDBM50139925(CHEMBL3764246 | US10577361, E37)
Affinity DataKi:  79nMAssay Description:Displacement of [125I]-7-OH-PIPAT from rat brain dopamine D3 receptor after 45 mins by microplate scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Aptuit

Curated by ChEMBL
LigandPNGBDBM50139854(CHEMBL3763200 | US10577361, E17)
Affinity DataKi:  100nMAssay Description:Displacement of [125I]-7-OH-PIPAT from rat brain dopamine D3 receptor after 45 mins by microplate scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Aptuit

Curated by ChEMBL
LigandPNGBDBM50139866(CHEMBL3764191 | US10577361, E28)
Affinity DataKi:  100nMAssay Description:Displacement of [125I]-7-OH-PIPAT from rat brain dopamine D3 receptor after 45 mins by microplate scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Aptuit

Curated by ChEMBL
LigandPNGBDBM50139898(CHEMBL3764639 | US10577361, E31)
Affinity DataKi:  100nMAssay Description:Displacement of [125I]-7-OH-PIPAT from rat brain dopamine D3 receptor after 45 mins by microplate scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Aptuit

Curated by ChEMBL
LigandPNGBDBM50139857(CHEMBL3765422)
Affinity DataKi:  100nMAssay Description:Displacement of [125I]-7-OH-PIPAT from rat brain dopamine D3 receptor after 45 mins by microplate scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Aptuit

Curated by ChEMBL
LigandPNGBDBM50139861(CHEMBL3764557 | US10577361, E7)
Affinity DataKi:  125nMAssay Description:Displacement of [125I]-7-OH-PIPAT from rat brain dopamine D3 receptor after 45 mins by microplate scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Aptuit

Curated by ChEMBL
LigandPNGBDBM50139897(CHEMBL3764830 | US10577361, E33)
Affinity DataKi:  126nMAssay Description:Displacement of [125I]-7-OH-PIPAT from rat brain dopamine D3 receptor after 45 mins by microplate scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Aptuit

Curated by ChEMBL
LigandPNGBDBM50139888(CHEMBL3764739 | US10577361, E24)
Affinity DataKi:  126nMAssay Description:Displacement of [125I]-7-OH-PIPAT from rat brain dopamine D3 receptor after 45 mins by microplate scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Aptuit

Curated by ChEMBL
LigandPNGBDBM50139861(CHEMBL3764557 | US10577361, E7)
Affinity DataKi:  126nMAssay Description:Agonist activity at human dopamine D3 receptor expressed in CHO cells after 90 mins by [35S]-GTPgamma S assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Aptuit

Curated by ChEMBL
LigandPNGBDBM50139922(CHEMBL3765072 | US10577361, E21)
Affinity DataKi:  126nMAssay Description:Displacement of [125I]-7-OH-PIPAT from rat brain dopamine D3 receptor after 45 mins by microplate scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Aptuit

Curated by ChEMBL
LigandPNGBDBM50139856(CHEMBL3765169 | US10577361, E19)
Affinity DataKi:  158nMAssay Description:Displacement of [125I]-7-OH-PIPAT from rat brain dopamine D3 receptor after 45 mins by microplate scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Aptuit

Curated by ChEMBL
LigandPNGBDBM50139865(CHEMBL3764833 | US10577361, E38)
Affinity DataKi:  200nMAssay Description:Displacement of [125I]-7-OH-PIPAT from rat brain dopamine D3 receptor after 45 mins by microplate scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Aptuit

Curated by ChEMBL
LigandPNGBDBM50139863(CHEMBL3764586 | US10577361, E34)
Affinity DataKi:  200nMAssay Description:Displacement of [125I]-7-OH-PIPAT from rat brain dopamine D3 receptor after 45 mins by microplate scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Aptuit

Curated by ChEMBL
LigandPNGBDBM50139855(CHEMBL3764612 | US10577361, E18)
Affinity DataKi:  251nMAssay Description:Displacement of [125I]-7-OH-PIPAT from rat brain dopamine D3 receptor after 45 mins by microplate scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Aptuit

Curated by ChEMBL
LigandPNGBDBM50139867(CHEMBL3764884 | US10577361, E26)
Affinity DataKi:  251nMAssay Description:Displacement of [125I]-7-OH-PIPAT from rat brain dopamine D3 receptor after 45 mins by microplate scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Aptuit

Curated by ChEMBL
LigandPNGBDBM50139859(CHEMBL3764212 | US10577361, E23)
Affinity DataKi:  316nMAssay Description:Displacement of [125I]-7-OH-PIPAT from rat brain dopamine D3 receptor after 45 mins by microplate scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Aptuit

Curated by ChEMBL
LigandPNGBDBM50139853(CHEMBL3764143 | US10577361, E14)
Affinity DataKi:  398nMAssay Description:Displacement of [125I]-7-OH-PIPAT from rat brain dopamine D3 receptor after 45 mins by microplate scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Aptuit

Curated by ChEMBL
LigandPNGBDBM50139860(CHEMBL3765754 | US10577361, E1)
Affinity DataKi:  398nMAssay Description:Agonist activity at human dopamine D3 receptor expressed in CHO cells after 90 mins by [35S]-GTPgamma S assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Aptuit

Curated by ChEMBL
LigandPNGBDBM50139860(CHEMBL3765754 | US10577361, E1)
Affinity DataKi:  398nMAssay Description:Displacement of [125I]-7-OH-PIPAT from rat brain dopamine D3 receptor after 45 mins by microplate scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Aptuit

Curated by ChEMBL
LigandPNGBDBM50139864(CHEMBL3765402 | US10577361, E36)
Affinity DataKi:  501nMAssay Description:Displacement of [125I]-7-OH-PIPAT from rat brain dopamine D3 receptor after 45 mins by microplate scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Aptuit

Curated by ChEMBL
LigandPNGBDBM50370572(CHEMBL85606 | SB-277011)
Affinity DataKi:  501nMAssay Description:Displacement of [125I]-7-OH-PIPAT from rat brain dopamine D2 receptor after 45 mins by microplate scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Aptuit

Curated by ChEMBL
LigandPNGBDBM50139882(CHEMBL3764251)
Affinity DataKi:  631nMAssay Description:Displacement of [125I]-7-OH-PIPAT from rat brain dopamine D3 receptor after 45 mins by microplate scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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