Compile Data Set for Download or QSAR
maximum 50k data
Found 13 Enz. Inhib. hit(s) with all data for entry = 50001762
TargetThromboxane-A synthase(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50017914(3-(1-Ethyl-5-pyridin-3-ylmethyl-1H-pyrrol-2-yl)-2-...)
Affinity DataIC50:  42nMAssay Description:Inhibition of thromboxane A2 synthetase as reduced ADP-induced aggregation of human platelet rich plasma in the presence of pig aortal microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50017903(3-(1-tert-Butyl-5-pyridin-3-ylmethyl-1H-pyrrol-3-y...)
Affinity DataIC50:  44nMAssay Description:Inhibition of thromboxane A2 synthetase as reduced ADP-induced aggregation of human platelet rich plasma in the presence of pig aortal microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50017905(2-Methyl-3-(1-methyl-5-pyridin-3-ylmethyl-1H-pyrro...)
Affinity DataIC50:  50nMAssay Description:Inhibition of thromboxane A2 synthetase as reduced ADP-induced aggregation of human platelet rich plasma in the presence of pig aortal microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50017909(3-(5-Imidazol-1-ylmethyl-1-methyl-1H-pyrrol-2-yl)-...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of thromboxane A2 synthetase as reduced ADP-induced aggregation of human platelet rich plasma in the presence of pig aortal microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50017896((E)-3-(4-Imidazol-1-ylmethyl-phenyl)-acrylic acid ...)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of thromboxane A2 synthetase as reduced ADP-induced aggregation of human platelet rich plasma in the presence of pig aortal microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50017912(3-(5-Imidazol-1-ylmethyl-1-methyl-1H-pyrrol-3-yl)-...)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of thromboxane A2 synthetase as reduced ADP-induced aggregation of human platelet rich plasma in the presence of pig aortal microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50017915(3-(1-Isopropyl-5-pyridin-3-ylmethyl-1H-pyrrol-2-yl...)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibition of thromboxane A2 synthetase as reduced ADP-induced aggregation of human platelet rich plasma in the presence of pig aortal microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50017908(3-(5-Imidazol-1-ylmethyl-1-methyl-1H-pyrrol-2-yl)-...)
Affinity DataIC50:  3.80E+3nMAssay Description:Inhibition of thromboxane A2 synthetase as reduced ADP-induced aggregation of human platelet rich plasma in the presence of pig aortal microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50017910(3-(5-Imidazol-1-ylmethyl-1-methyl-1H-pyrrol-3-yl)-...)
Affinity DataIC50:  4.60E+3nMAssay Description:Inhibition of thromboxane A2 synthetase as reduced ADP-induced aggregation of human platelet rich plasma in the presence of pig aortal microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50017913(2-(5-Imidazol-1-ylmethyl-1-methyl-1H-pyrrol-2-yl)-...)
Affinity DataIC50:  9.10E+3nMAssay Description:Inhibition of thromboxane A2 synthetase as reduced ADP-induced aggregation of human platelet rich plasma in the presence of pig aortal microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50017901(3-(5-Imidazol-1-ylmethyl-1H-pyrrol-2-yl)-2-methyl-...)
Affinity DataIC50:  9.10E+3nMAssay Description:Inhibition of thromboxane A2 synthetase as reduced ADP-induced aggregation of human platelet rich plasma in the presence of pig aortal microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50017898(2-Methyl-3-(1-phenyl-5-pyridin-3-ylmethyl-1H-pyrro...)
Affinity DataIC50:  2.40E+4nMAssay Description:Inhibition of thromboxane A2 synthetase as reduced ADP-induced aggregation of human platelet rich plasma in the presence of pig aortal microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50017907(3-[1-(2,2-Dimethyl-propyl)-5-pyridin-3-ylmethyl-1H...)
Affinity DataIC50:  7.80E+4nMAssay Description:Inhibition of thromboxane A2 synthetase as reduced ADP-induced aggregation of human platelet rich plasma in the presence of pig aortal microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed