Compile Data Set for Download or QSAR
Report error Found 85 Enz. Inhib. hit(s) with all data for entry = 50047377
TargetProteasome subunit beta type-5(Human)
Nanjing Forestry University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50163687BDBM50163687(CHEMBL3793848)
Affinity DataIC50: 0.760nMAssay Description:Inhibition of chymotrypsin like activity of human 20S proteasome using Suc-Leu-Leu-Val-Tyr-AMC as substrate preincubated for 10 mins followed by subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/10/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Nanjing Forestry University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50163687BDBM50163687(CHEMBL3793848)
Affinity DataIC50: 0.760nMAssay Description:Inhibition of chymotrypsin like activity of human 20S proteasome using Suc-Leu-Leu-Val-Tyr-AMC as substrate preincubated for 10 mins followed by subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/10/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Nanjing Forestry University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50163559BDBM50163559(CHEMBL3794168)
Affinity DataIC50: 1.10nMAssay Description:Inhibition of chymotrypsin like activity of human 20S proteasome using Suc-Leu-Leu-Val-Tyr-AMC as substrate preincubated for 10 mins followed by subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/10/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Nanjing Forestry University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50163559BDBM50163559(CHEMBL3794168)
Affinity DataIC50: 1.12nMAssay Description:Inhibition of chymotrypsin like activity of human 20S proteasome using Suc-Leu-Leu-Val-Tyr-AMC as substrate preincubated for 10 mins followed by subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/10/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Nanjing Forestry University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50163685BDBM50163685(CHEMBL3793581)
Affinity DataIC50: 1.15nMAssay Description:Inhibition of chymotrypsin like activity of human 20S proteasome using Suc-Leu-Leu-Val-Tyr-AMC as substrate preincubated for 10 mins followed by subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/10/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Nanjing Forestry University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50163673BDBM50163673(CHEMBL3793238)
Affinity DataIC50: 1.16nMAssay Description:Inhibition of chymotrypsin like activity of human 20S proteasome using Suc-Leu-Leu-Val-Tyr-AMC as substrate preincubated for 10 mins followed by subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/10/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Nanjing Forestry University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50163698BDBM50163698(CHEMBL3794310)
Affinity DataIC50: 1.16nMAssay Description:Inhibition of chymotrypsin like activity of human 20S proteasome using Suc-Leu-Leu-Val-Tyr-AMC as substrate preincubated for 10 mins followed by subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/10/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Nanjing Forestry University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50163698BDBM50163698(CHEMBL3794310)
Affinity DataIC50: 1.20nMAssay Description:Inhibition of chymotrypsin like activity of human 20S proteasome using Suc-Leu-Leu-Val-Tyr-AMC as substrate preincubated for 10 mins followed by subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/10/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Nanjing Forestry University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50160867BDBM50160867(CHEMBL499361)
Affinity DataIC50: 1.20nMAssay Description:Inhibition of chymotrypsin like activity of human 20S proteasome using Suc-Leu-Leu-Val-Tyr-AMC as substrate preincubated for 10 mins followed by subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/10/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Nanjing Forestry University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50163673BDBM50163673(CHEMBL3793238)
Affinity DataIC50: 1.20nMAssay Description:Inhibition of chymotrypsin like activity of human 20S proteasome using Suc-Leu-Leu-Val-Tyr-AMC as substrate preincubated for 10 mins followed by subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/10/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Nanjing Forestry University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50163685BDBM50163685(CHEMBL3793581)
Affinity DataIC50: 1.20nMAssay Description:Inhibition of chymotrypsin like activity of human 20S proteasome using Suc-Leu-Leu-Val-Tyr-AMC as substrate preincubated for 10 mins followed by subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/10/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Nanjing Forestry University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50160867BDBM50160867(CHEMBL499361)
