Compile Data Set for Download or QSAR
maximum 50k data
Report error Found 114 Enz. Inhib. hit(s) with all data for entry = 50047281
TargetTrypsin(Human)
Southern Research

Curated by ChEMBL
LigandPNGBDBM50158159(CHEMBL3780036)
Affinity DataKi:  100nMAssay Description:Inhibition of human recombinant trypsin using H2N(EEdansyl)GKQLRVVNGG (KDabcyl)-NH2 as substrate by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTrypsin(Human)
Southern Research

Curated by ChEMBL
LigandPNGBDBM50158155(CHEMBL3781354)
Affinity DataKi:  150nMAssay Description:Inhibition of human recombinant trypsin using H2N(EEdansyl)GKQLRVVNGG (KDabcyl)-NH2 as substrate by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetHepatocyte growth factor activator(Human)
Southern Research

Curated by ChEMBL
LigandPNGBDBM50158157(CHEMBL3780434)
Affinity DataKi:  160nMAssay Description:Inhibition of human recombinant hepatocyte growth factor activator using H2N(EEdansyl)GKQLRVVNGG (KDabcyl)-NH2 as substrate by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCoagulation factor X(Human)
Southern Research

Curated by ChEMBL
LigandPNGBDBM50158159(CHEMBL3780036)
Affinity DataKi:  180nMAssay Description:Inhibition of human recombinant factor 10a using H2N(EEdansyl)GKQLRVVNGG (KDabcyl)-NH2 as substrate by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCoagulation factor X(Human)
Southern Research

Curated by ChEMBL
LigandPNGBDBM50158157(CHEMBL3780434)
Affinity DataKi:  200nMAssay Description:Inhibition of human recombinant factor 10a using H2N(EEdansyl)GKQLRVVNGG (KDabcyl)-NH2 as substrate by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTrypsin(Human)
Southern Research

Curated by ChEMBL
LigandPNGBDBM50158157(CHEMBL3780434)
Affinity DataKi:  210nMAssay Description:Inhibition of human recombinant trypsin using H2N(EEdansyl)GKQLRVVNGG (KDabcyl)-NH2 as substrate by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSerine protease hepsin(Human)
Southern Research

Curated by ChEMBL
LigandPNGBDBM50158154(CHEMBL3781784)
Affinity DataKi:  210nMAssay Description:Inhibition of human recombinant hepsin using H2N(EEdansyl)GKQLRVVNGG (KDabcyl)-NH2 as substrate by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetHepatocyte growth factor activator(Human)
Southern Research

Curated by ChEMBL
LigandPNGBDBM50158155(CHEMBL3781354)
Affinity DataKi:  230nMAssay Description:Inhibition of human recombinant hepatocyte growth factor activator using H2N(EEdansyl)GKQLRVVNGG (KDabcyl)-NH2 as substrate by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCoagulation factor X(Human)
Southern Research

Curated by ChEMBL
LigandPNGBDBM50158160(CHEMBL3780584)
Affinity DataKi:  240nMAssay Description:Inhibition of human recombinant factor 10a using H2N(EEdansyl)GKQLRVVNGG (KDabcyl)-NH2 as substrate by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCoagulation factor X(Human)
Southern Research

Curated by ChEMBL
LigandPNGBDBM50158155(CHEMBL3781354)
Affinity DataKi:  250nMAssay Description:Inhibition of human recombinant factor 10a using H2N(EEdansyl)GKQLRVVNGG (KDabcyl)-NH2 as substrate by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSuppressor of tumorigenicity 14 protein(Human)
Southern Research

Curated by ChEMBL
LigandPNGBDBM50158154(CHEMBL3781784)
Affinity DataKi:  280nMAssay Description:Inhibition of human recombinant matripase catalytic domain using H2N(EEdansyl)GKQLRVVNGG (KDabcyl)-NH2 as substrate by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSerine protease hepsin(Human)
Southern Research

Curated by ChEMBL
LigandPNGBDBM50158152(CHEMBL3780269)
Affinity DataKi:  310nMAssay Description:Inhibition of human recombinant hepsin using H2N(EEdansyl)GKQLRVVNGG (KDabcyl)-NH2 as substrate by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTrypsin(Human)
Southern Research

