Compile Data Set for Download or QSAR
Report error Found 25 Enz. Inhib. hit(s) with all data for entry = 50047442
TargetC-terminal-binding protein 2(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50167976(CHEMBL3799940)
Affinity DataIC50: 170nMAssay Description:Inhibition of recombinant His6-tagged CtBP2 (31 to 384 residues) (unknown origin) dehydrogenase activity expressed in Escherichia coli BL21-Codonplus...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2017
Entry Details Article
PubMed
TargetC-terminal-binding protein 2(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50167975(CHEMBL3798669)
Affinity DataIC50: 180nMAssay Description:Inhibition of recombinant His6-tagged CtBP2 (31 to 384 residues) (unknown origin) dehydrogenase activity expressed in Escherichia coli BL21-Codonplus...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2017
Entry Details Article
PubMed
TargetC-terminal-binding protein 2(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50167967(CHEMBL3797778)
Affinity DataIC50: 240nMAssay Description:Inhibition of recombinant His6-tagged CtBP2 (31 to 384 residues) (unknown origin) dehydrogenase activity expressed in Escherichia coli BL21-Codonplus...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2017
Entry Details Article
PubMed
TargetC-terminal-binding protein 2(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50167980(CHEMBL3800609)
Affinity DataIC50: 300nMAssay Description:Inhibition of recombinant His6-tagged CtBP2 (31 to 384 residues) (unknown origin) dehydrogenase activity expressed in Escherichia coli BL21-Codonplus...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2017
Entry Details Article
PubMed
TargetC-terminal-binding protein 2(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50167969(CHEMBL3800006)
Affinity DataIC50: 320nMAssay Description:Inhibition of recombinant His6-tagged CtBP2 (31 to 384 residues) (unknown origin) dehydrogenase activity expressed in Escherichia coli BL21-Codonplus...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2017
Entry Details Article
PubMed
TargetC-terminal-binding protein 2(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50167970(CHEMBL3800187)
Affinity DataIC50: 480nMAssay Description:Inhibition of recombinant His6-tagged CtBP2 (31 to 384 residues) (unknown origin) dehydrogenase activity expressed in Escherichia coli BL21-Codonplus...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2017
Entry Details Article
PubMed
TargetC-terminal-binding protein 2(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50167979(CHEMBL3799689)
Affinity DataIC50: 720nMAssay Description:Inhibition of recombinant His6-tagged CtBP2 (31 to 384 residues) (unknown origin) dehydrogenase activity expressed in Escherichia coli BL21-Codonplus...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2017
Entry Details Article
PubMed
TargetC-terminal-binding protein 2(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50167973(CHEMBL3799251)
Affinity DataIC50: 880nMAssay Description:Inhibition of recombinant His6-tagged CtBP2 (31 to 384 residues) (unknown origin) dehydrogenase activity expressed in Escherichia coli BL21-Codonplus...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2017
Entry Details Article
PubMed
TargetC-terminal-binding protein 2(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50167981(CHEMBL3797935)
Affinity DataIC50: 900nMAssay Description:Inhibition of recombinant His6-tagged CtBP2 (31 to 384 residues) (unknown origin) dehydrogenase activity expressed in Escherichia coli BL21-Codonplus...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2017
Entry Details Article
PubMed
TargetC-terminal-binding protein 2(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50167972(CHEMBL3800334)
Affinity DataIC50: 2.16E+3nMAssay Description:Inhibition of recombinant His6-tagged CtBP2 (31 to 384 residues) (unknown origin) dehydrogenase activity expressed in Escherichia coli BL21-Codonplus...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2017
Entry Details Article
PubMed
TargetC-terminal-binding protein 2(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50167978(CHEMBL3798743)
Affinity DataIC50: 7.34E+3nMAssay Description:Inhibition of recombinant His6-tagged CtBP2 (31 to 384 residues) (unknown origin) dehydrogenase activity expressed in Escherichia coli BL21-Codonplus...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2017
Entry Details Article
PubMed
TargetC-terminal-binding protein 2(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50167977(CHEMBL3800103)
Affinity DataIC50: 7.65E+3nMAssay Description:Inhibition of recombinant His6-tagged CtBP2 (31 to 384 residues) (unknown origin) dehydrogenase activity expressed in Escherichia coli BL21-Codonplus...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2017
Entry Details Article
PubMed
TargetC-terminal-binding protein 2(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50167971(CHEMBL3800267)
Affinity DataIC50: 8.73E+3nMAssay Description:Inhibition of recombinant His6-tagged CtBP2 (31 to 384 residues) (unknown origin) dehydrogenase activity expressed in Escherichia coli BL21-Codonplus...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2017