Affinity DataIC50: 1.20nMAssay Description:Inhibition of chymotrypsin like activity of human 20S proteasome using Suc-Leu-Leu-Val-Tyr-AMC as substrate preincubated for 10 mins followed by subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/10/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Nanjing Forestry University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50163565BDBM50163565(CHEMBL3794136)
Affinity DataIC50: 1.26nMAssay Description:Inhibition of chymotrypsin like activity of human 20S proteasome using Suc-Leu-Leu-Val-Tyr-AMC as substrate preincubated for 10 mins followed by subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/10/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Nanjing Forestry University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50163565BDBM50163565(CHEMBL3794136)
Affinity DataIC50: 1.30nMAssay Description:Inhibition of chymotrypsin like activity of human 20S proteasome using Suc-Leu-Leu-Val-Tyr-AMC as substrate preincubated for 10 mins followed by subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/10/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Nanjing Forestry University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50163689BDBM50163689(CHEMBL3794207)
Affinity DataIC50: 1.30nMAssay Description:Inhibition of chymotrypsin like activity of human 20S proteasome using Suc-Leu-Leu-Val-Tyr-AMC as substrate preincubated for 10 mins followed by subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/10/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Nanjing Forestry University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50163689BDBM50163689(CHEMBL3794207)
Affinity DataIC50: 1.34nMAssay Description:Inhibition of chymotrypsin like activity of human 20S proteasome using Suc-Leu-Leu-Val-Tyr-AMC as substrate preincubated for 10 mins followed by subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/10/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Nanjing Forestry University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50163668BDBM50163668(CHEMBL3793242)
Affinity DataIC50: 1.46nMAssay Description:Inhibition of chymotrypsin like activity of human 20S proteasome using Suc-Leu-Leu-Val-Tyr-AMC as substrate preincubated for 10 mins followed by subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/10/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Nanjing Forestry University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50163668BDBM50163668(CHEMBL3793242)
Affinity DataIC50: 1.5nMAssay Description:Inhibition of chymotrypsin like activity of human 20S proteasome using Suc-Leu-Leu-Val-Tyr-AMC as substrate preincubated for 10 mins followed by subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/10/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Nanjing Forestry University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50160868BDBM50160868(CHEMBL499504)
Affinity DataIC50: 1.60nMAssay Description:Inhibition of chymotrypsin like activity of human 20S proteasome using Suc-Leu-Leu-Val-Tyr-AMC as substrate preincubated for 10 mins followed by subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/10/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Nanjing Forestry University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50160868BDBM50160868(CHEMBL499504)
Affinity DataIC50: 1.60nMAssay Description:Inhibition of chymotrypsin like activity of human 20S proteasome using Suc-Leu-Leu-Val-Tyr-AMC as substrate preincubated for 10 mins followed by subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/10/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Nanjing Forestry University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50069989BDBM50069989(CHEMBL325041 | (R)-3-methyl-1-((S)-3-phenyl-2-(pyr...)
Affinity DataIC50: 1.90nMAssay Description:Inhibition of chymotrypsin like activity of human 20S proteasome using Suc-Leu-Leu-Val-Tyr-AMC as substrate preincubated for 10 mins followed by subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/10/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Nanjing Forestry University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50163555BDBM50163555(CHEMBL606394)
Affinity DataIC50: 1.90nMAssay Description:Inhibition of chymotrypsin like activity of human 20S proteasome using Suc-Leu-Leu-Val-Tyr-AMC as substrate preincubated for 10 mins followed by subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/10/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Nanjing Forestry University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50069989BDBM50069989(CHEMBL325041 | (R)-3-methyl-1-((S)-3-phenyl-2-(pyr...)