Curated by ChEMBL
LigandPNGBDBM50158101(CHEMBL3781673)
Affinity DataKi:  310nMAssay Description:Inhibition of human recombinant trypsin using H2N(EEdansyl)GKQLRVVNGG (KDabcyl)-NH2 as substrate by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSuppressor of tumorigenicity 14 protein(Human)
Southern Research

Curated by ChEMBL
LigandPNGBDBM50158151(CHEMBL3780273)
Affinity DataKi:  330nMAssay Description:Inhibition of human recombinant matripase catalytic domain using H2N(EEdansyl)GKQLRVVNGG (KDabcyl)-NH2 as substrate by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTrypsin(Human)
Southern Research

Curated by ChEMBL
LigandPNGBDBM50158161(CHEMBL3781405)
Affinity DataKi:  330nMAssay Description:Inhibition of human recombinant trypsin using H2N(EEdansyl)GKQLRVVNGG (KDabcyl)-NH2 as substrate by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTrypsin(Human)
Southern Research

Curated by ChEMBL
LigandPNGBDBM50158150(CHEMBL3780005)
Affinity DataKi:  340nMAssay Description:Inhibition of human recombinant trypsin using H2N(EEdansyl)GKQLRVVNGG (KDabcyl)-NH2 as substrate by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetHepatocyte growth factor activator(Human)
Southern Research

Curated by ChEMBL
LigandPNGBDBM50158151(CHEMBL3780273)
Affinity DataKi:  350nMAssay Description:Inhibition of human recombinant hepatocyte growth factor activator using H2N(EEdansyl)GKQLRVVNGG (KDabcyl)-NH2 as substrate by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSuppressor of tumorigenicity 14 protein(Human)
Southern Research

Curated by ChEMBL
LigandPNGBDBM50158101(CHEMBL3781673)
Affinity DataKi:  350nMAssay Description:Inhibition of human recombinant matripase catalytic domain using H2N(EEdansyl)GKQLRVVNGG (KDabcyl)-NH2 as substrate by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetHepatocyte growth factor activator(Human)
Southern Research

Curated by ChEMBL
LigandPNGBDBM50158153(CHEMBL3780548)
Affinity DataKi:  380nMAssay Description:Inhibition of human recombinant hepatocyte growth factor activator using H2N(EEdansyl)GKQLRVVNGG (KDabcyl)-NH2 as substrate by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCoagulation factor X(Human)
Southern Research

Curated by ChEMBL
LigandPNGBDBM50157632(CHEMBL3781349)
Affinity DataKi:  380nMAssay Description:Inhibition of human recombinant factor 10a using H2N(EEdansyl)GKQLRVVNGG (KDabcyl)-NH2 as substrate by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTrypsin(Human)
Southern Research

Curated by ChEMBL
LigandPNGBDBM50158154(CHEMBL3781784)
Affinity DataKi:  390nMAssay Description:Inhibition of human recombinant trypsin using H2N(EEdansyl)GKQLRVVNGG (KDabcyl)-NH2 as substrate by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCoagulation factor X(Human)
Southern Research

Curated by ChEMBL
LigandPNGBDBM50157633(CHEMBL3779949)
Affinity DataKi:  400nMAssay Description:Inhibition of human recombinant factor 10a using H2N(EEdansyl)GKQLRVVNGG (KDabcyl)-NH2 as substrate by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTrypsin(Human)
Southern Research

Curated by ChEMBL
LigandPNGBDBM50158151(CHEMBL3780273)
Affinity DataKi:  420nMAssay Description:Inhibition of human recombinant trypsin using H2N(EEdansyl)GKQLRVVNGG (KDabcyl)-NH2 as substrate by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTrypsin(Human)
Southern Research

Curated by ChEMBL
LigandPNGBDBM50157632(CHEMBL3781349)
Affinity DataKi:  430nMAssay Description:Inhibition of human recombinant trypsin using H2N(EEdansyl)GKQLRVVNGG (KDabcyl)-NH2 as substrate by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetHepatocyte growth factor activator(Human)
Southern Research

Curated by ChEMBL
LigandPNGBDBM50158159(CHEMBL3780036)
Affinity DataKi:  430nMAssay Description:Inhibition of human recombinant hepatocyte growth factor activator using H2N(EEdansyl)GKQLRVVNGG (KDabcyl)-NH2 as substrate by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetHepatocyte growth factor activator(Human)
Southern Research

Curated by ChEMBL
LigandPNGBDBM50158101(CHEMBL3781673)
Affinity DataKi:  440nMAssay Description:Inhibition of human recombinant hepatocyte growth factor activator using H2N(EEdansyl)GKQLRVVNGG (KDabcyl)-NH2 as substrate by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSuppressor of tumorigenicity 14 protein(Human)
Southern Research

Curated by ChEMBL
LigandPNGBDBM50158161(CHEMBL3781405)
Affinity DataKi:  470nMAssay Description:Inhibition of human recombinant matripase catalytic domain using H2N(EEdansyl)GKQLRVVNGG (KDabcyl)-NH2 as substrate by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetHepatocyte growth factor activator(Human)
Southern Research

Curated by ChEMBL
LigandPNGBDBM50157632(CHEMBL3781349)
Affinity DataKi:  480nMAssay Description:Inhibition of human recombinant hepatocyte growth factor activator using H2N(EEdansyl)GKQLRVVNGG (KDabcyl)-NH2 as substrate by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTrypsin(Human)
Southern Research

Curated by ChEMBL
LigandPNGBDBM50158153(CHEMBL3780548)
Affinity DataKi:  500nMAssay Description:Compound was evaluated for potency towards nicotinic acetylcholine receptor in rat P2 brain membranes using [3H]-nicotine as a radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSuppressor of tumorigenicity 14 protein(Human)
Southern Research

Curated by ChEMBL
LigandPNGBDBM50157633(CHEMBL3779949)
Affinity DataKi:  510nMAssay Description:Inhibition of human recombinant matripase catalytic domain using H2N(EEdansyl)GKQLRVVNGG (KDabcyl)-NH2 as substrate by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCoagulation factor X(Human)
Southern Research

Curated by ChEMBL
LigandPNGBDBM50158151(CHEMBL3780273)
Affinity DataKi:  510nMAssay Description:Inhibition of human recombinant factor 10a using H2N(EEdansyl)GKQLRVVNGG (KDabcyl)-NH2 as substrate by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetHepatocyte growth factor activator(Human)
Southern Research

Curated by ChEMBL
LigandPNGBDBM50158150(CHEMBL3780005)
Affinity DataKi:  520nMAssay Description:Inhibition of human recombinant hepatocyte growth factor activator using H2N(EEdansyl)GKQLRVVNGG (KDabcyl)-NH2 as substrate by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSuppressor of tumorigenicity 14 protein(Human)
Southern Research

Curated by ChEMBL
LigandPNGBDBM50158150(CHEMBL3780005)
Affinity DataKi:  520nMAssay Description:Inhibition of human recombinant matripase catalytic domain using H2N(EEdansyl)GKQLRVVNGG (KDabcyl)-NH2 as substrate by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSuppressor of tumorigenicity 14 protein(Human)
Southern Research

Curated by ChEMBL
LigandPNGBDBM50157632(CHEMBL3781349)
Affinity DataKi:  530nMAssay Description:Inhibition of human recombinant matripase catalytic domain using H2N(EEdansyl)GKQLRVVNGG (KDabcyl)-NH2 as substrate by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSerine protease hepsin(Human)
Southern Research

Curated by ChEMBL
LigandPNGBDBM50158101(CHEMBL3781673)
Affinity DataKi:  530nMAssay Description:Inhibition of human recombinant hepsin using H2N(EEdansyl)GKQLRVVNGG (KDabcyl)-NH2 as substrate by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSerine protease hepsin(Human)
Southern Research

Curated by ChEMBL
LigandPNGBDBM50157632(CHEMBL3781349)
Affinity DataKi:  540nMAssay Description:Inhibition of human recombinant hepsin using H2N(EEdansyl)GKQLRVVNGG (KDabcyl)-NH2 as substrate by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTrypsin(Human)
Southern Research

Curated by ChEMBL
LigandPNGBDBM50158158(CHEMBL3780208)
Affinity DataKi:  550nMAssay Description:Inhibition of human recombinant trypsin using H2N(EEdansyl)GKQLRVVNGG (KDabcyl)-NH2 as substrate by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSerine protease hepsin(Human)
Southern Research

