Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50047806
TargetHypoxia-inducible factor 1-alpha(Human)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50190657(CHEMBL1194747)
Affinity DataIC50: 730nMAssay Description:Displacement of GST-tagged p300-CH1 domain (323 to 423 residues) from synthetic biotinylated HIF-1alpha C-TAD domain (786 to 826 residues) (unknown o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2018
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50190661(CHEMBL3901938)
Affinity DataIC50: 1.90E+3nMAssay Description:Displacement of GST-tagged p300-CH1 domain (323 to 423 residues) from synthetic biotinylated HIF-1alpha C-TAD domain (786 to 826 residues) (unknown o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2018
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50190659(CHEMBL3912024)
Affinity DataIC50: 2.20E+3nMAssay Description:Displacement of GST-tagged p300-CH1 domain (323 to 423 residues) from synthetic biotinylated HIF-1alpha C-TAD domain (786 to 826 residues) (unknown o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2018
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50190656(CHEMBL3910426)
Affinity DataIC50: 2.40E+3nMAssay Description:Displacement of GST-tagged p300-CH1 domain (323 to 423 residues) from synthetic biotinylated HIF-1alpha C-TAD domain (786 to 826 residues) (unknown o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2018
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50269764(Discorhabdin A | (+)-Discorhabdin B | discorhabdin...)
Affinity DataIC50: 3.70E+3nMAssay Description:Displacement of GST-tagged p300-CH1 domain (323 to 423 residues) from synthetic biotinylated HIF-1alpha C-TAD domain (786 to 826 residues) (unknown o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2018
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50312636(Makaluvamine F | (-)-Makaluvamine F | CHEMBL509890)
Affinity DataIC50: 8.30E+3nMAssay Description:Displacement of GST-tagged p300-CH1 domain (323 to 423 residues) from synthetic biotinylated HIF-1alpha C-TAD domain (786 to 826 residues) (unknown o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2018
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50190660(CHEMBL3920971)
Affinity DataIC50: 3.52E+4nMAssay Description:Displacement of GST-tagged p300-CH1 domain (323 to 423 residues) from synthetic biotinylated HIF-1alpha C-TAD domain (786 to 826 residues) (unknown o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2018
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50190658(CHEMBL3938903)
Affinity DataIC50: 1.00E+5nMAssay Description:Displacement of GST-tagged p300-CH1 domain (323 to 423 residues) from synthetic biotinylated HIF-1alpha C-TAD domain (786 to 826 residues) (unknown o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2018
Entry Details Article
PubMed