Affinity DataIC50: 1.90nMAssay Description:Inhibition of chymotrypsin like activity of human 20S proteasome using Suc-Leu-Leu-Val-Tyr-AMC as substrate preincubated for 10 mins followed by subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/10/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Nanjing Forestry University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50163561BDBM50163561(CHEMBL3792511)
Affinity DataIC50: 1.90nMAssay Description:Inhibition of chymotrypsin like activity of human 20S proteasome using Suc-Leu-Leu-Val-Tyr-AMC as substrate preincubated for 10 mins followed by subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/10/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Nanjing Forestry University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50163561BDBM50163561(CHEMBL3792511)
Affinity DataIC50: 1.92nMAssay Description:Inhibition of chymotrypsin like activity of human 20S proteasome using Suc-Leu-Leu-Val-Tyr-AMC as substrate preincubated for 10 mins followed by subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/10/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Nanjing Forestry University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50163555BDBM50163555(CHEMBL606394)
Affinity DataIC50: 1.92nMAssay Description:Inhibition of chymotrypsin like activity of human 20S proteasome using Suc-Leu-Leu-Val-Tyr-AMC as substrate preincubated for 10 mins followed by subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/10/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Nanjing Forestry University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50163703BDBM50163703(CHEMBL3792573)
Affinity DataIC50: 2.30nMAssay Description:Inhibition of chymotrypsin like activity of human 20S proteasome using Suc-Leu-Leu-Val-Tyr-AMC as substrate preincubated for 10 mins followed by subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/10/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Nanjing Forestry University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50163703BDBM50163703(CHEMBL3792573)
Affinity DataIC50: 2.34nMAssay Description:Inhibition of chymotrypsin like activity of human 20S proteasome using Suc-Leu-Leu-Val-Tyr-AMC as substrate preincubated for 10 mins followed by subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/10/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Nanjing Forestry University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50163693BDBM50163693(CHEMBL3793093)
Affinity DataIC50: 2.46nMAssay Description:Inhibition of chymotrypsin like activity of human 20S proteasome using Suc-Leu-Leu-Val-Tyr-AMC as substrate preincubated for 10 mins followed by subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/10/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Nanjing Forestry University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50163693BDBM50163693(CHEMBL3793093)
Affinity DataIC50: 2.5nMAssay Description:Inhibition of chymotrypsin like activity of human 20S proteasome using Suc-Leu-Leu-Val-Tyr-AMC as substrate preincubated for 10 mins followed by subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/10/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Nanjing Forestry University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50163704BDBM50163704(CHEMBL3793863)
Affinity DataIC50: 2.70nMAssay Description:Inhibition of chymotrypsin like activity of human 20S proteasome using Suc-Leu-Leu-Val-Tyr-AMC as substrate preincubated for 10 mins followed by subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/10/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Nanjing Forestry University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50163704BDBM50163704(CHEMBL3793863)
Affinity DataIC50: 2.73nMAssay Description:Inhibition of chymotrypsin like activity of human 20S proteasome using Suc-Leu-Leu-Val-Tyr-AMC as substrate preincubated for 10 mins followed by subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/10/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Nanjing Forestry University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50163557BDBM50163557(CHEMBL3792854)
Affinity DataIC50: 3.20nMAssay Description:Inhibition of chymotrypsin like activity of human 20S proteasome using Suc-Leu-Leu-Val-Tyr-AMC as substrate preincubated for 10 mins followed by subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/10/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Nanjing Forestry University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50163557BDBM50163557(CHEMBL3792854)
Affinity DataIC50: 3.21nMAssay Description:Inhibition of chymotrypsin like activity of human 20S proteasome using Suc-Leu-Leu-Val-Tyr-AMC as substrate preincubated for 10 mins followed by subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/10/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Nanjing Forestry University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50163715BDBM50163715(CHEMBL3793683)
Affinity DataIC50: 3.30nMAssay Description:Inhibition of chymotrypsin like activity of human 20S proteasome using Suc-Leu-Leu-Val-Tyr-AMC as substrate preincubated for 10 mins followed by subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/10/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Nanjing Forestry University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50163715BDBM50163715(CHEMBL3793683)
Affinity DataIC50: 3.34nMAssay Description:Inhibition of chymotrypsin like activity of human 20S proteasome using Suc-Leu-Leu-Val-Tyr-AMC as substrate preincubated for 10 mins followed by subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/10/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Nanjing Forestry University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50163669BDBM50163669(CHEMBL3793066)
Affinity DataIC50: 3.37nMAssay Description:Inhibition of chymotrypsin like activity of human 20S proteasome using Suc-Leu-Leu-Val-Tyr-AMC as substrate preincubated for 10 mins followed by subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/10/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Nanjing Forestry University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50163669BDBM50163669(CHEMBL3793066)
Affinity DataIC50: 3.40nMAssay Description:Inhibition of chymotrypsin like activity of human 20S proteasome using Suc-Leu-Leu-Val-Tyr-AMC as substrate preincubated for 10 mins followed by subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/10/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Nanjing Forestry University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50163663BDBM50163663(CHEMBL3794171)
Affinity DataIC50: 3.67nMAssay Description:Inhibition of chymotrypsin like activity of human 20S proteasome using Suc-Leu-Leu-Val-Tyr-AMC as substrate preincubated for 10 mins followed by subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/10/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Nanjing Forestry University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50163663BDBM50163663(CHEMBL3794171)
Affinity DataIC50: 3.70nMAssay Description:Inhibition of chymotrypsin like activity of human 20S proteasome using Suc-Leu-Leu-Val-Tyr-AMC as substrate preincubated for 10 mins followed by subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/10/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Nanjing Forestry University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50163558BDBM50163558(CHEMBL3793344)
Affinity DataIC50: 4.18nMAssay Description:Inhibition of chymotrypsin like activity of human 20S proteasome using Suc-Leu-Leu-Val-Tyr-AMC as substrate preincubated for 10 mins followed by subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/10/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Nanjing Forestry University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50163558BDBM50163558(CHEMBL3793344)
Affinity DataIC50: 4.20nMAssay Description:Inhibition of chymotrypsin like activity of human 20S proteasome using Suc-Leu-Leu-Val-Tyr-AMC as substrate preincubated for 10 mins followed by subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/10/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Nanjing Forestry University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50163649BDBM50163649(CHEMBL1169560)
Affinity DataIC50: 4.26nMAssay Description:Inhibition of chymotrypsin like activity of human 20S proteasome using Suc-Leu-Leu-Val-Tyr-AMC as substrate preincubated for 10 mins followed by subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/10/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Nanjing Forestry University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50163649BDBM50163649(CHEMBL1169560)
Affinity DataIC50: 4.30nMAssay Description:Inhibition of chymotrypsin like activity of human 20S proteasome using Suc-Leu-Leu-Val-Tyr-AMC as substrate preincubated for 10 mins followed by subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/10/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Nanjing Forestry University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50163718BDBM50163718(CHEMBL499083)
Affinity DataIC50: 4.37nMAssay Description:Inhibition of chymotrypsin like activity of human 20S proteasome using Suc-Leu-Leu-Val-Tyr-AMC as substrate preincubated for 10 mins followed by subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/10/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Nanjing Forestry University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50163718BDBM50163718(CHEMBL499083)
Affinity DataIC50: 4.40nMAssay Description:Inhibition of chymotrypsin like activity of human 20S proteasome using Suc-Leu-Leu-Val-Tyr-AMC as substrate preincubated for 10 mins followed by subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/10/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Nanjing Forestry University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50163724BDBM50163724(CHEMBL3793107)
Affinity DataIC50: 4.60nMAssay Description:Inhibition of chymotrypsin like activity of human 20S proteasome using Suc-Leu-Leu-Val-Tyr-AMC as substrate preincubated for 10 mins followed by subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/10/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Nanjing Forestry University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50163556BDBM50163556(CHEMBL3794440)
Affinity DataIC50: 4.85nMAssay Description:Inhibition of chymotrypsin like activity of human 20S proteasome using Suc-Leu-Leu-Val-Tyr-AMC as substrate preincubated for 10 mins followed by subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/10/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Nanjing Forestry University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50163556BDBM50163556(CHEMBL3794440)
Affinity DataIC50: 4.90nMAssay Description:Inhibition of chymotrypsin like activity of human 20S proteasome using Suc-Leu-Leu-Val-Tyr-AMC as substrate preincubated for 10 mins followed by subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/10/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Nanjing Forestry University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50163560BDBM50163560(CHEMBL3792730)
Affinity DataIC50: 5.17nMAssay Description:Inhibition of chymotrypsin like activity of human 20S proteasome using Suc-Leu-Leu-Val-Tyr-AMC as substrate preincubated for 10 mins followed by subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/10/2017
Entry Details Article
PubMed
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