Curated by ChEMBL
LigandPNGBDBM50158159(CHEMBL3780036)
Affinity DataKi:  560nMAssay Description:Inhibition of human recombinant hepsin using H2N(EEdansyl)GKQLRVVNGG (KDabcyl)-NH2 as substrate by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSuppressor of tumorigenicity 14 protein(Human)
Southern Research

Curated by ChEMBL
LigandPNGBDBM50158155(CHEMBL3781354)
Affinity DataKi:  580nMAssay Description:Compound was evaluated for inhibitory activity towards nicotinic acetylcholine receptor in rat P2 brain membranes using [3H]-nicotine as a radioligan...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTrypsin(Human)
Southern Research

Curated by ChEMBL
LigandPNGBDBM50158152(CHEMBL3780269)
Affinity DataKi:  590nMAssay Description:Inhibition of human recombinant trypsin using H2N(EEdansyl)GKQLRVVNGG (KDabcyl)-NH2 as substrate by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCoagulation factor X(Human)
Southern Research

Curated by ChEMBL
LigandPNGBDBM50158150(CHEMBL3780005)
Affinity DataKi:  610nMAssay Description:Inhibition of human recombinant factor 10a using H2N(EEdansyl)GKQLRVVNGG (KDabcyl)-NH2 as substrate by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCoagulation factor X(Human)
Southern Research

Curated by ChEMBL
LigandPNGBDBM50158101(CHEMBL3781673)
Affinity DataKi:  660nMAssay Description:Inhibition of human recombinant factor 10a using H2N(EEdansyl)GKQLRVVNGG (KDabcyl)-NH2 as substrate by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSerine protease hepsin(Human)
Southern Research

Curated by ChEMBL
LigandPNGBDBM50158150(CHEMBL3780005)
Affinity DataKi:  670nMAssay Description:Inhibition of human recombinant hepsin using H2N(EEdansyl)GKQLRVVNGG (KDabcyl)-NH2 as substrate by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSerine protease hepsin(Human)
Southern Research

Curated by ChEMBL
LigandPNGBDBM50158155(CHEMBL3781354)
Affinity DataKi:  690nMAssay Description:Inhibition of human recombinant hepsin using H2N(EEdansyl)GKQLRVVNGG (KDabcyl)-NH2 as substrate by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSerine protease hepsin(Human)
Southern Research

Curated by ChEMBL
LigandPNGBDBM50158151(CHEMBL3780273)
Affinity DataKi:  720nMAssay Description:Inhibition of human recombinant hepsin using H2N(EEdansyl)GKQLRVVNGG (KDabcyl)-NH2 as substrate by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCoagulation factor X(Human)
Southern Research

Curated by ChEMBL
LigandPNGBDBM50158153(CHEMBL3780548)
Affinity DataKi:  740nMAssay Description:Inhibition of human recombinant factor 10a using H2N(EEdansyl)GKQLRVVNGG (KDabcyl)-NH2 as substrate by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCoagulation factor X(Human)
Southern Research

Curated by ChEMBL
LigandPNGBDBM50158161(CHEMBL3781405)
Affinity DataKi:  750nMAssay Description:Inhibition of human recombinant factor 10a using H2N(EEdansyl)GKQLRVVNGG (KDabcyl)-NH2 as substrate by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSerine protease hepsin(Human)
Southern Research

Curated by ChEMBL
LigandPNGBDBM50158158(CHEMBL3780208)
Affinity DataKi:  760nMAssay Description:Inhibition of human recombinant hepsin using H2N(EEdansyl)GKQLRVVNGG (KDabcyl)-NH2 as substrate by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSerine protease hepsin(Human)
Southern Research

Curated by ChEMBL
LigandPNGBDBM50158156(CHEMBL3781626)
Affinity DataKi:  760nMAssay Description:Inhibition of human recombinant hepsin using H2N(EEdansyl)GKQLRVVNGG (KDabcyl)-NH2 as substrate by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTrypsin(Human)
Southern Research

Curated by ChEMBL
LigandPNGBDBM50158156(CHEMBL3781626)
Affinity DataKi:  760nMAssay Description:Inhibition of human recombinant trypsin using H2N(EEdansyl)GKQLRVVNGG (KDabcyl)-NH2 as substrate by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Displayed 1 to 50 (of 114 total ) | Next | Last >>
Jump to: