Compile Data Set for Download or QSAR
Report error Found 31 Enz. Inhib. hit(s) with all data for entry = 50047849
TargetEpidermal growth factor receptor(Human)
Norwegian University of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50193159BDBM50193159(CHEMBL3901622)
Affinity DataIC50: 0.400nMAssay Description:Inhibition of recombinant human GST-tagged EGFR cytoplasmic domain (668 to 1210 residues) expressed in baculovirus by Z'-LYTE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2018
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Norwegian University of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 5446BDBM5446(Erlotinib | OSI-774 | N-(3-ethynylphenyl)-6,7-bis(...)
Affinity DataIC50: 0.400nMAssay Description:Inhibition of recombinant human GST-tagged EGFR cytoplasmic domain (668 to 1210 residues) expressed in baculovirus by Z'-LYTE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2018
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEpidermal growth factor receptor(Human)
Norwegian University of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50193146BDBM50193146(CHEMBL3891846)
Affinity DataIC50: 0.600nMAssay Description:Inhibition of recombinant human GST-tagged EGFR cytoplasmic domain (668 to 1210 residues) expressed in baculovirus by Z'-LYTE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2018
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Norwegian University of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50193144BDBM50193144(CHEMBL3960853)
Affinity DataIC50: 1.10nMAssay Description:Inhibition of recombinant human GST-tagged EGFR cytoplasmic domain (668 to 1210 residues) expressed in baculovirus by Z'-LYTE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2018
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Norwegian University of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50193245BDBM50193245(CHEMBL3919609)
Affinity DataIC50: 1.5nMAssay Description:Inhibition of recombinant human GST-tagged EGFR cytoplasmic domain (668 to 1210 residues) expressed in baculovirus by Z'-LYTE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2018
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Norwegian University of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50193165BDBM50193165(CHEMBL3928512)
Affinity DataIC50: 2nMAssay Description:Inhibition of recombinant human GST-tagged EGFR cytoplasmic domain (668 to 1210 residues) expressed in baculovirus by Z'-LYTE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2018
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Norwegian University of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50193169BDBM50193169(CHEMBL3961553)
Affinity DataIC50: 2nMAssay Description:Inhibition of recombinant human GST-tagged EGFR cytoplasmic domain (668 to 1210 residues) expressed in baculovirus by Z'-LYTE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2018
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Norwegian University of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50193247BDBM50193247(CHEMBL3952157)
Affinity DataIC50: 2.70nMAssay Description:Inhibition of recombinant human GST-tagged EGFR cytoplasmic domain (668 to 1210 residues) expressed in baculovirus by Z'-LYTE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2018
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Norwegian University of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50193147BDBM50193147(CHEMBL3892567)
Affinity DataIC50: 3.90nMAssay Description:Inhibition of recombinant human GST-tagged EGFR cytoplasmic domain (668 to 1210 residues) expressed in baculovirus by Z'-LYTE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2018
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Norwegian University of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50193160BDBM50193160(CHEMBL3947406)
Affinity DataIC50: 4nMAssay Description:Inhibition of recombinant human GST-tagged EGFR cytoplasmic domain (668 to 1210 residues) expressed in baculovirus by Z'-LYTE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2018
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Norwegian University of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50193143BDBM50193143(CHEMBL3961961)
Affinity DataIC50: 4nMAssay Description:Inhibition of recombinant human GST-tagged EGFR cytoplasmic domain (668 to 1210 residues) expressed in baculovirus by Z'-LYTE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2018
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Norwegian University of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50193168BDBM50193168(CHEMBL3956112)
Affinity DataIC50: 4.60nMAssay Description:Inhibition of recombinant human GST-tagged EGFR cytoplasmic domain (668 to 1210 residues) expressed in baculovirus by Z'-LYTE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2018
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Norwegian University of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50193163BDBM50193163(CHEMBL3933539)
Affinity DataIC50: 5.30nMAssay Description:Inhibition of recombinant human GST-tagged EGFR cytoplasmic domain (668 to 1210 residues) expressed in baculovirus by Z'-LYTE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2018
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Norwegian University of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50193140BDBM50193140(CHEMBL3946396)
Affinity DataIC50: 7nMAssay Description:Inhibition of recombinant human GST-tagged EGFR cytoplasmic domain (668 to 1210 residues) expressed in baculovirus by Z'-LYTE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2018
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Norwegian University of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50193162BDBM50193162(CHEMBL3908303)
Affinity DataIC50: 11nMAssay Description:Inhibition of recombinant human GST-tagged EGFR cytoplasmic domain (668 to 1210 residues) expressed in baculovirus by Z'-LYTE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2018
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Norwegian University of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50193246BDBM50193246(CHEMBL3967219)