Entry Details Article
PubMed
TargetC-terminal-binding protein 2(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50167974(CHEMBL3798092)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant His6-tagged CtBP2 (31 to 384 residues) (unknown origin) dehydrogenase activity expressed in Escherichia coli BL21-Codonplus...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2017
Entry Details Article
PubMed
TargetC-terminal-binding protein 2(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50167651(CHEBI:30851 | Phenylpyruvate)
Affinity DataIC50: 1.16E+5nMAssay Description:Inhibition of recombinant His6-tagged CtBP2 (31 to 384 residues) (unknown origin) dehydrogenase activity expressed in Escherichia coli BL21-Codonplus...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2017
Entry Details Article
PubMed
TargetC-terminal-binding protein 2(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM19473(2-oxopropanoic acid | 2-Oxopropanoate | Pyruvate)
Affinity DataIC50: 3.00E+5nMAssay Description:Inhibition of recombinant His6-tagged CtBP2 (31 to 384 residues) (unknown origin) dehydrogenase activity expressed in Escherichia coli BL21-Codonplus...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2017
Entry Details Article
PubMed
TargetC-terminal-binding protein 2(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50167965(CHEMBL3248231 | US11192850, Compound 1)
Affinity DataIC50: 3.00E+5nMAssay Description:Inhibition of recombinant His6-tagged CtBP2 (31 to 384 residues) (unknown origin) dehydrogenase activity expressed in Escherichia coli BL21-Codonplus...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2017
Entry Details Article
PubMed
TargetC-terminal-binding protein 2(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50167966(CHEMBL3799480)
Affinity DataIC50: 3.00E+5nMAssay Description:Inhibition of recombinant His6-tagged CtBP2 (31 to 384 residues) (unknown origin) dehydrogenase activity expressed in Escherichia coli BL21-Codonplus...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2017
Entry Details Article
PubMed
TargetC-terminal-binding protein 2(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50102174(oxo(phenyl)acetic acid | phenylglyoxylic acid | 2-...)
Affinity DataIC50: 3.00E+5nMAssay Description:Inhibition of recombinant His6-tagged CtBP2 (31 to 384 residues) (unknown origin) dehydrogenase activity expressed in Escherichia coli BL21-Codonplus...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2017
Entry Details Article
PubMed
TargetC-terminal-binding protein 2(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50304072(3-phenylpropanoic acid | HYDROCINNAMIC ACID | Phen...)
Affinity DataIC50: 3.00E+5nMAssay Description:Inhibition of recombinant His6-tagged CtBP2 (31 to 384 residues) (unknown origin) dehydrogenase activity expressed in Escherichia coli BL21-Codonplus...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2017
Entry Details Article
PubMed
TargetC-terminal-binding protein 2(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50167968(CHEMBL3800510)
Affinity DataIC50: 3.00E+5nMAssay Description:Inhibition of recombinant His6-tagged CtBP2 (31 to 384 residues) (unknown origin) dehydrogenase activity expressed in Escherichia coli BL21-Codonplus...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2017
Entry Details Article
PubMed
TargetC-terminal-binding protein 2(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM154571(4-Methylthio 2-oxobutyric acid (MTOB))
Affinity DataIC50: 3.00E+5nMAssay Description:Inhibition of recombinant His6-tagged CtBP2 (31 to 384 residues) (unknown origin) dehydrogenase activity expressed in Escherichia coli BL21-Codonplus...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2017
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetC-terminal-binding protein 2(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50167963(CHEMBL3799698)
Affinity DataIC50: 3.00E+5nMAssay Description:Inhibition of recombinant His6-tagged CtBP2 (31 to 384 residues) (unknown origin) dehydrogenase activity expressed in Escherichia coli BL21-Codonplus...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2017
Entry Details Article
PubMed
TargetC-terminal-binding protein 2(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50167964(CHEMBL3799891)
Affinity DataIC50: 3.00E+5nMAssay Description:Inhibition of recombinant His6-tagged CtBP2 (31 to 384 residues) (unknown origin) dehydrogenase activity expressed in Escherichia coli BL21-Codonplus...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2017
Entry Details Article
PubMed
TargetC-terminal-binding protein 2(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50167962(CHEMBL3798514)
Affinity DataIC50: 3.00E+5nMAssay Description:Inhibition of recombinant His6-tagged CtBP2 (31 to 384 residues) (unknown origin) dehydrogenase activity expressed in Escherichia coli BL21-Codonplus...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2017
Entry Details Article
PubMed