Compile Data Set for Download or QSAR
Report error Found 14 Enz. Inhib. hit(s) with all data for entry = 50047394
TargetNischarin(Rat)
Medical University of Gdansk

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50164835BDBM50164835(CHEMBL3800398)
Affinity DataKi:  32nMAssay Description:Displacement of [3H]clonidine from Imidazoline receptor 1 in Sprague-Dawley rat kidney P2 membranes after 45 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2017
Entry Details Article
PubMed
TargetNischarin(Rat)
Medical University of Gdansk

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50164841BDBM50164841(CHEMBL3798191)
Affinity DataKi:  79nMAssay Description:Displacement of [3H]clonidine from Imidazoline receptor 1 in Sprague-Dawley rat kidney P2 membranes after 45 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2017
Entry Details Article
PubMed
TargetNischarin(Rat)
Medical University of Gdansk

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50164834BDBM50164834(CHEMBL3798638)
Affinity DataKi:  468nMAssay Description:Displacement of [3H]clonidine from Imidazoline receptor 1 in Sprague-Dawley rat kidney P2 membranes after 45 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2017
Entry Details Article
PubMed
TargetNischarin(Rat)
Medical University of Gdansk

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50164837BDBM50164837(CHEMBL3800446)
Affinity DataKi:  789nMAssay Description:Displacement of [3H]clonidine from Imidazoline receptor 1 in Sprague-Dawley rat kidney P2 membranes after 45 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2017
Entry Details Article
PubMed
TargetNischarin(Rat)
Medical University of Gdansk

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50164842BDBM50164842(CHEMBL3798387)
Affinity DataKi:  1.00E+3nMAssay Description:Displacement of [3H]clonidine from Imidazoline receptor 1 in Sprague-Dawley rat kidney P2 membranes after 45 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2017
Entry Details Article
PubMed
TargetNischarin(Rat)
Medical University of Gdansk

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50164838BDBM50164838(CHEMBL3797854)
Affinity DataKi:  5.58E+3nMAssay Description:Displacement of [3H]clonidine from Imidazoline receptor 1 in Sprague-Dawley rat kidney P2 membranes after 45 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2017
Entry Details Article
PubMed
TargetNischarin(Rat)
Medical University of Gdansk

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50164839BDBM50164839(CHEMBL3797661)
Affinity DataKi:  9.63E+3nMAssay Description:Displacement of [3H]clonidine from Imidazoline receptor 1 in Sprague-Dawley rat kidney P2 membranes after 45 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2017
Entry Details Article
PubMed
TargetNischarin(Rat)
Medical University of Gdansk

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50164840BDBM50164840(CHEMBL3799780)
Affinity DataKi:  1.03E+4nMAssay Description:Displacement of [3H]clonidine from Imidazoline receptor 1 in Sprague-Dawley rat kidney P2 membranes after 45 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2017
Entry Details Article
PubMed
TargetNischarin(Rat)
Medical University of Gdansk

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50164836BDBM50164836(CHEMBL3798967)
Affinity DataKi:  1.05E+4nMAssay Description:Displacement of [3H]clonidine from Imidazoline receptor 1 in Sprague-Dawley rat kidney P2 membranes after 45 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2017
Entry Details Article
PubMed
TargetNischarin(Rat)
Medical University of Gdansk

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50164833BDBM50164833(CHEMBL3799346)
Affinity DataKi:  1.46E+4nMAssay Description:Displacement of [3H]clonidine from Imidazoline receptor 1 in Sprague-Dawley rat kidney P2 membranes after 45 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2017
Entry Details Article
PubMed
TargetNischarin(Rat)
Medical University of Gdansk

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50164845BDBM50164845(CHEMBL3799081)
Affinity DataKi:  3.63E+4nMAssay Description:Displacement of [3H]clonidine from Imidazoline receptor 1 in Sprague-Dawley rat kidney P2 membranes after 45 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2017
Entry Details Article
PubMed
TargetNischarin(Rat)
Medical University of Gdansk

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50164843BDBM50164843(CHEMBL3800486)
Affinity DataKi:  4.58E+4nMAssay Description:Displacement of [3H]clonidine from Imidazoline receptor 1 in Sprague-Dawley rat kidney P2 membranes after 45 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2017
Entry Details Article
PubMed
TargetNischarin(Rat)
Medical University of Gdansk

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50164832BDBM50164832(CHEMBL3797481)
Affinity DataKi:  8.14E+4nMAssay Description:Displacement of [3H]clonidine from Imidazoline receptor 1 in Sprague-Dawley rat kidney P2 membranes after 45 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2017
Entry Details Article
PubMed
TargetNischarin(Rat)
Medical University of Gdansk

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50164844BDBM50164844(CHEMBL3798276)
Affinity DataKi:  5.88E+5nMAssay Description:Displacement of [3H]clonidine from Imidazoline receptor 1 in Sprague-Dawley rat kidney P2 membranes after 45 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2017
Entry Details Article
PubMed