Affinity DataIC50: 13nMAssay Description:Inhibition of recombinant human GST-tagged EGFR cytoplasmic domain (668 to 1210 residues) expressed in baculovirus by Z'-LYTE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2018
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Norwegian University of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50193158BDBM50193158(CHEMBL3943438)
Affinity DataIC50: 14nMAssay Description:Inhibition of recombinant human GST-tagged EGFR cytoplasmic domain (668 to 1210 residues) expressed in baculovirus by Z'-LYTE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2018
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Norwegian University of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50193157BDBM50193157(CHEMBL3934461)
Affinity DataIC50: 22nMAssay Description:Inhibition of recombinant human GST-tagged EGFR cytoplasmic domain (668 to 1210 residues) expressed in baculovirus by Z'-LYTE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2018
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Norwegian University of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50193186BDBM50193186(CHEMBL3972981)
Affinity DataIC50: 22nMAssay Description:Inhibition of recombinant human GST-tagged EGFR cytoplasmic domain (668 to 1210 residues) expressed in baculovirus by Z'-LYTE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2018
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Norwegian University of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50193142BDBM50193142(CHEMBL3953210)
Affinity DataIC50: 24nMAssay Description:Inhibition of recombinant human GST-tagged EGFR cytoplasmic domain (668 to 1210 residues) expressed in baculovirus by Z'-LYTE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2018
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Norwegian University of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50193156BDBM50193156(CHEMBL3925584)
Affinity DataIC50: 24nMAssay Description:Inhibition of recombinant human GST-tagged EGFR cytoplasmic domain (668 to 1210 residues) expressed in baculovirus by Z'-LYTE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2018
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Norwegian University of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50193170BDBM50193170(CHEMBL3973601)
Affinity DataIC50: 27nMAssay Description:Inhibition of recombinant human GST-tagged EGFR cytoplasmic domain (668 to 1210 residues) expressed in baculovirus by Z'-LYTE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2018
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Norwegian University of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50193248BDBM50193248(CHEMBL3952877)
Affinity DataIC50: 28nMAssay Description:Inhibition of recombinant human GST-tagged EGFR cytoplasmic domain (668 to 1210 residues) expressed in baculovirus by Z'-LYTE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2018
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Norwegian University of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50193166BDBM50193166(CHEMBL3929584)
Affinity DataIC50: 29nMAssay Description:Inhibition of recombinant human GST-tagged EGFR cytoplasmic domain (668 to 1210 residues) expressed in baculovirus by Z'-LYTE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2018
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Norwegian University of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50193167BDBM50193167(CHEMBL3975699)
Affinity DataIC50: 44nMAssay Description:Inhibition of recombinant human GST-tagged EGFR cytoplasmic domain (668 to 1210 residues) expressed in baculovirus by Z'-LYTE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2018
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Norwegian University of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50193161BDBM50193161(CHEMBL3937527)
Affinity DataIC50: 56nMAssay Description:Inhibition of recombinant human GST-tagged EGFR cytoplasmic domain (668 to 1210 residues) expressed in baculovirus by Z'-LYTE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2018
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Norwegian University of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50193139BDBM50193139(CHEMBL3939429)
Affinity DataIC50: 74nMAssay Description:Inhibition of recombinant human GST-tagged EGFR cytoplasmic domain (668 to 1210 residues) expressed in baculovirus by Z'-LYTE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2018
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Norwegian University of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50193141BDBM50193141(CHEMBL3981621)
Affinity DataIC50: 93nMAssay Description:Inhibition of recombinant human GST-tagged EGFR cytoplasmic domain (668 to 1210 residues) expressed in baculovirus by Z'-LYTE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2018
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Norwegian University of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50193164BDBM50193164(CHEMBL3962640)
Affinity DataIC50: 100nMAssay Description:Inhibition of recombinant human GST-tagged EGFR cytoplasmic domain (668 to 1210 residues) expressed in baculovirus by Z'-LYTE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2018
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Norwegian University of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50193155BDBM50193155(CHEMBL3944121)
Affinity DataIC50: 100nMAssay Description:Inhibition of recombinant human GST-tagged EGFR cytoplasmic domain (668 to 1210 residues) expressed in baculovirus by Z'-LYTE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2018
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Norwegian University of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50193148BDBM50193148(CHEMBL3935149)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of recombinant human GST-tagged EGFR cytoplasmic domain (668 to 1210 residues) expressed in baculovirus by Z'-LYTE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2018
Entry Details Article
PubMed